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6MRX
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BU of 6mrx by Molmil
Sialidase26 apo
分子名称: Sialidase26
著者Zaramela, L.S, Martino, C, Alisson-Silva, F, Rees, S.D, Diaz, S.L, Chuzel, L, Ganatra, M.B, Taron, C.H, Zuniga, C, Chang, G, Varki, A, Zengler, K.
登録日2018-10-15
公開日2019-10-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Gut bacteria responding to dietary change encode sialidases that exhibit preference for red meat-associated carbohydrates.
Nat Microbiol, 4, 2019
7OO4
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HaloTag Engineering for Enhanced Fluorogenicity and Kinetics with a Styrylpyridine Dye
分子名称: 4-[(E)-2-[1-(7-chloranylheptyl)pyridin-1-ium-4-yl]ethenyl]-N,N-dimethyl-aniline, CHLORIDE ION, Haloalkane dehalogenase
著者Stein, A, Liang, A.D.
登録日2021-05-26
公開日2021-07-21
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献HaloTag Engineering for Enhanced Fluorogenicity and Kinetics with a Styrylpyridium Dye.
Chembiochem, 22, 2021
4X93
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BU of 4x93 by Molmil
Crystal structure of Lysosomal Phospholipase A2 crystallized in the presence of methyl arachidonyl fluorophosphonate (tetragonal form)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ...
著者Glukhova, A, Tesmer, J.J.G.
登録日2014-12-11
公開日2015-03-25
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure and function of lysosomal phospholipase A2 and lecithin:cholesterol acyltransferase.
Nat Commun, 6, 2015
5KAT
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BU of 5kat by Molmil
The structure of SAV2435 bound to TETRAPHENYLPHOSPHONIUM
分子名称: GLYCEROL, SA2223 protein, TETRAPHENYLPHOSPHONIUM
著者Moreno, A, Wade, H.
登録日2016-06-02
公開日2016-08-24
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.101 Å)
主引用文献Solution Binding and Structural Analyses Reveal Potential Multidrug Resistance Functions for SAV2435 and CTR107 and Other GyrI-like Proteins.
Biochemistry, 55, 2016
6ZSB
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BU of 6zsb by Molmil
Human mitochondrial ribosome in complex with mRNA and P-site tRNA
分子名称: 12S mitochondrial rRNA, 16S mitochondrial rRNA, 28S ribosomal protein S10, ...
著者Aibara, S, Singh, V, Modelska, A, Amunts, A.
登録日2020-07-15
公開日2020-09-16
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Structural basis of mitochondrial translation.
Elife, 9, 2020
3OO6
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BU of 3oo6 by Molmil
Crystal structures and biochemical characterization of the bacterial solute receptor AcbH reveal an unprecedented exclusive substrate preference for b-D-galactopyranose
分子名称: ABC transporter binding protein AcbH, SULFATE ION, beta-D-galactopyranose
著者Vahedi-Faridi, A, Bulut, H, Licht, A.
登録日2010-08-30
公開日2010-12-29
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystal structures of the bacterial solute receptor AcbH displaying an exclusive substrate preference for beta-D-galactopyranose
J.Mol.Biol., 406, 2011
5NAT
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BU of 5nat by Molmil
Complement factor D in complex with the inhibitor (S)-Pyrrolidine-1,2-dicarboxylic acid 1-[(1-methyl-1H-indol-3-yl)-amide] 2-[(3-trifluoromethoxy-phenyl)-amide]
分子名称: (2~{S})-~{N}1-(1-methylindol-3-yl)-~{N}2-[3-(trifluoromethyloxy)phenyl]pyrrolidine-1,2-dicarboxamide, Complement factor D, GLYCEROL
著者Mac Sweeney, A, Ostermann, N.
登録日2017-02-28
公開日2018-03-21
最終更新日2019-10-02
実験手法X-RAY DIFFRACTION (1.17 Å)
主引用文献Discovery of Highly Potent and Selective Small-Molecule Reversible Factor D Inhibitors Demonstrating Alternative Complement Pathway Inhibition in Vivo.
J.Med.Chem., 60, 2017
3OP0
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BU of 3op0 by Molmil
Crystal structure of Cbl-c (Cbl-3) TKB domain in complex with EGFR pY1069 peptide
分子名称: Epidermal growth factor receptor, NICKEL (II) ION, SODIUM ION, ...
