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1QKM
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BU of 1qkm by Molmil
HUMAN OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PARTIAL AGONIST GENISTEIN
分子名称: ESTROGEN RECEPTOR BETA, GENISTEIN
著者Pike, A.C.W, Brzozowski, A.M, Carlquist, M.
登録日1999-07-27
公開日2000-07-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure of the Ligand-Binding Domain of Oestrogen Receptor Beta in the Presence of a Partial Agonist and a Full Antagonist
Embo J., 18, 1999
4A3H
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BU of 4a3h by Molmil
2',4' DINITROPHENYL-2-DEOXY-2-FLURO-B-D-CELLOBIOSIDE COMPLEX OF THE ENDOGLUCANASE CEL5A FROM BACILLUS AGARADHAERENS AT 1.6 A RESOLUTION
分子名称: 2,4-DINITROPHENYL-2-DEOXY-2-FLUORO-BETA-D-CELLOBIOSIDE, PROTEIN (ENDOGLUCANASE)
著者Davies, G.J, Brzozowski, A.M, Andersen, K, Schulein, M, Mackenzie, L, Withers, S.G.
登録日1998-07-22
公開日1999-07-23
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Snapshots along an enzymatic reaction coordinate: analysis of a retaining beta-glycoside hydrolase.
Biochemistry, 37, 1998
4UNE
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BU of 4une by Molmil
Human insulin B26Phe mutant crystal structure
分子名称: INSULIN A CHAIN, INSULIN B CHAIN, SULFATE ION
著者Zakova, L, Klevtikova, E, Lepsik, M, Collinsova, M, Watson, C.J, Turkenburg, J.P, Jiracek, J, Brzozowski, A.M.
登録日2014-05-28
公開日2014-10-15
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Human Insulin Analogues Modified at the B26 Site Reveal a Hormone Conformation that is Undetected in the Receptor Complex
Acta Crystallogr.,Sect.D, 70, 2014
4UNG
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BU of 4ung by Molmil
Human insulin B26Asn mutant crystal structure
分子名称: INSULIN A CHAIN, INSULIN B CHAIN, SULFATE ION
著者Zakova, L, Klevtikova, E, Lepsik, M, Collinsova, M, Watson, C.J, Turkenburg, J.P, Jiracek, J, Brzozowski, A.M.
登録日2014-05-28
公開日2014-10-15
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Human Insulin Analogues Modified at the B26 Site Reveal a Hormone Conformation that is Undetected in the Receptor Complex
Acta Crystallogr.,Sect.D, 70, 2014
4UNH
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BU of 4unh by Molmil
Human insulin B26Gly mutant crystal structure
分子名称: INSULIN A CHAIN, INSULIN B CHAIN, SULFATE ION
著者Zakova, L, Klevtikova, E, Lepsik, M, Collinsova, M, Watson, C.J, Turkenburg, J.P, Jiracek, J, Brzozowski, A.M.
登録日2014-05-28
公開日2014-10-15
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Human Insulin Analogues Modified at the B26 Site Reveal a Hormone Conformation that is Undetected in the Receptor Complex
Acta Crystallogr.,Sect.D, 70, 2014
1UTD
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BU of 1utd by Molmil
The structure of the trp RNA-binding attenuation protein (TRAP) bound to a 63-nucleotide RNA molecule containing GAGUUU repeats
分子名称: 5'-R(*GP*UP*UP*UP*GP*AP)-3', TRANSCRIPTION ATTENUATION PROTEIN MTRB, TRYPTOPHAN
著者Hopcroft, N.H, Manfredo, A, Wendt, A.L, Brzozowski, A.M, Gollnick, P, Antson, A.A.
登録日2003-12-08
公開日2004-01-15
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Interaction of RNA with Trap: The Role of Triplet Repeats and Separating Spacer Nucleotides
J.Mol.Biol., 338, 2004
1W8P
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Structural properties of the B25Tyr-NMe-B26Phe insulin mutant.
分子名称: INSULIN A-CHAIN, INSULIN B-CHAIN, PHENOL, ...
著者Zakowa, L, Au-Alvarez, O, Dodson, E.J, Dodson, G.G, Brzozowski, A.M.
登録日2004-09-24
公開日2005-02-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Towards the Insulin-Igf-I Intermediate Structures: Functional and Structural Properties of the B25Tyr-Nme-B26Phe Insulin Mutant.
Biochemistry, 43, 2004
1W9X
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Bacillus halmapalus alpha amylase
分子名称: 4,6-dideoxy-4-{[(1S,4R,5S,6S)-4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-4,6-dideoxy-4-{[(1S,4R,5S,6S)-4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-beta-D-glucopyranose, ALPHA AMYLASE, CALCIUM ION, ...
著者Davies, G.J, Brzozowski, A.M, Dauter, Z, Rasmussen, M.D, Borchert, T.V, Wilson, K.S.
