5K8Q
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5k8q by Molmil](/molmil-images/mine/5k8q) | Crystal Structure of Calcium-loaded Calmodulin in complex with STRA6 CaMBP2-site peptide. | 分子名称: | CALCIUM ION, Calmodulin, IMIDAZOLE, ... | 著者 | Stowe, S.D, Clarke, O.B, Cavalier, M.C, Godoy-Ruiz, R, Mancia, F, Weber, D.J. | 登録日 | 2016-05-30 | 公開日 | 2016-08-24 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.739 Å) | 主引用文献 | Structure of the STRA6 receptor for retinol uptake. Science, 353, 2016
|
|
5IPZ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ipz by Molmil](/molmil-images/mine/5ipz) | Crystal structure of human carbonic anhydrase isozyme IV with 5-(2-amino-1,3-thiazol-4-yl)-2-chlorobenzenesulfonamide | 分子名称: | 5-(2-amino-1,3-thiazol-4-yl)-2-chlorobenzene-1-sulfonamide, Carbonic anhydrase 4, ZINC ION | 著者 | Smirnov, A, Manakova, E, Grazulis, S. | 登録日 | 2016-03-10 | 公開日 | 2017-03-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Intrinsic thermodynamics of high affinity inhibitor binding to recombinant human carbonic anhydrase IV. Eur. Biophys. J., 47, 2018
|
|
5KN7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5kn7 by Molmil](/molmil-images/mine/5kn7) | Lipid A secondary acyltransferase LpxM from Acinetobacter baumannii | 分子名称: | DODECYL-BETA-D-MALTOSIDE, GLYCEROL, Lipid A biosynthesis lauroyl acyltransferase, ... | 著者 | Dovala, D.L, Hu, Q, Metzger IV, L.E. | 登録日 | 2016-06-27 | 公開日 | 2016-09-28 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Structure-guided enzymology of the lipid A acyltransferase LpxM reveals a dual activity mechanism. Proc.Natl.Acad.Sci.USA, 113, 2016
|
|
5J8R
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5j8r by Molmil](/molmil-images/mine/5j8r) | Crystal Structure of the Catalytic Domain of Human Protein Tyrosine Phosphatase non-receptor Type 12 - K61R mutant | 分子名称: | Tyrosine-protein phosphatase non-receptor type 12 | 著者 | Li, H, Yang, F, Xu, Y.F, Wang, W.J, Xiao, P, Yu, X, Sun, J.P. | 登録日 | 2016-04-08 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.043 Å) | 主引用文献 | Crystal structure and substrate specificity of PTPN12. Cell Rep, 15, 2016
|
|
5JNM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5jnm by Molmil](/molmil-images/mine/5jnm) | Crystal structure of MtlD from Staphylococcus aureus at 1.7-Angstrom resolution | 分子名称: | Mannitol-1-phosphate 5-dehydrogenase, SULFATE ION | 著者 | Ta, H.M, Nguyen, T, Kim, T, Kim, K.K. | 登録日 | 2016-04-30 | 公開日 | 2017-11-08 | 最終更新日 | 2019-09-04 | 実験手法 | X-RAY DIFFRACTION (1.701 Å) | 主引用文献 | Targeting Mannitol Metabolism as an Alternative Antimicrobial Strategy Based on the Structure-Function Study of Mannitol-1-Phosphate Dehydrogenase in Staphylococcus aureus. Mbio, 10, 2019
|
|
5K9R
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5k9r by Molmil](/molmil-images/mine/5k9r) | PDE10a with imidazopyrazine inhibitor | 分子名称: | 4-[5-[1-(2-methoxyethyl)pyrazol-4-yl]-2-(quinolin-2-yloxymethyl)imidazo[1,2-a]pyrazin-8-yl]morpholine, MAGNESIUM ION, ZINC ION, ... | 著者 | Gibbs, A.G, Schubert, C. | 登録日 | 2016-06-01 | 公開日 | 2016-08-24 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors. Bioorg.Med.Chem.Lett., 26, 2016
|
|
5KNK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5knk by Molmil](/molmil-images/mine/5knk) | Lipid A secondary acyltransferase LpxM from Acinetobacter baumannii with catalytic residue substitution (E127A) | 分子名称: | DODECYL-BETA-D-MALTOSIDE, GLYCEROL, Lipid A biosynthesis lauroyl acyltransferase, ... | 著者 | Dovala, D.L, Hu, Q, Metzger IV, L.E. | 登録日 | 2016-06-28 | 公開日 | 2016-09-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-guided enzymology of the lipid A acyltransferase LpxM reveals a dual activity mechanism. Proc.Natl.Acad.Sci.USA, 113, 2016
|
|
5KX6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5kx6 by Molmil](/molmil-images/mine/5kx6) | The structure of Arabidopsis thaliana FUT1 Mutant R284K in complex with GDP | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, ... | 著者 | Alahuhta, P.M, Lunin, V.V. | 登録日 | 2016-07-20 | 公開日 | 2016-09-28 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural, mutagenic and in silico studies of xyloglucan fucosylation in Arabidopsis thaliana suggest a water-mediated mechanism. Plant J., 91, 2017
