7CBU
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![BU of 7cbu by Molmil](/molmil-images/mine/7cbu) | Blasnase-T13A with L-Asp | 分子名称: | ASPARTIC ACID, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Ran, T, Jiao, L, Wang, W. | 登録日 | 2020-06-14 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structures of l-asparaginase from Bacillus licheniformis Reveal an Essential Residue for its Substrate Stereoselectivity. J.Agric.Food Chem., 69, 2021
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7CB4
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![BU of 7cb4 by Molmil](/molmil-images/mine/7cb4) | Crystal structures of of BlAsnase | 分子名称: | FORMIC ACID, GLYCEROL, L-asparaginase, ... | 著者 | Lu, F, Ran, T, Jiao, L, Wang, W. | 登録日 | 2020-06-10 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.04 Å) | 主引用文献 | Structures of l-asparaginase from Bacillus licheniformis Reveal an Essential Residue for its Substrate Stereoselectivity. J.Agric.Food Chem., 69, 2021
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7C8Q
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![BU of 7c8q by Molmil](/molmil-images/mine/7c8q) | Blasnase-T13A with D-asn | 分子名称: | Asparaginase, D-ASPARAGINE, FORMIC ACID, ... | 著者 | Lu, F, Ran, T, Jiao, L, Wang, W. | 登録日 | 2020-06-03 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Structures of l-asparaginase from Bacillus licheniformis Reveal an Essential Residue for its Substrate Stereoselectivity. J.Agric.Food Chem., 69, 2021
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7C8X
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![BU of 7c8x by Molmil](/molmil-images/mine/7c8x) | Blasnase-T13A with L-asn | 分子名称: | ASPARAGINE, Asparaginase, FORMIC ACID, ... | 著者 | Lu, F, Ran, T, Jiao, L, Wang, W. | 登録日 | 2020-06-03 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.994 Å) | 主引用文献 | Structures of l-asparaginase from Bacillus licheniformis Reveal an Essential Residue for its Substrate Stereoselectivity. J.Agric.Food Chem., 69, 2021
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7CBR
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![BU of 7cbr by Molmil](/molmil-images/mine/7cbr) | Blasnase-T13A with D-asn | 分子名称: | D-ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Ran, T, Jiao, L, Wang, W. | 登録日 | 2020-06-13 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structures of l-asparaginase from Bacillus licheniformis Reveal an Essential Residue for its Substrate Stereoselectivity. J.Agric.Food Chem., 69, 2021
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7CBW
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![BU of 7cbw by Molmil](/molmil-images/mine/7cbw) | Blasnase-T13A with D-asn | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Ran, T, Jiao, L, Wang, W. | 登録日 | 2020-06-15 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.978 Å) | 主引用文献 | Structures of l-asparaginase from Bacillus licheniformis Reveal an Essential Residue for its Substrate Stereoselectivity. J.Agric.Food Chem., 69, 2021
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7DTA
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7DAT
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![BU of 7dat by Molmil](/molmil-images/mine/7dat) | The crystal structure of COVID-19 main protease treated by AF | 分子名称: | COVID-19 MAIN PROTEASE, GOLD ION | 著者 | He, Z.S, He, B, Cao, P, Jiang, H.D, Gong, Y, Gao, X.Y. | 登録日 | 2020-10-18 | 公開日 | 2021-11-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | A comparison of Remdesivir versus gold cluster in COVID-19 animal model: A better therapeutic outcome of gold cluster. Nano Today, 44, 2022
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7DAV
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![BU of 7dav by Molmil](/molmil-images/mine/7dav) | The native crystal structure of COVID-19 main protease | 分子名称: | COVID-19 MAIN PROTEASE | 著者 | He, Z.S, He, B, Cao, P, Jiang, H.D, Gong, Y, Gao, X.Y. | 登録日 | 2020-10-18 | 公開日 | 2021-11-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | A comparison of Remdesivir versus gold cluster in COVID-19 animal model: A better therapeutic outcome of gold cluster. Nano Today, 44, 2022
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7DAU
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![BU of 7dau by Molmil](/molmil-images/mine/7dau) | The crystal structure of COVID-19 main protease treated by GA | 分子名称: | COVID-19 MAIN PROTEASE, GOLD ION | 著者 | He, Z.S, He, B, Cao, P, Jiang, H.D, Gong, Y, Gao, X.Y. | 登録日 | 2020-10-18 | 公開日 | 2021-11-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | A comparison of Remdesivir versus gold cluster in COVID-19 animal model: A better therapeutic outcome of gold cluster. Nano Today, 44, 2022
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7F36
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![BU of 7f36 by Molmil](/molmil-images/mine/7f36) | TacT complexed with acetyl-glycyl-tRNAGly | 分子名称: | ACETYLAMINO-ACETIC ACID, CALCIUM ION, N-acetyltransferase domain-containing protein, ... | 著者 | Yashiro, Y, Tomita, K. | 登録日 | 2021-06-15 | 公開日 | 2021-12-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.098 Å) | 主引用文献 | Molecular basis of glycyl-tRNAGly acetylation by TacT from Salmonella Typhimurium Cell Rep, 37, 2021
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7F37
