3LWE
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![BU of 3lwe by Molmil](/molmil-images/mine/3lwe) | The crystal structure of MPP8 | 分子名称: | M-phase phosphoprotein 8 | 著者 | Li, Z, Li, Z, Ruan, J, Xu, C, Tong, Y, Pan, P.W, Tempel, W, Crombet, L, Min, J, Zang, J, Structural Genomics Consortium (SGC) | 登録日 | 2010-02-23 | 公開日 | 2010-03-02 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural basis for specific binding of human MPP8 chromodomain to histone H3 methylated at lysine 9. Plos One, 6, 2011
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8IMG
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![BU of 8img by Molmil](/molmil-images/mine/8img) | Human cGAS catalytic domain bound with C20 | 分子名称: | 2-[2-hydroxy-2-oxoethyl-[3-(7-methoxy-4-methyl-2-oxidanylidene-chromen-3-yl)propanoyl]amino]ethanoic acid, Cyclic GMP-AMP synthase, ZINC ION | 著者 | Zhao, W.F, Li, J.M, Xu, Y.C. | 登録日 | 2023-03-06 | 公開日 | 2024-01-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Discovery of novel cGAS inhibitors based on natural flavonoids. Bioorg.Chem., 140, 2023
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4GAX
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![BU of 4gax by Molmil](/molmil-images/mine/4gax) | Crystal Structure of an alpha-Bisabolol synthase mutant | 分子名称: | Amorpha-4,11-diene synthase | 著者 | Li, J, Peng, Z. | 登録日 | 2012-07-26 | 公開日 | 2013-03-13 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.9948 Å) | 主引用文献 | Rational engineering of plasticity residues of sesquiterpene synthases from Artemisia annua: product specificity and catalytic efficiency. Biochem.J., 451, 2013
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7SL6
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![BU of 7sl6 by Molmil](/molmil-images/mine/7sl6) | |
7SL7
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![BU of 7sl7 by Molmil](/molmil-images/mine/7sl7) | |
7SL2
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![BU of 7sl2 by Molmil](/molmil-images/mine/7sl2) | |
7SL3
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![BU of 7sl3 by Molmil](/molmil-images/mine/7sl3) | |
7SL4
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7SL1
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8IMF
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8IME
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![BU of 8ime by Molmil](/molmil-images/mine/8ime) | Human cGAS catalytic domain bound with baicalin | 分子名称: | 5,6-dihydroxy-4-oxo-2-phenyl-4H-chromen-7-yl beta-D-glucopyranosiduronic acid, Cyclic GMP-AMP synthase, ZINC ION | 著者 | Zhao, W.F, Xu, Y.C. | 登録日 | 2023-03-06 | 公開日 | 2024-01-03 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | Discovery of novel cGAS inhibitors based on natural flavonoids. Bioorg.Chem., 140, 2023
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6LLB
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![BU of 6llb by Molmil](/molmil-images/mine/6llb) | Crystal structure of mpy-RNase J (mutant S247A), an archaeal RNase J from Methanolobus psychrophilus R15, in complex with 6 nt RNA | 分子名称: | MPY-RNase J, RNA (5'-R(P*AP*AP*AP*AP*AP*A)-3'), SULFATE ION, ... | 著者 | Li, D.F, Hou, Y.J, Guo, L. | 登録日 | 2019-12-22 | 公開日 | 2020-01-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | A newly identified duplex RNA unwinding activity of archaeal RNase J depends on processive exoribonucleolysis coupled steric occlusion by its structural archaeal loops. Rna Biol., 17, 2020
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6KZ8
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![BU of 6kz8 by Molmil](/molmil-images/mine/6kz8) | Crystal structure of plant Phospholipase D alpha complex with phosphatidic acid | 分子名称: | 1,2-DIOCTANOYL-SN-GLYCERO-3-PHOSPHATE, CALCIUM ION, Phospholipase D alpha 1 | 著者 | Li, J.X, Yu, F, Zhang, P. | 登録日 | 2019-09-23 | 公開日 | 2019-11-13 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.291 Å) | 主引用文献 | Crystal structure of plant PLD alpha 1 reveals catalytic and regulatory mechanisms of eukaryotic phospholipase D. Cell Res., 30, 2020
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6KZ9
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5QII
