3ZNC
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![BU of 3znc by Molmil](/molmil-images/mine/3znc) | MURINE CARBONIC ANHYDRASE IV COMPLEXED WITH BRINZOLAMIDE | 分子名称: | (+)-4-ETHYLAMINO-3,4-DIHYDRO-2-(METHOXY)PROPYL-2H-THIENO[3,2-E]-1,2-THIAZINE-6-SULFONAMIDE-1,1-DIOXIDE, CARBONIC ANHYDRASE IV, ZINC ION | 著者 | Stams, T, Chen, Y, Christianson, D.W. | 登録日 | 1998-02-10 | 公開日 | 1999-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structures of murine carbonic anhydrase IV and human carbonic anhydrase II complexed with brinzolamide: molecular basis of isozyme-drug discrimination. Protein Sci., 7, 1998
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3OUM
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![BU of 3oum by Molmil](/molmil-images/mine/3oum) | Crystal Structure of toxoflavin-degrading enzyme in complex with toxoflavin | 分子名称: | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione, MANGANESE (II) ION, toxoflavin-degrading enzyme | 著者 | Kim, M.I, Rhee, S. | 登録日 | 2010-09-15 | 公開日 | 2011-08-10 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural and functional analysis of phytotoxin toxoflavin-degrading enzyme Plos One, 6, 2011
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3OUL
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![BU of 3oul by Molmil](/molmil-images/mine/3oul) | |
3OJG
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![BU of 3ojg by Molmil](/molmil-images/mine/3ojg) | Structure of an inactive lactonase from Geobacillus kaustophilus with bound N-butyryl-DL-homoserine lactone | 分子名称: | FE (III) ION, N-[(3S)-2-oxotetrahydrofuran-3-yl]butanamide, Phosphotriesterase, ... | 著者 | Xue, B, Chow, J.Y, Tung, A, Robinson, R.C. | 登録日 | 2010-08-22 | 公開日 | 2010-10-27 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Directed evolution of a thermostable quorum-quenching lactonase from the amidohydrolase superfamily J.Biol.Chem., 285, 2010
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1QAL
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![BU of 1qal by Molmil](/molmil-images/mine/1qal) | THE ACTIVE SITE BASE CONTROLS COFACTOR REACTIVITY IN ESCHERICHIA COLI AMINE OXIDASE : X-RAY CRYSTALLOGRAPHIC STUDIES WITH MUTATIONAL VARIANTS | 分子名称: | CALCIUM ION, COPPER (II) ION, COPPER AMINE OXIDASE | 著者 | Murray, J.M, Wilmot, C.M, Saysell, C.G, Jaeger, J, Knowles, P.F, Phillips, S.E, McPherson, M.J. | 登録日 | 1999-03-19 | 公開日 | 1999-08-24 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The active site base controls cofactor reactivity in Escherichia coli amine oxidase: x-ray crystallographic studies with mutational variants. Biochemistry, 38, 1999
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1TCE
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![BU of 1tce by Molmil](/molmil-images/mine/1tce) | SOLUTION NMR STRUCTURE OF THE SHC SH2 DOMAIN COMPLEXED WITH A TYROSINE-PHOSPHORYLATED PEPTIDE FROM THE T-CELL RECEPTOR, MINIMIZED AVERAGE STRUCTURE | 分子名称: | PHOSPHOPEPTIDE OF THE ZETA CHAIN OF T CELL RECEPTOR, SHC | 著者 | Zhou, M.-M, Meadows, R.P, Logan, T.M, Yoon, H.S, Wade, W.R, Ravichandran, K.S, Burakoff, S.J, Feisk, S.W. | 登録日 | 1996-03-27 | 公開日 | 1997-05-15 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the Shc SH2 domain complexed with a tyrosine-phosphorylated peptide from the T-cell receptor. Proc.Natl.Acad.Sci.USA, 92, 1995
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1QAF
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![BU of 1qaf by Molmil](/molmil-images/mine/1qaf) | THE ACTIVE SITE BASE CONTROLS COFACTOR REACTIVITY IN ESCHERICHIA COLI AMINE OXIDASE : X-RAY CRYSTALLOGRAPHIC STUDIES WITH MUTATIONAL VARIANTS | 分子名称: | CALCIUM ION, COPPER (II) ION, GLYCEROL, ... | 著者 | Murray, J.M, Wilmot, C.M, Saysell, C.G, Jaeger, J, Knowles, P.F, Phillips, S.E, McPherson, M.J. | 登録日 | 1999-03-11 | 公開日 | 1999-08-23 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The active site base controls cofactor reactivity in Escherichia coli amine oxidase: x-ray crystallographic studies with mutational variants. Biochemistry, 38, 1999
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1P6C
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![BU of 1p6c by Molmil](/molmil-images/mine/1p6c) | crystal structure of phosphotriesterase triple mutant H254G/H257W/L303T complexed with diisopropylmethylphosphonate | 分子名称: | DIETHYL 4-METHYLBENZYLPHOSPHONATE, METHYLPHOSPHONIC ACID DIISOPROPYL ESTER, Parathion hydrolase, ... | 著者 | Hill, C.M, Li, W, Thoden, J.B, Holden, H.M, Raushel, F.M. | 登録日 | 2003-04-29 | 公開日 | 2003-09-16 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Enhanced degradation of chemical warfare agents through molecular engineering of the phosphotriesterase active site. J.Am.Chem.Soc., 125, 2003
