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6RVX
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BU of 6rvx by Molmil
Inward-open structure of the ASCT2 (SLC1A5) mutant C467R in presence of TBOA
分子名称: Neutral amino acid transporter B(0)
著者Garaeva, A.A, Guskov, A, Slotboom, D.J, Paulino, C.
登録日2019-06-03
公開日2019-08-07
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (3.61 Å)
主引用文献A one-gate elevator mechanism for the human neutral amino acid transporter ASCT2.
Nat Commun, 10, 2019
4QTN
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BU of 4qtn by Molmil
Crystal structure of the Vitamin B3 transporter PnuC
分子名称: Nicotinamide riboside, Nicotinamide riboside transporter PnuC, octyl beta-D-glucopyranoside
著者Guskov, A, Jaehme, M, Slotboom, D.J.
登録日2014-07-08
公開日2014-10-08
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the Vitamin B3 transporter PnuC
Nat.Struct.Mol.Biol., 2014
4DVE
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BU of 4dve by Molmil
Crystal structure at 2.1 A of the S-component for biotin from an ECF-type ABC transporter
分子名称: BIOTIN, Biotin transporter BioY, nonyl beta-D-glucopyranoside
著者Berntsson, R.P.-A, ter Beek, J, Majsnerowska, M, Duurkens, R, Puri, P, Poolman, B, Slotboom, D.J.
登録日2012-02-23
公開日2012-08-29
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Structural divergence of paralogous S components from ECF-type ABC transporters.
Proc.Natl.Acad.Sci.USA, 109, 2012
4C1T
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BU of 4c1t by Molmil
Structure of the xylo-oligosaccharide specific solute binding protein from Bifidobacterium animalis subsp. lactis Bl-04 in complex with arabinoxylotriose
分子名称: PENTAETHYLENE GLYCOL, SUGAR TRANSPORTER SOLUTE-BINDING PROTEIN, alpha-L-arabinofuranose-(1-2)-beta-D-xylopyranose-(1-4)-beta-D-xylopyranose-(1-4)-beta-D-xylopyranose
著者Fredslund, F, Ejby, M, Vujicic-Zagar, A, Svensson, B, Slotboom, D.J, Abou Hachem, M.
登録日2013-08-13
公開日2013-10-30
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Structural Basis for Arabinoxylo-Oligosaccharide Capture by the Probiotic Bifidobacterium Animalis Subsp. Lactis Bl-04
Mol.Microbiol., 90, 2013
6RVY
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BU of 6rvy by Molmil
Inward-open structure of the ASCT2 (SLC1A5) mutant C467R in absence of substrate
分子名称: Neutral amino acid transporter B(0)
著者Garaeva, A.A, Guskov, A, Slotboom, D.J, Paulino, C.
登録日2019-06-03
公開日2019-08-07
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (4.13 Å)
主引用文献A one-gate elevator mechanism for the human neutral amino acid transporter ASCT2.
Nat Commun, 10, 2019
4POP
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BU of 4pop by Molmil
ThiT with LMG139 bound
分子名称: 2-(2-METHOXYETHOXY)ETHANOL, 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, 4-[(4-amino-2-methylpyrimidin-5-yl)methyl]-3-methylthiophene-2-carbaldehyde, ...
著者Swier, L.J.Y.M, Guskov, A, Slotboom, D.J.
登録日2014-02-26
公開日2014-09-17
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure-Based Design of Potent Small-Molecule Binders to the S-Component of the ECF Transporter for Thiamine.
Chembiochem, 16, 2015
4POV
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BU of 4pov by Molmil
ThiT with LMG135 bound
分子名称: 2-(2-METHOXYETHOXY)ETHANOL, 4-[(4-amino-2-methylpyrimidin-5-yl)methyl]-3-methylthiophene-2-carbaldehyde, CHLORIDE ION, ...
著者Swier, L.J.Y.M, Guskov, A, Slotboom, D.J.
登録日2014-02-26
公開日2014-09-17
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure-Based Design of Potent Small-Molecule Binders to the S-Component of the ECF Transporter for Thiamine.