登録日2004-10-20
公開日2005-02-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure of a Bacillus Halmapalus Family 13 Alpha-Amylase, Bha, in Complex with an Acarbose-Derived Nonasaccharide at 2.1 A Resolution
Acta Crystallogr.,Sect.D, 61, 2005
1UOH
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HUMAN GANKYRIN
分子名称: 26S PROTEASOME NON-ATPASE REGULATORY SUBUNIT 10
著者Krzywda, S, Brzozowski, A.M, Wilkinson, A.J.
登録日2003-09-17
公開日2003-10-30
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Crystal Structure of Gankyrin, an Oncoprotein Found in Complexes with Cyclin-Dependent Kinase 4, a 19 S Proteasomal ATPase Regulator, and the Tumor Suppressors Rb and P53
J.Biol.Chem., 279, 2004
1LV7
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BU of 1lv7 by Molmil
Crystal Structure of the AAA domain of FtsH
分子名称: FtsH, SULFATE ION
著者Krzywda, S, Brzozowski, A.M, Verma, C, Karata, K, Ogura, T, Wilkinson, A.J.
登録日2002-05-26
公開日2002-10-09
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The crystal structure of the AAA domain of the ATP-dependent protease FtsH of Escherichia coli at 1.5 A resolution.
Structure, 10, 2002
8CLS
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BU of 8cls by Molmil
Drosophila melanogaster insulin receptor ectodomain in complex with DILP5
分子名称: Insulin-like receptor, Probable insulin-like peptide 5, Probable insulin-like peptide 5 A chain
著者Viola, C.M, Brzozowski, A.M, Shafi, T.
登録日2023-02-17
公開日2023-12-20
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Structural conservation of insulin/IGF signalling axis at the insulin receptors level in Drosophila and humans.
Nat Commun, 14, 2023
1GWR
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HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-OESTRADIOL AND TIF2 NRBOX3 PEPTIDE
分子名称: ESTRADIOL, OESTROGEN RECEPTOR, TRANSCRIPTION INTERMEDIARY FACTOR-2
著者Pike, A.C.W, Brzozowski, A.M.
登録日2002-03-22
公開日2002-08-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Interaction of Transcriptional Intermediary Factor 2 Nuclear Receptor Box Peptides with the Coactivator Binding Site of Estrogen Receptor Alpha.
J.Biol.Chem., 277, 2002
1HJ1
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BU of 1hj1 by Molmil
RAT OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PURE ANTIOESTROGEN ICI164,384
分子名称: N-BUTYL-11-[(7R,8R,9S,13S,14S,17S)-3,17-DIHYDROXY-13-METHYL-7,8,9,11,12,13,14,15,16,17-DECAHYDRO-6H-CYCLOPENTA[A]PHENANTHREN-7-YL]-N-METHYLUNDECANAMIDE, NICKEL (II) ION, OESTROGEN RECEPTOR BETA, ...
著者Pike, A.C.W, Brzozowski, A.M, Carlquist, M.
登録日2001-01-08
公開日2002-01-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Insights Into the Mode of Action of a Pure Antiestrogen
Structure, 9, 2001
1GWQ
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HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE CORE AND TIF2 NRBOX2 PEPTIDE
分子名称: NUCLEAR RECEPTOR COACTIVATOR 2, OESTROGEN RECEPTOR, RALOXIFENE CORE
著者Pike, A.C.W, Brzozowski, A.M.
登録日2002-03-22
公開日2002-08-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Interaction of Transcriptional Intermediary Factor 2 Nuclear Receptor Box Peptides with the Coactivator Binding Site of Estrogen Receptor Alpha.
J.Biol.Chem., 277, 2002
2VVL
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BU of 2vvl by Molmil
The structure of MAO-N-D3, a variant of monoamine oxidase from Aspergillus niger.
分子名称: 1,2-ETHANEDIOL, FLAVIN-ADENINE DINUCLEOTIDE, MONOAMINE OXIDASE N
著者Atkin, K.E, Hart, S, Turkenburg, J.P, Brzozowski, A.M, Grogan, G.J.
登録日2008-06-10
公開日2008-11-04
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献The Structure of Monoamine Oxidase from Aspergillus Niger Provides a Molecular Context for Improvements in Activity Obtained by Directed Evolution.
J.Mol.Biol., 384, 2008
2WUU
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BU of 2wuu by Molmil
Structure of N-myristoyltransferase from L. donovani
分子名称: 2-oxopentadecyl-CoA, N-MYRISTOYLTRANSFERASE
著者Brannigan, J.A, Smith, B.A, Yu, Z, Hodgkinson, M.R, Leatherbarrow, R.J, Tate, E.W, Brzozowski, A.M, Smith, D.F, Wilkinson, A.J.
登録日2009-10-09
公開日2009-12-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献N-Myristoyltransferase from Leishmania Donovani: Structural and Functional Characterisation of a Potential Drug Target for Visceral Leishmaniasis.