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3Q8W
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![BU of 3q8w by Molmil](/molmil-images/mine/3q8w) | A b-aminoacyl containing thiazolidine derivative and DPPIV complex | 分子名称: | Dipeptidyl peptidase 4, N-(4-{[({(2R)-3-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-1,3-thiazolidin-2-yl}carbonyl)amino]methyl}phenyl)-D-valine | 著者 | Lee, J.O, Song, D.H. | 登録日 | 2011-01-07 | 公開日 | 2011-03-16 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (3.64 Å) | 主引用文献 | Discovery of b-aminoacyl containing thiazolidine derivatives as potent and selective dipeptidyl peptidase IV inhibitors To be Published
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3OGN
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![BU of 3ogn by Molmil](/molmil-images/mine/3ogn) | |
1SLU
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![BU of 1slu by Molmil](/molmil-images/mine/1slu) | |
1QAK
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![BU of 1qak by Molmil](/molmil-images/mine/1qak) | THE ACTIVE SITE BASE CONTROLS COFACTOR REACTIVITY IN ESCHERICHIA COLI AMINE OXIDASE : X-RAY CRYSTALLOGRAPHIC STUDIES WITH MUTATIONAL VARIANTS | 分子名称: | CALCIUM ION, COPPER (II) ION, COPPER AMINE OXIDASE | 著者 | Murray, J.M, Wilmot, C.M, Saysell, C.G, Jaeger, J, Knowles, P.F, Phillips, S.E, McPherson, M.J. | 登録日 | 1999-03-15 | 公開日 | 1999-08-24 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The active site base controls cofactor reactivity in Escherichia coli amine oxidase: x-ray crystallographic studies with mutational variants. Biochemistry, 38, 1999
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1SLV
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![BU of 1slv by Molmil](/molmil-images/mine/1slv) | |
1VKH
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![BU of 1vkh by Molmil](/molmil-images/mine/1vkh) | |
6ILQ
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![BU of 6ilq by Molmil](/molmil-images/mine/6ilq) | Crystal structure of PPARgamma with compound BR101549 | 分子名称: | Nuclear receptor coactivator 1, Peroxisome proliferator-activated receptor gamma, ethyl [2-butyl-6-oxo-1-{[2'-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl}-4-(propan-2-yl)-1,6-dihydropyrimidin-5-yl]acetate | 著者 | Hong, E, Jang, T.H, Chin, J, Kim, K.H, Jung, W, Kim, S.H. | 登録日 | 2018-10-19 | 公開日 | 2019-09-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.408 Å) | 主引用文献 | Identification of BR101549 as a lead candidate of non-TZD PPAR gamma agonist for the treatment of type 2 diabetes: Proof-of-concept evaluation and SAR. Bioorg.Med.Chem.Lett., 29, 2019
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6JPV
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![BU of 6jpv by Molmil](/molmil-images/mine/6jpv) | |
6HQ2
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![BU of 6hq2 by Molmil](/molmil-images/mine/6hq2) | |
6K39
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![BU of 6k39 by Molmil](/molmil-images/mine/6k39) | |
6ITS
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![BU of 6its by Molmil](/molmil-images/mine/6its) | |
6HQ7
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![BU of 6hq7 by Molmil](/molmil-images/mine/6hq7) | |
6HQ3
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![BU of 6hq3 by Molmil](/molmil-images/mine/6hq3) | |
6HQ4
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![BU of 6hq4 by Molmil](/molmil-images/mine/6hq4) | |
6HQ5
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![BU of 6hq5 by Molmil](/molmil-images/mine/6hq5) | Structure of EAL Enzyme Bd1971 - cAMP and cyclic-di-GMP bound form | 分子名称: | 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), ADENOSINE-3',5'-CYCLIC-MONOPHOSPHATE, CALCIUM ION, ... | 著者 | Lovering, A.L, Cadby, I.T. | 登録日 | 2018-09-24 | 公開日 | 2019-07-31 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.83 Å) | 主引用文献 | Nucleotide signaling pathway convergence in a cAMP-sensing bacterial c-di-GMP phosphodiesterase. Embo J., 38, 2019
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6KTY
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![BU of 6kty by Molmil](/molmil-images/mine/6kty) | |
6L18
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![BU of 6l18 by Molmil](/molmil-images/mine/6l18) | |