8GER
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![BU of 8ger by Molmil](/molmil-images/mine/8ger) | |
1NRL
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![BU of 1nrl by Molmil](/molmil-images/mine/1nrl) | Crystal Structure of the human PXR-LBD in complex with an SRC-1 coactivator peptide and SR12813 | 分子名称: | Nuclear Receptor Coactivator 1 isoform 3, Orphan nuclear receptor PXR, [2-(3,5-DI-TERT-BUTYL-4-HYDROXY-PHENYL)-1-(DIETHOXY-PHOSPHORYL)-VINYL]-PHOSPHONIC ACID DIETHLYL ESTER | 著者 | Watkins, R.E, Davis-Searles, P.R, Lambert, M.H, Redinbo, M.R. | 登録日 | 2003-01-25 | 公開日 | 2003-08-19 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Coactivator binding promotes the specific interaction between ligand and the pregnane X receptor J.Mol.Biol., 331, 2003
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1MX1
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![BU of 1mx1 by Molmil](/molmil-images/mine/1mx1) | Crystal Structure of Human Liver Carboxylesterase in complex with tacrine | 分子名称: | 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, N-acetyl-alpha-neuraminic acid, ... | 著者 | Bencharit, S, Morton, C.L, Hyatt, J.L, Kuhn, P, Danks, M.K, Potter, P.M, Redinbo, M.R. | 登録日 | 2002-10-01 | 公開日 | 2003-04-22 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal Structure of Human Carboxylesterase 1 Complexed with the Alzheimer's
Drug Tacrine: From Binding Promiscuity to Selective Inhibition CHEM.BIOL., 10, 2003
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8DTQ
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![BU of 8dtq by Molmil](/molmil-images/mine/8dtq) | Crystal Structure of Staphylococcus aureus pSK41 Cop | 分子名称: | CHLORIDE ION, Helix-turn-helix domain, SODIUM ION | 著者 | Walton, W.G, Eakes, T.C, Redinbo, M.R, McLaughlin, K.J. | 登録日 | 2022-07-26 | 公開日 | 2023-08-02 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | pSK41/pGO1-family conjugative plasmids of Staphylococcus aureus encode a cryptic repressor of replication. Plasmid, 128, 2023
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1RRJ
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![BU of 1rrj by Molmil](/molmil-images/mine/1rrj) | Structural Mechanisms of Camptothecin Resistance by Mutations in Human Topoisomerase I | 分子名称: | (S)-10-[(DIMETHYLAMINO)METHYL]-4-ETHYL-4,9-DIHYDROXY-1H-PYRANO[3',4':6,7]INOLIZINO[1,2-B]-QUINOLINE-3,14(4H,12H)-DIONE, 2-(1-DIMETHYLAMINOMETHYL-2-HYDROXY-8-HYDROXYMETHYL-9-OXO-9,11-DIHYDRO-INDOLIZINO[1,2-B]QUINOLIN-7-YL)-2-HYDROXY-BUTYRIC ACID, 5'-D(*AP*AP*AP*AP*AP*GP*AP*CP*TP*T*GP*GP*AP*AP*AP*AP*AP*TP*TP*TP*TP*T)-3', ... | 著者 | Chrencik, J.E, Staker, B.L, Burgin, A.B, Stewart, L, Redinbo, M.R. | 登録日 | 2003-12-08 | 公開日 | 2004-07-06 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Mechanisms of camptothecin resistance by human topoisomerase I mutations J.Mol.Biol., 339, 2004
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1YUC
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![BU of 1yuc by Molmil](/molmil-images/mine/1yuc) | Human Nuclear Receptor Liver Receptor Homologue-1, LRH-1, Bound to Phospholipid and a Fragment of Human SHP | 分子名称: | GLYCEROL, L-ALPHA-PHOSPHATIDYL-BETA-OLEOYL-GAMMA-PALMITOYL-PHOSPHATIDYLETHANOLAMINE, Nuclear receptor 0B2, ... | 著者 | Ortlund, E.A, Yoonkwang, L, Solomon, I.H, Hager, J.M, Safi, R, Choi, Y, Guan, Z, Tripathy, A, Raetz, C.R.H, McDonnell, D.P, Moore, D.D, Redinbo, M.R. | 登録日 | 2005-02-13 | 公開日 | 2005-03-01 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Modulation of human nuclear receptor LRH-1 activity by phospholipids and SHP Nat.Struct.Mol.Biol., 12, 2005
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1A36
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![BU of 1a36 by Molmil](/molmil-images/mine/1a36) | TOPOISOMERASE I/DNA COMPLEX | 分子名称: | DNA (5'-D(*AP*AP*AP*AP*AP*GP*AP*CP*TP*TP*AP*GP*AP*AP*AP*AP*A P*TP*TP*TP*TP*T)- 3'), DNA (5'-D(*AP*AP*AP*AP*AP*TP*TP*TP*TP*TP*CP*TP*AP*AP*GP*TP*C P*TP*TP*TP*TP*T)- 3'), TOPOISOMERASE I | 著者 | Stewart, L, Redinbo, M.R, Qiu, X, Champoux, J.J, Hol, W.G.J. | 登録日 | 1998-01-29 | 公開日 | 1998-08-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | A model for the mechanism of human topoisomerase I. Science, 279, 1998
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1YA8