著者Chaikuad, A, Guo, K, Cooper, C.D.O, Ayinampudi, V, Krojer, T, Ugochukwu, E, Muniz, J.R.C, Vollmar, M, Canning, P, von Delft, F, Arrowsmith, C.H, Weigelt, J, Edwards, A.M, Bountra, C, Bullock, A, Structural Genomics Consortium (SGC)
登録日2010-08-31
公開日2010-10-20
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献Crystal structure of Cbl-c (Cbl-3) TKB domain in complex with EGFR pY1069 peptide
To be Published
6ZVK
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BU of 6zvk by Molmil
The Halastavi arva virus (HalV) intergenic region IRES promotes translation by the simplest possible initiation mechanism
分子名称: 18S RIBOSOMAL RNA, 28S RIBOSOMAL RNA, 40S RIBOSOMAL PROTEIN ES17, ...
著者Abaeva, I.S, Vicens, Q, Bochler, A, Soufari, H, Simonetti, A, Pestova, T, Hashem, Y, Hellen, C.U.T.
登録日2020-07-24
公開日2020-12-23
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.49 Å)
主引用文献The Halastavi arva Virus Intergenic Region IRES Promotes Translation by the Simplest Possible Initiation Mechanism.
Cell Rep, 33, 2020
7A4M
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BU of 7a4m by Molmil
Cryo-EM structure of mouse heavy-chain apoferritin at 1.22 A
分子名称: FE (III) ION, Ferritin heavy chain, ZINC ION
著者Nakane, T, Kotecha, A, Sente, A, Yamashita, K, McMullan, G, Masiulis, S, Brown, P.M.G.E, Grigoras, I.T, Malinauskaite, L, Malinauskas, T, Miehling, J, Yu, L, Karia, D, Pechnikova, E.V, de Jong, E, Keizer, J, Bischoff, M, McCormack, J, Tiemeijer, P, Hardwick, S.W, Chirgadze, D.Y, Murshudov, G, Aricescu, A.R, Scheres, S.H.W.
登録日2020-08-20
公開日2020-10-28
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (1.22 Å)
主引用文献Single-particle cryo-EM at atomic resolution.
Nature, 587, 2020
7OSD
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BU of 7osd by Molmil
NMR Solution Structure of Peptide 12: First-in-class cyclic Temporin L analogue with antibacterial and antibiofilm activities
分子名称: PHE-VAL-PRO-TRP-PHE-LYS-LYS-PHE-DLE-GLU-ARG-ILE-LEU-NH2
著者Brancaccio, D, Carotenuto, A.
登録日2021-06-08
公開日2021-08-11
最終更新日2021-08-25
実験手法SOLUTION NMR
主引用文献First-in-Class Cyclic Temporin L Analogue: Design, Synthesis, and Antimicrobial Assessment.
J.Med.Chem., 64, 2021
7A5V
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CryoEM structure of a human gamma-aminobutyric acid receptor, the GABA(A)R-beta3 homopentamer, in complex with histamine and megabody Mb25 in lipid nanodisc
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ...
著者Nakane, T, Kotecha, A, Sente, A, Yamashita, K, McMullan, G, Masiulis, S, Brown, P.M.G.E, Grigoras, I.T, Malinauskaite, L, Malinauskas, T, Miehling, J, Yu, L, Karia, D, Pechnikova, E.V, de Jong, E, Keizer, J, Bischoff, M, McCormack, J, Tiemeijer, P, Hardwick, S.W, Chirgadze, D.Y, Murshudov, G, Aricescu, A.R, Scheres, S.H.W.
登録日2020-08-22
公開日2020-11-18
最終更新日2020-11-25
実験手法ELECTRON MICROSCOPY (1.7 Å)
主引用文献Single-particle cryo-EM at atomic resolution.
Nature, 587, 2020
8AA4
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BU of 8aa4 by Molmil
SusC components of the dextran utilisation system (utilisome)
分子名称: SusC homolog
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8AA1
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BU of 8aa1 by Molmil
Core SusCD transporter units from the levan utilisome with levan fructo-oligosaccharides DP 8-12
分子名称: MAGNESIUM ION, SusC homolog, SusD homolog, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
7OS8
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BU of 7os8 by Molmil
NMR SOLUTION STRUCTURE OF [Pro3,DLeu9]TL
分子名称: PHE-VAL-PRO-TRP-PHE-SER-LYS-PHE-DLE-GLY-ARG-ILE-LEU-NH2
著者Brancaccio, D, Carotenuto, A.
登録日2021-06-08
公開日2021-08-11
最終更新日2021-08-25
実験手法SOLUTION NMR
主引用文献First-in-Class Cyclic Temporin L Analogue: Design, Synthesis, and Antimicrobial Assessment.