|
|
5KWK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5kwk by Molmil](/molmil-images/mine/5kwk) | The structure of Arabidopsis thaliana FUT1 in complex with GDP | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, ... | 著者 | Alahuhta, P.M, Lunin, V.V. | 登録日 | 2016-07-18 | 公開日 | 2016-09-28 | 最終更新日 | 2018-05-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural, mutagenic and in silico studies of xyloglucan fucosylation in Arabidopsis thaliana suggest a water-mediated mechanism. Plant J., 91, 2017
|
|
5KOE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5koe by Molmil](/molmil-images/mine/5koe) | The structure of Arabidopsis thaliana FUT1 in complex with XXLG | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CHLORIDE ION, ... | 著者 | Alahuhta, P.M, Lunin, V.V. | 登録日 | 2016-06-30 | 公開日 | 2016-09-28 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Structural, mutagenic and in silico studies of xyloglucan fucosylation in Arabidopsis thaliana suggest a water-mediated mechanism. Plant J., 91, 2017
|
|
1XJD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1xjd by Molmil](/molmil-images/mine/1xjd) | |
1Y02
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1y02 by Molmil](/molmil-images/mine/1y02) | Crystal Structure of a FYVE-type domain from caspase regulator CARP2 | 分子名称: | FYVE-RING finger protein SAKURA, ZINC ION | 著者 | Tibbetts, M.D, Gu, L, Shiozaki, E.N, Shi, Y. | 登録日 | 2004-11-14 | 公開日 | 2004-12-28 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of a FYVE-type zinc finger domain from the caspase regulator CARP2. STRUCTURE, 12, 2004
|
|
2ACL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2acl by Molmil](/molmil-images/mine/2acl) | Liver X-Receptor alpha Ligand Binding Domain with SB313987 | 分子名称: | 1-BENZYL-3-(4-METHOXYPHENYLAMINO)-4-PHENYLPYRROLE-2,5-DIONE, Oxysterols receptor LXR-alpha, RETINOIC ACID, ... | 著者 | Jaye, M.C, Krawiec, J.A, Campobasso, N, Smallwood, A, Qiu, C, Lu, Q, Kerrigan, J.J. | 登録日 | 2005-07-19 | 公開日 | 2005-09-20 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Discovery of substituted maleimides as liver x receptor agonists and determination of a ligand-bound crystal structure. J.Med.Chem., 48, 2005
|
|
1Z8M
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1z8m by Molmil](/molmil-images/mine/1z8m) | |
1NCJ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1ncj by Molmil](/molmil-images/mine/1ncj) | N-CADHERIN, TWO-DOMAIN FRAGMENT | 分子名称: | CALCIUM ION, PROTEIN (N-CADHERIN), URANYL (VI) ION | 著者 | Tamura, K, Shan, W.-S, Hendrickson, W.A, Colman, D.R, Shapiro, L. | 登録日 | 1999-02-02 | 公開日 | 1999-03-18 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | Structure-function analysis of cell adhesion by neural (N-) cadherin. Neuron, 20, 1998
|
|
1P6C
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1p6c by Molmil](/molmil-images/mine/1p6c) | crystal structure of phosphotriesterase triple mutant H254G/H257W/L303T complexed with diisopropylmethylphosphonate | 分子名称: | DIETHYL 4-METHYLBENZYLPHOSPHONATE, METHYLPHOSPHONIC ACID DIISOPROPYL ESTER, Parathion hydrolase, ... | 著者 | Hill, C.M, Li, W, Thoden, J.B, Holden, H.M, Raushel, F.M. | 登録日 | 2003-04-29 | 公開日 | 2003-09-16 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Enhanced degradation of chemical warfare agents through molecular engineering of the phosphotriesterase active site. J.Am.Chem.Soc., 125, 2003
|
|
1QAL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1qal by Molmil](/molmil-images/mine/1qal) | THE ACTIVE SITE BASE CONTROLS COFACTOR REACTIVITY IN ESCHERICHIA COLI AMINE OXIDASE : X-RAY CRYSTALLOGRAPHIC STUDIES WITH MUTATIONAL VARIANTS | 分子名称: | CALCIUM ION, COPPER (II) ION, COPPER AMINE OXIDASE | 著者 | Murray, J.M, Wilmot, C.M, Saysell, C.G, Jaeger, J, Knowles, P.F, Phillips, S.E, McPherson, M.J. | 登録日 | 1999-03-19 | 公開日 | 1999-08-24 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The active site base controls cofactor reactivity in Escherichia coli amine oxidase: x-ray crystallographic studies with mutational variants. Biochemistry, 38, 1999
|
|
1P6B