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![BU of 1ya8 by Molmil](/molmil-images/mine/1ya8) | Crystal Structure of Human Liver Carboxylesterase in complex with cleavage products of Mevastatin | 分子名称: | (1S,7S,8S,8AR)-1,2,3,7,8,8A-HEXAHYDRO-7-METHYL-8-[2-[(2R,4R)-TETRAHYDRO-4-HY DROXY-6-OXO-2H-PYRAN-2-YL]ETHYL]-1-NAPHTHALENOL, 2-METHYLBUTANOIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Fleming, C.D, Bencharit, S, Edwards, C.C, Hyatt, J.L, Morton, C.L, Howard-Williams, E.L, Potter, P.M, Redinbo, M.R. | 登録日 | 2004-12-17 | 公開日 | 2005-08-02 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural insights into drug processing by human carboxylesterase 1: tamoxifen, mevastatin, and inhibition by benzil. J.Mol.Biol., 352, 2005
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1YAJ
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![BU of 1yaj by Molmil](/molmil-images/mine/1yaj) | Crystal Structure of Human Liver Carboxylesterase in complex with benzil | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BENZOIC ACID, CES1 protein, ... | 著者 | Fleming, C.D, Bencharit, S, Edwards, C.C, Hyatt, J.L, Morton, C.M, Howard-Williams, E.L, Potter, P.M, Redinbo, M.R. | 登録日 | 2004-12-17 | 公開日 | 2005-08-02 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structural insights into drug processing by human carboxylesterase 1: tamoxifen, mevastatin, and inhibition by benzil. J.Mol.Biol., 352, 2005
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1YA4
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![BU of 1ya4 by Molmil](/molmil-images/mine/1ya4) | Crystal Structure of Human Liver Carboxylesterase 1 in complex with tamoxifen | 分子名称: | (Z)-2-[4-(1,2)-DIPHENYL-1-BUTENYL)-PHENOXY]-N,N-DIMETHYLETHANAMINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CES1 protein, ... | 著者 | Fleming, C.D, Bencharit, S, Edwards, C.C, Hyatt, J.L, Morton, C.L, Howard-Williams, E.L, Potter, P.M, Redinbo, M.R. | 登録日 | 2004-12-17 | 公開日 | 2005-08-02 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structural insights into drug processing by human carboxylesterase 1: tamoxifen, mevastatin, and inhibition by benzil. J.Mol.Biol., 352, 2005
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4EQX
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![BU of 4eqx by Molmil](/molmil-images/mine/4eqx) | Crystal Structure of the C43S Mutant of Staphylococcus aureus CoADR | 分子名称: | CHLORIDE ION, Coenzyme A disulfide reductase, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Edwards, J.S, Wallace, B.D, Wallen, J.R, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-19 | 公開日 | 2012-10-17 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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1YAH
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![BU of 1yah by Molmil](/molmil-images/mine/1yah) | Crystal Structure of Human Liver Carboxylesterase complexed to Etyl Acetate; A Fatty Acid Ethyl Ester Analogue | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CES1 protein, ETHYL ACETATE, ... | 著者 | Fleming, C.D, Bencahrit, S, Edwards, C.C, Hyatt, J.L, Morton, C.L, Howard-Williams, E.L, Potter, P.M, Redinbo, M.R. | 登録日 | 2004-12-17 | 公開日 | 2005-08-02 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural insights into drug processing by human carboxylesterase 1: tamoxifen, mevastatin, and inhibition by benzil. J.Mol.Biol., 352, 2005
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4EQR
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![BU of 4eqr by Molmil](/molmil-images/mine/4eqr) | Crystal structure of the Y361F mutant of Staphylococcus aureus CoADR | 分子名称: | CHLORIDE ION, COENZYME A, Coenzyme A disulfide reductase, ... | 著者 | Wallace, B.D, Edwards, J.S, Wallen, J.R, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-19 | 公開日 | 2012-10-17 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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2A66