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![BU of 7f37 by Molmil](/molmil-images/mine/7f37) | Crystal structure of AtaT2-AtaR2 complex | 分子名称: | DUF1778 domain-containing protein, GNAT family N-acetyltransferase | 著者 | Yashiro, Y, Tomita, K. | 登録日 | 2021-06-15 | 公開日 | 2021-12-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.896 Å) | 主引用文献 | Molecular basis of glycyl-tRNAGly acetylation by TacT from Salmonella Typhimurium Cell Rep, 37, 2021
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7F2S
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![BU of 7f2s by Molmil](/molmil-images/mine/7f2s) | Crystal structure of anti S-gatifloxacin antibody Fab fragment apo form | 分子名称: | 1,2-ETHANEDIOL, Antibody Fab fragment heavy chain, Antibody Fab fragment light chain, ... | 著者 | Wang, L.T, Jiao, W.Y, Shen, X, Lei, H.T. | 登録日 | 2021-06-14 | 公開日 | 2021-12-29 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | Conformational adaptability determining antibody recognition to distomer: structure analysis of enantioselective antibody against chiral drug gatifloxacin Rsc Adv, 11, 2021
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7F35
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![BU of 7f35 by Molmil](/molmil-images/mine/7f35) | Crystal structure of anti S-gatifloxacin antibody Fab fragment in complex with S-gatifloxacin | 分子名称: | 1,2-ETHANEDIOL, 1-cyclopropyl-6-fluoro-8-methoxy-7-[(3S)-3-methylpiperazin-1-yl]-4-oxo-1,4-dihydroquinoline-3-carboxylic acid, Antibody Fab fragment heavy chain, ... | 著者 | Wang, L.T, Jiao, W.Y, Shen, X, Lei, H.T. | 登録日 | 2021-06-15 | 公開日 | 2021-12-29 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Conformational adaptability determining antibody recognition to distomer: structure analysis of enantioselective antibody against chiral drug gatifloxacin Rsc Adv, 11, 2021
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7FAR
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![BU of 7far by Molmil](/molmil-images/mine/7far) | Crystal structure of PDE5A in complex with inhibitor L12 | 分子名称: | 5-[bis(fluoranyl)methoxy]-2-[(4-chlorophenyl)methyl]-10-(3-methoxypropyl)-3,10-diazatricyclo[6.4.1.0^{4,13}]trideca-1,4(13),5,7-tetraen-9-one, MAGNESIUM ION, ZINC ION, ... | 著者 | Wu, D, Huang, Y.Y, Luo, H.B. | 登録日 | 2021-07-07 | 公開日 | 2022-05-18 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.40006471 Å) | 主引用文献 | Free energy perturbation (FEP)-guided scaffold hopping. Acta Pharm Sin B, 12, 2022
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7FAQ
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![BU of 7faq by Molmil](/molmil-images/mine/7faq) | Crystal structure of PDE5A in complex with inhibitor L1 | 分子名称: | 2-[(4-chlorophenyl)methyl]-5-methoxy-3,10-diazatricyclo[6.4.1.0^{4,13}]trideca-1,4(13),5,7-tetraen-9-one, MAGNESIUM ION, SULFATE ION, ... | 著者 | Wu, D, Huang, Y.Y, Luo, H.B. | 登録日 | 2021-07-07 | 公開日 | 2022-05-18 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.200136 Å) | 主引用文献 | Free energy perturbation (FEP)-guided scaffold hopping. Acta Pharm Sin B, 12, 2022
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7EXC
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![BU of 7exc by Molmil](/molmil-images/mine/7exc) | Crystal structure of T2R-TTL-1129A2 complex | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GLYCEROL, ... | 著者 | Yang, J.H, Yan, W. | 登録日 | 2021-05-26 | 公開日 | 2022-06-01 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Structure-Based Design and Synthesis of N-Substituted 3-Amino-beta-Carboline Derivatives as Potent alpha beta-Tubulin Degradation Agents J.Med.Chem., 65, 2022
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6UJG
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![BU of 6ujg by Molmil](/molmil-images/mine/6ujg) | |
6UMD
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6UME
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![BU of 6ume by Molmil](/molmil-images/mine/6ume) | |
6UMC
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![BU of 6umc by Molmil](/molmil-images/mine/6umc) | |
6UMF
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7JTQ
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7YP3
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![BU of 7yp3 by Molmil](/molmil-images/mine/7yp3) | Crystal structure of elaiophylin glycosyltransferase in complex with elaiophylin | 分子名称: | ACETATE ION, Elaiophylin, GLYCEROL, ... | 著者 | Xu, T, Liu, Q, Gan, Q, Liu, J. | 登録日 | 2022-08-02 | 公開日 | 2022-11-02 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Substrate-induced dimerization of elaiophylin glycosyltransferase reveals a novel self-activating form of glycosyltransferase for symmetric glycosylation. Acta Crystallogr D Struct Biol, 78, 2022
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7YP6
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![BU of 7yp6 by Molmil](/molmil-images/mine/7yp6) | Crystal structure of elaiophylin glycosyltransferase in complex with UDP | 分子名称: | Glycosyltransferase, R-1,2-PROPANEDIOL, URIDINE-5'-DIPHOSPHATE | 著者 | Xu, T, Liu, Q, Gan, Q, Liu, J. | 登録日 | 2022-08-02 | 公開日 | 2022-11-02 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Substrate-induced dimerization of elaiophylin glycosyltransferase reveals a novel self-activating form of glycosyltransferase for symmetric glycosylation. Acta Crystallogr D Struct Biol, 78, 2022
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