J.Med.Chem., 64, 2021
8AA0
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Levan utilisation machinery (utilisome) with levan fructo-oligosaccharides DP 8-12
分子名称: DUF4960 domain-containing protein, Glycoside hydrolase family 32, MAGNESIUM ION, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8AA2
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BU of 8aa2 by Molmil
Inactive levan utilisation machinery (utilisome) in the presence of levan fructo-oligosaccharides DP 15-25
分子名称: DUF4960 domain-containing protein, Glycoside hydrolase family 32, MAGNESIUM ION, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
5N7E
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BU of 5n7e by Molmil
Crystal structure of the Dbl-homology domain of Bcr-Abl in complex with monobody Mb(Bcr-DH_4).
分子名称: Breakpoint cluster region protein, Mb(Bcr-DH_4)
著者Reckel, S, Reynaud, A, Pojer, F, Hantschel, O.
登録日2017-02-20
公開日2017-12-27
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.647 Å)
主引用文献Structural and functional dissection of the DH and PH domains of oncogenic Bcr-Abl tyrosine kinase.
Nat Commun, 8, 2017
8AA3
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BU of 8aa3 by Molmil
Core SusCD transporter units from the inactive levan utilisome in the presence of levan fructo-oligosaccharides DP 15-25
分子名称: MAGNESIUM ION, SusC homolog, SusD homolog, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
3ORH
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BU of 3orh by Molmil
Human guanidinoacetate N-methyltransferase with SAH
分子名称: Guanidinoacetate N-methyltransferase, S-ADENOSYL-L-HOMOCYSTEINE
著者Dong, A, Wu, H, Zeng, H, Loppnau, P, Sundstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Plotnikov, A.N, Structural Genomics Consortium (SGC)
登録日2010-09-07
公開日2010-09-15
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献The crystal structure of human guanidinoacetate N-methyltransferase with SAH
TO BE PUBLISHED
8A9Y
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BU of 8a9y by Molmil
Substrate-free levan utilisation machinery (utilisome)
分子名称: DUF4960 domain-containing protein, Glycoside hydrolase family 32, MAGNESIUM ION, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
6ZS9
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BU of 6zs9 by Molmil
Human mitochondrial ribosome in complex with ribosome recycling factor
分子名称: 12S rRNA, 16S rRNA, 28S ribosomal protein S10, ...
著者Aibara, S, Singh, V, Modelska, A, Amunts, A.
登録日2020-07-15
公開日2020-10-14
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Structural basis of mitochondrial translation.
Elife, 9, 2020
5A7Q
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BU of 5a7q by Molmil
Crystal structure of human JMJD2A in complex with compound 30
分子名称: 1,2-ETHANEDIOL, 2-(5-azanyl-2-oxidanyl-phenyl)pyridine-4-carboxylic acid, CHLORIDE ION, ...
著者Velupillai, S, Krojer, T, Gileadi, C, Johansson, C, Korczynska, M, Le, D.D, Younger, N, Gregori-Puigjane, E, Tumber, A, Iwasa, E, Pollock, S.B, Ortiz Torres, I, Kopec, J, Dixon-Clarke, S, MacKenzie, A, Nowak, R, von Delft, F, Arrowsmith, C.H, Bountra, C, Edwards, A, Shoichet, B.K, Fujimori, D.G, Oppermann, U.
登録日2015-07-09
公開日2016-01-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Docking and Linking of Fragments to Discover Jumonji Histone Demethylase Inhibitors.
J.Med.Chem., 59, 2016
4LAV
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BU of 4lav by Molmil
Crystal Structure Analysis of FKBP52, Crystal Form II
分子名称: Peptidyl-prolyl cis-trans isomerase FKBP4, SULFATE ION
著者Bracher, A, Kozany, C, Haehle, A, Wild, P, Zacharias, M, Hausch, F.
登録日2013-06-20
公開日2013-08-21
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structures of the Free and Ligand-Bound FK1-FK2 Domain Segment of FKBP52 Reveal a Flexible Inter-Domain Hinge.
J.Mol.Biol., 425, 2013
7F5Y
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BU of 7f5y by Molmil
Crystal structure of the single-stranded dna-binding protein from Mycobacterium tuberculosis- Form III
分子名称: FORMIC ACID, Single-stranded DNA-binding protein
著者Srikalaivani, R, Paul, A, Sriram, R, Narayanan, S, Gopal, B, Vijayan, M.
登録日2021-06-23
公開日2022-05-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Structural variability of Mycobacterium tuberculosis SSB and susceptibility to inhibition.
Curr.Sci., 122, 2022

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