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![BU of 2a66 by Molmil](/molmil-images/mine/2a66) | Human Liver Receptor Homologue DNA-Binding Domain (hLRH-1 DBD) in Complex with dsDNA from the hCYP7A1 Promoter | 分子名称: | 5'-D(*CP*TP*GP*GP*CP*CP*TP*TP*GP*AP*AP*C)-3', 5'-D(*GP*TP*TP*CP*AP*AP*GP*GP*CP*CP*AP*G)-3', ACETATE ION, ... | 著者 | Solomon, I.H, Hager, J.M, Safi, R, McDonnell, D.P, Redinbo, M.R, Ortlund, E.A. | 登録日 | 2005-07-01 | 公開日 | 2005-12-06 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal Structure of the Human LRH-1 DBD-DNA Complex Reveals Ftz-F1 Domain Positioning is Required for Receptor Activity. J.Mol.Biol., 354, 2005
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4EMW
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![BU of 4emw by Molmil](/molmil-images/mine/4emw) | Crystal Structure of Staphylococcus aureus bound with the covalent inhibitor EtVC-CoA | 分子名称: | CHLORIDE ION, Coenzyme A disulfide reductase, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Edwards, J.S, Wallace, B.D, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-12 | 公開日 | 2012-10-17 | 最終更新日 | 2019-07-17 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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4EQW
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![BU of 4eqw by Molmil](/molmil-images/mine/4eqw) | Crystal Structure of the Y361F, Y419F Mutant of Staphylococcus aureus CoADR | 分子名称: | CHLORIDE ION, COENZYME A, Coenzyme A disulfide reductase, ... | 著者 | Edwards, J.S, Wallace, B.D, Wallen, J.R, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-19 | 公開日 | 2012-10-17 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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4EM4
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![BU of 4em4 by Molmil](/molmil-images/mine/4em4) | Crystal Structure of Staphylococcus aureus bound with the covalent inhibitor Pethyl-VS-CoA | 分子名称: | CHLORIDE ION, Coenzyme A disulfide reductase, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Wallace, B.D, Edwards, J.S, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-11 | 公開日 | 2012-10-17 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.821 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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4EM3
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![BU of 4em3 by Molmil](/molmil-images/mine/4em3) | Crystal Structure of Staphylococcus aureus bound with the covalent inhibitor MeVS-CoA | 分子名称: | CHLORIDE ION, Coenzyme A disulfide reductase, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Wallace, B.D, Edwards, J.S, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-11 | 公開日 | 2012-10-17 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.977 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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4EQS
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![BU of 4eqs by Molmil](/molmil-images/mine/4eqs) | Crystal structure of the Y419F mutant of Staphylococcus aureus CoADR | 分子名称: | CHLORIDE ION, COENZYME A, Coenzyme A disulfide reductase, ... | 著者 | Wallace, B.D, Edwards, J.S, Wallen, J.R, Claiborne, A, Redinbo, M.R. | 登録日 | 2012-04-19 | 公開日 | 2012-10-17 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A-Disulfide Reductase by Coenzyme A-Mimetics: Mechanistic and Structural Insights. Biochemistry, 51, 2012
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3GS3
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![BU of 3gs3 by Molmil](/molmil-images/mine/3gs3) | |
3K4D
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![BU of 3k4d by Molmil](/molmil-images/mine/3k4d) | Crystal structure of E. coli beta-glucuronidase with the glucaro-d-lactam inhibitor bound | 分子名称: | (2S,3R,4S,5R)-3,4,5-trihydroxy-6-oxopiperidine-2-carboxylic acid, Beta-glucuronidase | 著者 | Wallace, B.D, Redinbo, M.R. | 登録日 | 2009-10-05 | 公開日 | 2010-11-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.393 Å) | 主引用文献 | Alleviating cancer drug toxicity by inhibiting a bacterial enzyme. Science, 330, 2010
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3K9B
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![BU of 3k9b by Molmil](/molmil-images/mine/3k9b) | |
3K4A
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![BU of 3k4a by Molmil](/molmil-images/mine/3k4a) | |
3K46
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![BU of 3k46 by Molmil](/molmil-images/mine/3k46) | |
1ILH
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![BU of 1ilh by Molmil](/molmil-images/mine/1ilh) | |