7FH0
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4EI4
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![BU of 4ei4 by Molmil](/molmil-images/mine/4ei4) | JAK1 kinase (JH1 domain) in complex with compound 20 | 分子名称: | (1R,3R)-3-(2-methylimidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(8H)-yl)cyclohexanol, Tyrosine-protein kinase JAK1 | 著者 | Eigenbrot, C, Steffek, M. | 登録日 | 2012-04-04 | 公開日 | 2012-07-04 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Discovery and optimization of C-2 methyl imidazopyrrolopyridines as potent and orally bioavailable JAK1 inhibitors with selectivity over JAK2. J.Med.Chem., 55, 2012
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4EHZ
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![BU of 4ehz by Molmil](/molmil-images/mine/4ehz) | The Jak1 kinase domain in complex with inhibitor | 分子名称: | 1,2-ETHANEDIOL, 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine, Tyrosine-protein kinase JAK1 | 著者 | Lupardus, P.J, Steffek, M. | 登録日 | 2012-04-04 | 公開日 | 2012-07-04 | 最終更新日 | 2013-01-23 | 実験手法 | X-RAY DIFFRACTION (2.174 Å) | 主引用文献 | Discovery and optimization of C-2 methyl imidazopyrrolopyridines as potent and orally bioavailable JAK1 inhibitors with selectivity over JAK2. J.Med.Chem., 55, 2012
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4F09
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4F08
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5ZGM
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![BU of 5zgm by Molmil](/molmil-images/mine/5zgm) | Crystal Structure of Parvalbumin SPVI, the Major Allergens in Mustelus griseus | 分子名称: | CALCIUM ION, Parvalbumin SPVI, SULFATE ION | 著者 | Yang, R.Q, Chen, Y.L, Jin, T.C, Cao, M.J. | 登録日 | 2018-03-09 | 公開日 | 2018-08-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.399 Å) | 主引用文献 | Purification, Characterization, and Crystal Structure of Parvalbumins, the Major Allergens in Mustelus griseus. J. Agric. Food Chem., 66, 2018
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6AG0
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![BU of 6ag0 by Molmil](/molmil-images/mine/6ag0) | The X-ray Crystallographic Structure of Maltooligosaccharide-forming Amylase from Bacillus stearothermophilus STB04 | 分子名称: | 4,6-dideoxy-4-{[(1S,4R,5S,6S)-4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, Alpha-amylase, CALCIUM ION | 著者 | Li, Z.F, Li, Y.L, Ban, X.F, Zhang, C.Y, Jin, T.C, Xie, X.F, Gu, Z.B, Li, C.M. | 登録日 | 2018-08-09 | 公開日 | 2018-10-10 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structure of a maltooligosaccharide-forming amylase from Bacillus stearothermophilus STB04. Int.J.Biol.Macromol., 138, 2019
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5ZH6
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![BU of 5zh6 by Molmil](/molmil-images/mine/5zh6) | Crystal structure of Parvalbumin SPV-II of Mustelus griseus | 分子名称: | CALCIUM ION, Parvalbumin SPV-II, SULFATE ION | 著者 | Yang, R.Q, Chen, Y.L, Jin, T.C, Cao, M.J. | 登録日 | 2018-03-11 | 公開日 | 2018-08-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Purification, Characterization, and Crystal Structure of Parvalbumins, the Major Allergens in Mustelus griseus. J. Agric. Food Chem., 66, 2018
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5ZHQ
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6JLC
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6JQB
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![BU of 6jqb by Molmil](/molmil-images/mine/6jqb) | The structure of maltooligosaccharide-forming amylase from Pseudomonas saccharophila STB07 with pseudo-maltoheptaose | 分子名称: | 1,2-ETHANEDIOL, ACARBOSE DERIVED HEPTASACCHARIDE, CALCIUM ION, ... | 著者 | Li, Z.F, Ban, X.F, Zhang, Z.Q, Li, C.M, Gu, Z.B, Jin, T.C, Li, Y.L, Shang, Y.H. | 登録日 | 2019-03-30 | 公開日 | 2020-04-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.101 Å) | 主引用文献 | Structure of maltotetraose-forming amylase from Pseudomonas saccharophila STB07 provides insights into its product specificity. Int.J.Biol.Macromol., 154, 2020
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6KI0