Chembiochem, 16, 2015
4FAJ
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BU of 4faj by Molmil
Structure and mode of peptide binding of pheromone receptor PrgZ
分子名称: GLYCEROL, PrgZ, Sex pheromone cCF10, ...
著者Berntsson, R.P.-A, Schuurman-Wolters, G.K, Dunny, K, Slotboom, D.J, Poolman, B.
登録日2012-05-22
公開日2012-09-12
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure and Mode of Peptide Binding of Pheromone Receptor PrgZ.
J.Biol.Chem., 287, 2012
4G4P
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BU of 4g4p by Molmil
Crystal structure of glutamine-binding protein from Enterococcus faecalis at 1.5 A
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Amino acid ABC transporter, amino acid-binding/permease protein, ...
著者Fulyani, F, Guskov, A, Zagar, A.V, Slotboom, D.-J, Poolman, B.
登録日2012-07-16
公開日2013-07-17
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Functional Diversity of Tandem Substrate-Binding Domains in ABC Transporters from Pathogenic Bacteria.
Structure, 21, 2013
3RYA
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BU of 3rya by Molmil
Lactococcal OppA complexed with SLSQLSSQS
分子名称: Oligopeptide, Oligopeptide-binding protein oppA
著者Berntsson, R.P.-A, Thunnissen, A.-M.W.H, Poolman, B, Slotboom, D.-J.
登録日2011-05-11
公開日2011-06-29
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Importance of a Hydrophobic Pocket for Peptide Binding in Lactococcal OppA.
J.Bacteriol., 193, 2011
3RYB
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BU of 3ryb by Molmil
Lactococcal OppA complexed with SLSQSLSQS
分子名称: Oligopeptide, Oligopeptide-binding protein oppA
著者Berntsson, R.P.-A, Thunnissen, A.-M.W.H, Poolman, B, Slotboom, D.-J.
登録日2011-05-11
公開日2011-06-29
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Importance of a Hydrophobic Pocket for Peptide Binding in Lactococcal OppA.
J.Bacteriol., 193, 2011
6SGF
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BU of 6sgf by Molmil
Molecular insight into a new low affinity xylan binding module CBM86, from the xylanolytic gut symbiont Roseburia intestinalis.
分子名称: Beta-xylanase, CADMIUM ION, CHLORIDE ION, ...
著者Ejby, M, Abou Hachem, M, Leth, M.L, Guskov, A, Slotboom, D.
登録日2019-08-04
公開日2019-11-20
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.756 Å)
主引用文献Molecular insight into a new low-affinity xylan binding module from the xylanolytic gut symbiont Roseburia intestinalis.
Febs J., 287, 2020
8AFA
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BU of 8afa by Molmil
Cryo-EM structure of a substrate-bound glutamate transporter homologue GltTk encapsulated within a nanodisc
分子名称: ASPARTIC ACID, Proton/glutamate symporter, SDF family
著者Whittaker, J.J, Guskov, A.
登録日2022-07-16
公開日2023-04-05
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.25 Å)
主引用文献Mutation in glutamate transporter homologue GltTk provides insights into pathologic mechanism of episodic ataxia 6.
Nat Commun, 14, 2023
3FTO
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BU of 3fto by Molmil
Crystal structure of OppA in a open conformation
分子名称: Oligopeptide-binding protein oppA
著者Berntsson, R.P.-A, Oktaviani, N.A, Fusetti, F, Thunnissen, A.-M.W.H, Poolman, B, Slotboom, D.-J.
登録日2009-01-13
公開日2009-03-31
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Selenomethionine incorporation in proteins expressed in Lactococcus lactis.
Protein Sci., 18, 2009
7Q10
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BU of 7q10 by Molmil
Acetyltrasferase(3) type IIIa in complex with 3-N-methyl-nemycin B
分子名称: 3N methyl nemycin B, ACETATE ION, Aminoglycoside N(3)-acetyltransferase III, ...
著者Pontillo, N, Guskov, A.