J.Mol.Biol., 396, 2010
5FAX
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BU of 5fax by Molmil
Structure of subtilase SubHal from Bacillus halmapalus
分子名称: CALCIUM ION, Subtilase SubHal from Bacillus halmapalus
著者Dohnalek, J, Brzozowski, A.M, Svendsen, A, Wilson, K.S.
登録日2015-12-12
公開日2016-05-18
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Stabilization of Enzymes by Metal Binding: Structures of Two Alkalophilic Bacillus Subtilases and Analysis of the Second Metal-Binding Site of the Subtilase Family
Book, 2016
5FBZ
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BU of 5fbz by Molmil
Structure of subtilase SubHal from Bacillus halmapalus - complex with chymotrypsin inhibitor CI2A
分子名称: Autoproteolytic fragment of enzyme subtilase SubHal, CALCIUM ION, Enzyme subtilase SubHal from Bacillus halmapalus, ...
著者Dohnalek, J, Brzozowski, A.M, Svendsen, A, Wilson, K.S.
登録日2015-12-14
公開日2016-05-18
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Stabilization of Enzymes by Metal Binding: Structures of Two Alkalophilic Bacillus Subtilases and Analysis of the Second Metal-Binding Site of the Subtilase Family
Book, 2016
3O0E
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BU of 3o0e by Molmil
Crystal structure of OmpF in complex with colicin peptide OBS1
分子名称: Colicin-E9, Porin OmpF, octyl beta-D-glucopyranoside
著者Wojdyla, J.A, Housden, N.G, Korczynska, J, Grishkovskaya, I, Kirkpatrick, N, Brzozowski, A.M, Kleanthous, C.
登録日2010-07-19
公開日2010-12-08
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.01 Å)
主引用文献Directed epitope delivery across the Escherichia coli outer membrane through the porin OmpF.
Proc.Natl.Acad.Sci.USA, 107, 2010
4OYY
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Humicola insolens cutinase
分子名称: Cutinase
著者Dauter, Z.D, Brzozowski, A.M, Turkenburg, J.P, Wilson, K.S.
登録日2014-02-13
公開日2014-07-30
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Thermodynamic and structural investigation of the specific SDS binding of humicola insolens cutinase.
Protein Sci., 23, 2014
4OYL
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Humicola insolens cutinase in complex with mono-ethylphosphate
分子名称: Cutinase
著者Dauter, Z.D, Brzozowski, A.M, Turkenburg, J.P, Wilson, K.S.
登録日2014-02-12
公開日2014-06-25
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Thermodynamic and structural investigation of the specific SDS binding of Humicola insolens cutinase.
Protein Sci., 23, 2014
2A3H
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CELLOBIOSE COMPLEX OF THE ENDOGLUCANASE CEL5A FROM BACILLUS AGARADHERANS AT 2.0 A RESOLUTION
分子名称: ENDOGLUCANASE, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose
著者Davies, G.J, Brzozowski, A.M, Andersen, K, Schulein, M.
登録日1998-01-22
公開日1999-03-16
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of the Bacillus agaradherans family 5 endoglucanase at 1.6 A and its cellobiose complex at 2.0 A resolution
Biochemistry, 37, 1998
1QFK
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STRUCTURE OF HUMAN FACTOR VIIA AND ITS IMPLICATIONS FOR THE TRIGGERING OF BLOOD COAGULATION
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, COAGULATION FACTOR VIIA HEAVY CHAIN, ...
著者Pike, A.C.W, Brzozowski, A.M, Roberts, S.M, Olsen, O.H, Persson, E.
登録日1999-04-12
公開日1999-08-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of human factor VIIa and its implications for the triggering of blood coagulation.
Proc.Natl.Acad.Sci.USA, 96, 1999
1QHP
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FIVE-DOMAIN ALPHA-AMYLASE FROM BACILLUS STEAROTHERMOPHILUS, MALTOSE COMPLEX
分子名称: ALPHA-AMYLASE, CALCIUM ION, SULFATE ION, ...
著者Dauter, Z, Dauter, M, Brzozowski, A.M, Christensen, S, Borchert, T.V, Beier, L, Wilson, K.S, Davies, G.J.
登録日1999-05-25
公開日2000-05-31
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献X-ray structure of Novamyl, the five-domain "maltogenic" alpha-amylase from Bacillus stearothermophilus: maltose and acarbose complexes at 1.7A resolution.
Biochemistry, 38, 1999
2BSX
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Crystal structure of the Plasmodium falciparum purine nucleoside phosphorylase complexed with inosine
分子名称: INOSINE, PURINE NUCLEOSIDE PHOSPHORYLASE
著者Schnick, C, Brzozowski, A.M, Dodson, E.J, Murshudov, G.N, Brannigan, J.A, Wilkinson, A.J.
登録日2005-05-24
公開日2005-08-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structures of Plasmodium Falciparum Purine Nucleoside Phosphorylase Complexed with Sulfate and its Natural Substrate Inosine
Acta Crystallogr.,Sect.D, 61, 2005

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