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![BU of 6ki0 by Molmil](/molmil-images/mine/6ki0) | Crystal Structure of Human ASC-CARD | 分子名称: | Maltose/maltodextrin-binding periplasmic protein,Apoptosis-associated speck-like protein containing a CARD, SULFATE ION, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Xu, Z.H, Jin, T.C. | 登録日 | 2019-07-16 | 公開日 | 2020-07-22 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Homotypic CARD-CARD interaction is critical for the activation of NLRP1 inflammasome. Cell Death Dis, 12, 2021
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6KXG
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7X4I
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2KP1
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2KP2
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6X5A
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![BU of 6x5a by Molmil](/molmil-images/mine/6x5a) | The mouse cGAS catalytic domain binding to human nucleosome that purified from HEK293T cells | 分子名称: | Cyclic GMP-AMP synthase, DNA (natural), Histone H2A type 1, ... | 著者 | Pengbiao, X, Pingwei, L, Baoyu, Z. | 登録日 | 2020-05-25 | 公開日 | 2020-09-16 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (4.36 Å) | 主引用文献 | The molecular basis of tight nuclear tethering and inactivation of cGAS. Nature, 587, 2020
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6X59
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![BU of 6x59 by Molmil](/molmil-images/mine/6x59) | The mouse cGAS catalytic domain binding to human assembled nucleosome | 分子名称: | Cyclic GMP-AMP synthase, DNA, Histone H2A type 1, ... | 著者 | Pengbiao, X, Pingwei, L, Baoyu, Z. | 登録日 | 2020-05-25 | 公開日 | 2020-09-16 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (2.98 Å) | 主引用文献 | The molecular basis of tight nuclear tethering and inactivation of cGAS. Nature, 587, 2020
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6XJD
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![BU of 6xjd by Molmil](/molmil-images/mine/6xjd) | Two mouse cGAS catalytic domain binding to human assembled nucleosome | 分子名称: | Cyclic GMP-AMP synthase, DNA (145-MER), Histone H2A type 1, ... | 著者 | Xu, P, Li, P, Zhao, B. | 登録日 | 2020-06-23 | 公開日 | 2020-09-16 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (6.8 Å) | 主引用文献 | The molecular basis of tight nuclear tethering and inactivation of cGAS. Nature, 587, 2020
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4NKG
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![BU of 4nkg by Molmil](/molmil-images/mine/4nkg) | Crystal structure of SspH1 LRR domain in complex PKN1 HR1b domain | 分子名称: | E3 ubiquitin-protein ligase sspH1, HEXANE-1,6-DIOL, Serine/threonine-protein kinase N1 | 著者 | Keszei, A.F.A, Xiaojing, T, Mccormick, C, Zeqiraj, E, Rohde, J.R, Tyers, M, Sicheri, F. | 登録日 | 2013-11-12 | 公開日 | 2013-12-11 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structure of an SspH1-PKN1 Complex Reveals the Basis for Host Substrate Recognition and Mechanism of Activation for a Bacterial E3 Ubiquitin Ligase. Mol.Cell.Biol., 34, 2014
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4NKH
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![BU of 4nkh by Molmil](/molmil-images/mine/4nkh) | Crystal structure of SspH1 LRR domain | 分子名称: | E3 ubiquitin-protein ligase sspH1 | 著者 | Keszei, A.F.A, Xiaojing, T, Mccormick, C, Zeqiraj, E, Rohde, J.R, Tyers, M, Sicheri, F. | 登録日 | 2013-11-12 | 公開日 | 2013-12-11 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Structure of an SspH1-PKN1 Complex Reveals the Basis for Host Substrate Recognition and Mechanism of Activation for a Bacterial E3 Ubiquitin Ligase. Mol.Cell.Biol., 34, 2014
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2DJJ
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6LOX
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![BU of 6lox by Molmil](/molmil-images/mine/6lox) | Crystal Structure of human glutaminase with macrocyclic inhibitor | 分子名称: | (E)-15,22-Dioxa-4,11-diaza-5(2,5)-thiadiazola-10(3,6)-pyridazina-1,14(1,3)-dibenzenacyclodocosaphan-18-ene-3,12-dione, Glutaminase kidney isoform, mitochondrial | 著者 | Bian, J, Li, Z, Xu, X, Wang, J, Li, L. | 登録日 | 2020-01-07 | 公開日 | 2021-01-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structure-Enabled Discovery of Novel Macrocyclic Inhibitors Targeting Glutaminase 1 Allosteric Binding Site. J.Med.Chem., 64, 2021
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2DJK
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