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![BU of 5qii by Molmil](/molmil-images/mine/5qii) | CRYSTAL STRUCTURE OF 11BETA-HSD1 DOUBLE MUTANT (L262R, F278E) COMPLEXED WITH 2-(3-(1-(4-CHLOROPHENYL)CYCLOPROPYL) -[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-8-YL)PROPAN-2-OL | 分子名称: | 2-{3-[1-(4-chlorophenyl)cyclopropyl][1,2,4]triazolo[4,3-a]pyridin-8-yl}propan-2-ol, Corticosteroid 11-beta-dehydrogenase isozyme 1, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Sheriff, S. | 登録日 | 2018-07-03 | 公開日 | 2018-12-19 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11 beta-Hydroxysteroid Dehydrogenase Type 1 (11 beta-HSD-1). ACS Med Chem Lett, 9, 2018
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5QIJ
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![BU of 5qij by Molmil](/molmil-images/mine/5qij) | CRYSTAL STRUCTURE OF MURINE 11B- HYDROXYSTEROIDDEHYDROGENASE COMPLEXED WITH 2-(3-(1-(4- CHLOROPHENYL)CYCLOPROPYL)-[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-8- YL)PROPAN-2-OL | 分子名称: | 2-{3-[1-(4-chlorophenyl)cyclopropyl][1,2,4]triazolo[4,3-a]pyridin-8-yl}propan-2-ol, Corticosteroid 11-beta-dehydrogenase isozyme 1, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Sheriff, S. | 登録日 | 2018-07-03 | 公開日 | 2018-12-19 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11 beta-Hydroxysteroid Dehydrogenase Type 1 (11 beta-HSD-1). ACS Med Chem Lett, 9, 2018
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8TTH
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![BU of 8tth by Molmil](/molmil-images/mine/8tth) | NorA single mutant - D307N at pH 7.5 | 分子名称: | Heavy Chain of FabDA1 Variable Domain, Light Chain of FabDA1 Variable Domain, Quinolone resistance protein NorA | 著者 | Li, J.P, Li, Y, Koide, A, Kuang, H.H, Torres, V.J, Koide, S, Wang, D.N, Traaseth, N.J. | 登録日 | 2023-08-13 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | ELECTRON MICROSCOPY (3.54 Å) | 主引用文献 | Proton-coupled transport mechanism of the efflux pump NorA. Nat Commun, 15, 2024
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7N9Z
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![BU of 7n9z by Molmil](/molmil-images/mine/7n9z) | E. coli cytochrome bo3 in MSP nanodisc | 分子名称: | 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, CARDIOLIPIN, ... | 著者 | Vallese, F, Clarke, O.B. | 登録日 | 2021-06-19 | 公開日 | 2021-09-01 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (2.19 Å) | 主引用文献 | Cryo-EM structures of Escherichia coli cytochrome bo 3 reveal bound phospholipids and ubiquinone-8 in a dynamic substrate binding site. Proc.Natl.Acad.Sci.USA, 118, 2021
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8TTG
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![BU of 8ttg by Molmil](/molmil-images/mine/8ttg) | NorA single mutant - E222Q at pH 7.5 | 分子名称: | FabDA1 CDRH3 loop, Quinolone resistance protein NorA | 著者 | Li, J.P, Li, Y, Koide, A, Kuang, H.H, Torres, V.J, Koide, S, Wang, D.N, Traaseth, N.J. | 登録日 | 2023-08-13 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | ELECTRON MICROSCOPY (3.35 Å) | 主引用文献 | Proton-coupled transport mechanism of the efflux pump NorA. Nat Commun, 15, 2024
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8TTE
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![BU of 8tte by Molmil](/molmil-images/mine/8tte) | Protonated state of NorA at pH 5.0 | 分子名称: | FabDA1 CDRH3 loop, Quinolone resistance protein NorA | 著者 | Li, J.P, Li, Y, Koide, A, Kuang, H.H, Torres, V.J, Koide, S, Wang, D.N, Traaseth, N.J. | 登録日 | 2023-08-13 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | ELECTRON MICROSCOPY (3.26 Å) | 主引用文献 | Proton-coupled transport mechanism of the efflux pump NorA. Nat Commun, 15, 2024
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8TTF
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![BU of 8ttf by Molmil](/molmil-images/mine/8ttf) | NorA double mutant - E222QD307N at pH 7.5 | 分子名称: | Heavy Chain of FabDA1 Variable Domain, Light Chain of FabDA1 Variable Domain, Quinolone resistance protein NorA | 著者 | Li, J.P, Li, Y, Koide, A, Kuang, H.H, Torres, V.J, Koide, S, Wang, D.N, Traaseth, N.J. | 登録日 | 2023-08-13 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | ELECTRON MICROSCOPY (3.61 Å) | 主引用文献 | Proton-coupled transport mechanism of the efflux pump NorA. Nat Commun, 15, 2024
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8XAI
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7STI
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7STJ
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7STK
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