1M03
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![BU of 1m03 by Molmil](/molmil-images/mine/1m03) | Mutant Streptomyces plicatus beta-hexosaminidase (D313A) in complex with product (GlcNAc) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-N-acetylhexosaminidase, CHLORIDE ION, ... | 著者 | Williams, S.J, Mark, B.L, Vocadlo, D.J, James, M.N.G, Withers, S.G. | 登録日 | 2002-06-11 | 公開日 | 2002-12-11 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Aspartate 313 in the Streptomyces plicatus hexosaminidase plays a critical
role in substrate-assisted catalysis by orienting the 2-acetamido group
and stabilizing the transition state. J.Biol.Chem., 277, 2002
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1M04
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![BU of 1m04 by Molmil](/molmil-images/mine/1m04) | Mutant Streptomyces plicatus beta-hexosaminidase (D313N) in complex with product (GlcNAc) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-N-acetylhexosaminidase, CHLORIDE ION, ... | 著者 | Williams, S.J, Mark, B.L, Vocadlo, D.J, James, M.N.G, Withers, S.G. | 登録日 | 2002-06-11 | 公開日 | 2002-12-11 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Aspartate 313 in the Streptomyces plicatus hexosaminidase plays a critical
role in substrate-assisted catalysis by orienting the 2-acetamido group
and stabilizing the transition state. J.Biol.Chem., 277, 2002
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8CX9
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![BU of 8cx9 by Molmil](/molmil-images/mine/8cx9) | Structure of the SARS-COV2 PLpro (C111S) in complex with a dimeric Ubv that inhibits activity by an unusual allosteric mechanism | 分子名称: | BROMIDE ION, CHLORIDE ION, Papain-like protease nsp3, ... | 著者 | Singer, A.U, Slater, C.L, Patel, A, Russel, R, Mark, B.L, Sidhu, S.S. | 登録日 | 2022-05-20 | 公開日 | 2023-01-25 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Ubiquitin variants potently inhibit SARS-CoV-2 PLpro and viral replication via a novel site distal to the protease active site. Plos Pathog., 18, 2022
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2OXN
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![BU of 2oxn by Molmil](/molmil-images/mine/2oxn) | |
3PSE
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![BU of 3pse by Molmil](/molmil-images/mine/3pse) | Structure of a viral OTU domain protease bound to interferon-stimulated gene 15 (ISG15) | 分子名称: | 1.7.6 3-bromanylpropan-1-amine, GLYCEROL, RNA polymerase, ... | 著者 | Bacik, J.P, James, T.W, Frias-Staheli, N, Garcia-Sastre, A, Mark, B.L. | 登録日 | 2010-12-01 | 公開日 | 2011-01-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis for the removal of ubiquitin and interferon-stimulated gene 15 by a viral ovarian tumor domain-containing protease. Proc.Natl.Acad.Sci.USA, 108, 2011
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3PT2
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![BU of 3pt2 by Molmil](/molmil-images/mine/3pt2) | Structure of a viral OTU domain protease bound to Ubiquitin | 分子名称: | 1.7.6 3-bromanylpropan-1-amine, ACETATE ION, RNA polymerase, ... | 著者 | James, T.W, Bacik, J.P, Frias-Staheli, N, Garcia-Sastre, A, Mark, B.L. | 登録日 | 2010-12-02 | 公開日 | 2011-01-19 | 最終更新日 | 2023-05-31 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural basis for the removal of ubiquitin and interferon-stimulated gene 15 by a viral ovarian tumor domain-containing protease. Proc.Natl.Acad.Sci.USA, 108, 2011
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3QBW
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![BU of 3qbw by Molmil](/molmil-images/mine/3qbw) | Crystal structure of pseudomonas aeruginosa 1,6-anhydro-n-actetylmuramic acid kinase (ANMK) bound to adenosine diphosphate | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Anhydro-N-acetylmuramic acid kinase, SULFATE ION | 著者 | Bacik, J.P, Martin, D.R, Mark, B.L. | 登録日 | 2011-01-14 | 公開日 | 2011-02-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Molecular Basis of 1,6-Anhydro Bond Cleavage and Phosphoryl Transfer by Pseudomonas aeruginosa 1,6-Anhydro-N-acetylmuramic Acid Kinase. J.Biol.Chem., 286, 2011