登録日2021-10-17
公開日2022-11-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献3-N-alkylation in aminoglycoside antibiotic neomycin B overcomes bacterial resistance mediated by acetyltransferase (3) IIIa
To Be Published
7Q1D
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BU of 7q1d by Molmil
Acetyltrasferase(3) type IIIa in complex with 3-N-methyl-nemycin B
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Aminoglycoside N(3)-acetyltransferase III, CHLORIDE ION, ...
著者Pontillo, N, Guskov, A.
登録日2021-10-18
公開日2022-11-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.43 Å)
主引用文献3-N-alkylation in aminoglycoside antibiotic neomycin B overcomes bacterial resistance mediated by acetyltransferase (3) IIIa
To Be Published
7Q0Q
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BU of 7q0q by Molmil
Acetyltrasferase(3) type IIIa in complex with 3-N-methyl-nemycin B
分子名称: 3N methyl nemycin B, ACETATE ION, Aminoglycoside N(3)-acetyltransferase III, ...
著者Pontillo, N, Guskov, A.
登録日2021-10-16
公開日2022-11-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献The 3-N-alkylation of the neomycin B outmaneuvers the aminoglycoside resistant enzyme acetyltransferase(3)IIIa via an unexpected mechanism
To Be Published
7Q1X
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BU of 7q1x by Molmil
Acetyltrasferase(3) type IIIa in complex with neomycin B
分子名称: Aminoglycoside N(3)-acetyltransferase III, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Pontillo, N, Guskov, A.
登録日2021-10-21
公開日2022-11-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献The 3-N-alkylation of the neomycin B outmaneuvers the aminoglycoside resistant enzyme acetyltransferase(3)IIIa via an unexpected mechanism
To Be Published
8PUJ
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BU of 8puj by Molmil
The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
分子名称: COB(II)INAMIDE, HYDROXIDE ION, SODIUM ION, ...
著者Whittaker, J, Martinez-Felices, J.M, Guskov, A, Slotboom, D.J.
登録日2023-07-17
公開日2024-07-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The surface-exposed lipo-protein of BtuG3 in complex with cyanocobinamide.
To Be Published
8PTD
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BU of 8ptd by Molmil
The surface-exposed lipo-protein of BtuG1 in complex with cyanocobalamin.
分子名称: COBALAMIN, GLYCEROL, HYDROXIDE ION, ...
著者Whittaker, J, Felices Martinez, J.M, Guskov, A, Slotboom, D.J.
登録日2023-07-14
公開日2024-07-24
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The surface-exposed lipo-protein of BtuG1 in complex with cyanocobalamin.
To Be Published
8PTF
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BU of 8ptf by Molmil
The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
分子名称: COB(II)INAMIDE, SODIUM ION, YncE family protein, ...
著者Whittaker, J, Felices Martinez, J.M, Guskov, A, Slotboom, D.J.
登録日2023-07-14
公開日2024-07-24
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The surface-exposed lipo-protein of BtuG1 in complex with cyanocobinamide.
To Be Published
8BAI
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BU of 8bai by Molmil
The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
分子名称: CYANOCOBALAMIN, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
著者Whittaker, J, Martinez Felices, J.M, Guskov, A, Slotboom, D.J.
登録日2022-10-11
公開日2023-10-25
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
To Be Published
8BAZ
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BU of 8baz by Molmil
The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
分子名称: COB(II)INAMIDE, CYANIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Whittaker, J, Martinez-Felices, J.M, Guskov, A, Slotboom, D.J.
登録日2022-10-12
公開日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The surface-exposed lipo-protein of BtuG2 in complex with cyanocobinamide.
To Be Published
8BB0
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BU of 8bb0 by Molmil
The surface-exposed lipo-protein of BtuG2 in complex with hydroxycobalamin.
分子名称: ACETATE ION, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
著者Whittaker, J, Felices Martinez, J.M, Guskov, A, Slotboom, D.J.
登録日2022-10-12
公開日2023-10-25
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The surface-exposed lipo-protein of BtuG2 in complex with hydroxycobinamide.
To Be Published
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