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1p6b by Molmil](/molmil-images/mine/1p6b) | X-ray structure of phosphotriesterase, triple mutant H254G/H257W/L303T | 分子名称: | DIETHYL 4-METHYLBENZYLPHOSPHONATE, ETHYL DIHYDROGEN PHOSPHATE, Parathion hydrolase, ... | 著者 | Hill, C.M, Li, W, Thoden, J.B, Holden, H.M, Raushel, F.M. | 登録日 | 2003-04-29 | 公開日 | 2003-09-16 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Enhanced degradation of chemical warfare agents through molecular engineering of the phosphotriesterase active site. J.Am.Chem.Soc., 125, 2003
|
|
1QAF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1qaf by Molmil](/molmil-images/mine/1qaf) | THE ACTIVE SITE BASE CONTROLS COFACTOR REACTIVITY IN ESCHERICHIA COLI AMINE OXIDASE : X-RAY CRYSTALLOGRAPHIC STUDIES WITH MUTATIONAL VARIANTS | 分子名称: | CALCIUM ION, COPPER (II) ION, GLYCEROL, ... | 著者 | Murray, J.M, Wilmot, C.M, Saysell, C.G, Jaeger, J, Knowles, P.F, Phillips, S.E, McPherson, M.J. | 登録日 | 1999-03-11 | 公開日 | 1999-08-23 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The active site base controls cofactor reactivity in Escherichia coli amine oxidase: x-ray crystallographic studies with mutational variants. Biochemistry, 38, 1999
|
|
1QAK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1qak by Molmil](/molmil-images/mine/1qak) | THE ACTIVE SITE BASE CONTROLS COFACTOR REACTIVITY IN ESCHERICHIA COLI AMINE OXIDASE : X-RAY CRYSTALLOGRAPHIC STUDIES WITH MUTATIONAL VARIANTS | 分子名称: | CALCIUM ION, COPPER (II) ION, COPPER AMINE OXIDASE | 著者 | Murray, J.M, Wilmot, C.M, Saysell, C.G, Jaeger, J, Knowles, P.F, Phillips, S.E, McPherson, M.J. | 登録日 | 1999-03-15 | 公開日 | 1999-08-24 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The active site base controls cofactor reactivity in Escherichia coli amine oxidase: x-ray crystallographic studies with mutational variants. Biochemistry, 38, 1999
|
|
1FAD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1fad by Molmil](/molmil-images/mine/1fad) | DEATH DOMAIN OF FAS-ASSOCIATED DEATH DOMAIN PROTEIN, RESIDUES 89-183 | 分子名称: | PROTEIN (FADD PROTEIN) | 著者 | Jeong, E.-J, Bang, S, Lee, T.H, Park, Y.-I, Sim, W.-S, Kim, K.-S. | 登録日 | 1999-03-23 | 公開日 | 1999-07-06 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | The solution structure of FADD death domain. Structural basis of death domain interactions of Fas and FADD. J.Biol.Chem., 274, 1999
|
|
1GBU
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1gbu by Molmil](/molmil-images/mine/1gbu) | DEOXY (BETA-(C93A,C112G)) HUMAN HEMOGLOBIN | 分子名称: | HEMOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION | 著者 | Vasquez, G.B, Ji, X, Fronticelli, C, Gilliland, G.L. | 登録日 | 1996-01-04 | 公開日 | 1997-01-11 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Cysteines beta93 and beta112 as probes of conformational and functional events at the human hemoglobin subunit interfaces. Biophys.J., 76, 1999
|
|
1GBV
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1gbv by Molmil](/molmil-images/mine/1gbv) | (ALPHA-OXY, BETA-(C112G)DEOXY) T-STATE HUMAN HEMOGLOBIN | 分子名称: | HEMOGLOBIN, OXYGEN MOLECULE, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Vasquez, G.B, Ji, X, Pechik, I, Fronticelli, C, Gilliland, G.L. | 登録日 | 1995-12-20 | 公開日 | 1997-01-11 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Cysteines beta93 and beta112 as probes of conformational and functional events at the human hemoglobin subunit interfaces. Biophys.J., 76, 1999
|
|
1AV4
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1av4 by Molmil](/molmil-images/mine/1av4) | |
1AVK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1avk by Molmil](/molmil-images/mine/1avk) | CRYSTAL STRUCTURES OF THE COPPER-CONTAINING AMINE OXIDASE FROM ARTHROBACTER GLOBIFORMIS IN THE HOLO-AND APO-FORMS: IMPLICATIONS FOR THE BIOGENESIS OF TOPA QUINONE | 分子名称: | AMINE OXIDASE | 著者 | Wilce, M.C.J, Guss, J.M, Freeman, H.C, Tanizawa, K, Yamaguchi, H. | 登録日 | 1997-09-16 | 公開日 | 1998-03-18 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structures of the copper-containing amine oxidase from Arthrobacter globiformis in the holo and apo forms: implications for the biogenesis of topaquinone. Biochemistry, 36, 1997
|
|