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3QBX
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![BU of 3qbx by Molmil](/molmil-images/mine/3qbx) | Crystal structure of pseudomonas aeruginosa 1,6-anhydro-n-actetylmuramic acid kinase (ANMK) bound to 1,6-anhydro-n-actetylmuramic acid | 分子名称: | 2-(2-ACETYLAMINO-4-HYDROXY-6,8-DIOXA-BICYCLO[3.2.1]OCT-3-YLOXY)-PROPIONIC ACID, Anhydro-N-acetylmuramic acid kinase, SULFATE ION | 著者 | Bacik, J.P, Martin, D.R, Mark, B.L. | 登録日 | 2011-01-14 | 公開日 | 2011-02-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Molecular Basis of 1,6-Anhydro Bond Cleavage and Phosphoryl Transfer by Pseudomonas aeruginosa 1,6-Anhydro-N-acetylmuramic Acid Kinase. J.Biol.Chem., 286, 2011
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3GS6
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![BU of 3gs6 by Molmil](/molmil-images/mine/3gs6) | Vibrio Cholerea family 3 glycoside hydrolase (NagZ)in complex with N-butyryl-PUGNAc | 分子名称: | Beta-hexosaminidase, GLYCEROL, [[(3R,4R,5S,6R)-3-(BUTANOYLAMINO)-4,5-DIHYDROXY-6-(HYDROXYMETHYL)OXAN-2-YLIDENE]AMINO] N-PHENYLCARBAMATE | 著者 | Balcewich, M.D, Mark, B.L. | 登録日 | 2009-03-26 | 公開日 | 2009-06-30 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Insight into a strategy for attenuating AmpC-mediated beta-lactam resistance: structural basis for selective inhibition of the glycoside hydrolase NagZ. Protein Sci., 18, 2009
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3GSM
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![BU of 3gsm by Molmil](/molmil-images/mine/3gsm) | Vibrio cholerae family 3 glycoside hydrolase (NagZ) bound to N-Valeryl-PUGNAc | 分子名称: | Beta-hexosaminidase, GLYCEROL, [[(3R,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)-3-(pentanoylamino)oxan-2-ylidene]amino] N-phenylcarbamate | 著者 | Balcewich, M.D, Mark, B.L. | 登録日 | 2009-03-27 | 公開日 | 2009-06-30 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Insight into a strategy for attenuating AmpC-mediated beta-lactam resistance: structural basis for selective inhibition of the glycoside hydrolase NagZ. Protein Sci., 18, 2009
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2WCA
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![BU of 2wca by Molmil](/molmil-images/mine/2wca) | BtGH84 in complex with n-butyl pugnac | 分子名称: | CALCIUM ION, O-GLCNACASE BT_4395, [[(3R,4R,5S,6R)-3-(BUTANOYLAMINO)-4,5-DIHYDROXY-6-(HYDROXYMETHYL)OXAN-2-YLIDENE]AMINO] N-PHENYLCARBAMATE | 著者 | He, Y, Davies, G.J. | 登録日 | 2009-03-10 | 公開日 | 2009-06-16 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Insight Into a Strategy for Attenuating Ampc- Mediated Beta-Lactam Resistance: Structural Basis for Selective Inhibition of the Glycoside Hydrolase Nagz. Protein Sci., 18, 2009
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5BSB
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![BU of 5bsb by Molmil](/molmil-images/mine/5bsb) | |
4YH5
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![BU of 4yh5 by Molmil](/molmil-images/mine/4yh5) | Lipomyces starkeyi levoglucosan kinase bound to ADP and Manganese | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ADENOSINE-5'-DIPHOSPHATE, Levoglucosan kinase, ... | 著者 | Bacik, J.P. | 登録日 | 2015-02-26 | 公開日 | 2015-09-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Producing Glucose 6-Phosphate from Cellulosic Biomass: STRUCTURAL INSIGHTS INTO LEVOGLUCOSAN BIOCONVERSION. J.Biol.Chem., 290, 2015
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4ZLU
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![BU of 4zlu by Molmil](/molmil-images/mine/4zlu) | |
4ZFV
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![BU of 4zfv by Molmil](/molmil-images/mine/4zfv) | |
5BVC
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![BU of 5bvc by Molmil](/molmil-images/mine/5bvc) | |