5TH9
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![BU of 5th9 by Molmil](/molmil-images/mine/5th9) | Structure determination of a potent, selective antibody inhibitor of human MMP9 (GS-5745 bound to MMP-9) | 分子名称: | CALCIUM ION, COBALT HEXAMMINE(III), GS-5745 Fab heavy chain, ... | 著者 | Appleby, T.C, Greenstein, A.E, Kwon, H.J. | 登録日 | 2016-09-29 | 公開日 | 2017-03-15 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.999 Å) | 主引用文献 | Biochemical characterization and structure determination of a potent, selective antibody inhibitor of human MMP9. J. Biol. Chem., 292, 2017
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5TH6
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![BU of 5th6 by Molmil](/molmil-images/mine/5th6) | Structure determination of a potent, selective antibody inhibitor of human MMP9 (apo MMP9) | 分子名称: | CALCIUM ION, Matrix metalloproteinase-9,Matrix metalloproteinase-9, ZINC ION | 著者 | Appleby, T.C, Greenstein, A.E, Kwon, H.J. | 登録日 | 2016-09-29 | 公開日 | 2017-03-01 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Biochemical characterization and structure determination of a potent, selective antibody inhibitor of human MMP9. J. Biol. Chem., 292, 2017
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5TZU
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![BU of 5tzu by Molmil](/molmil-images/mine/5tzu) | Crystal structure of human CD47 ECD bound to Fab of B6H12.2 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACETATE ION, ... | 著者 | Cardoso, R.M.F. | 登録日 | 2016-11-22 | 公開日 | 2017-03-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Anti-leukemic activity and tolerability of anti-human CD47 monoclonal antibodies. Blood Cancer J, 7, 2017
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5TZ2
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![BU of 5tz2 by Molmil](/molmil-images/mine/5tz2) | Crystal structure of human CD47 ECD bound to Fab of C47B222 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, C47B222 Fab Heavy Chain, ... | 著者 | Cardoso, R.M.F. | 登録日 | 2016-11-21 | 公開日 | 2017-03-15 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.302 Å) | 主引用文献 | Anti-leukemic activity and tolerability of anti-human CD47 monoclonal antibodies. Blood Cancer J, 7, 2017
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5TZT
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![BU of 5tzt by Molmil](/molmil-images/mine/5tzt) | |
2KXS
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![BU of 2kxs by Molmil](/molmil-images/mine/2kxs) | ZO1 ZU5 domain in complex with GRINL1A peptide | 分子名称: | Tight junction protein ZO-1,Myocardial zonula adherens protein | 著者 | Wen, W, Zhang, M. | 登録日 | 2010-05-12 | 公開日 | 2011-03-30 | 最終更新日 | 2024-04-10 | 実験手法 | SOLUTION NMR | 主引用文献 | Cdc42-dependent formation of the ZO-1/MRCKb complex at the leading edge controls cell migration Embo J., 30, 2011
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2KXR
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![BU of 2kxr by Molmil](/molmil-images/mine/2kxr) | ZO1 ZU5 domain MC/AA mutation | 分子名称: | Tight junction protein ZO-1 | 著者 | Wen, W, Zhang, M. | 登録日 | 2010-05-12 | 公開日 | 2011-03-30 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Cdc42-dependent formation of the ZO-1/MRCKb complex at the leading edge controls cell migration Embo J., 30, 2011
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1XWI
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![BU of 1xwi by Molmil](/molmil-images/mine/1xwi) | |
7X78
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![BU of 7x78 by Molmil](/molmil-images/mine/7x78) | L-fuculose 1-phosphate aldolase | 分子名称: | L-fuculose phosphate aldolase, MAGNESIUM ION, SULFATE ION | 著者 | Lou, X, Zhang, Q, Bartlam, M. | 登録日 | 2022-03-09 | 公開日 | 2022-04-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural characterization of an L-fuculose-1-phosphate aldolase from Klebsiella pneumoniae. Biochem.Biophys.Res.Commun., 607, 2022
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7XRE
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![BU of 7xre by Molmil](/molmil-images/mine/7xre) | Crystal structure of DgpA | 分子名称: | DgpA, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Ma, W, He, P. | 登録日 | 2022-05-10 | 公開日 | 2023-02-15 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.76 Å) | 主引用文献 | Structural mechanism of a dual-functional enzyme DgpA/B/C as both a C -glycoside cleaving enzyme and an O - to C -glycoside isomerase. Acta Pharm Sin B, 13, 2023
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7XRF
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![BU of 7xrf by Molmil](/molmil-images/mine/7xrf) | Crystal structaure of DgpB/C complex | 分子名称: | AP_endonuc_2 domain-containing protein, DgpB, MANGANESE (II) ION | 著者 | Ma, M, He, P. | 登録日 | 2022-05-10 | 公開日 | 2023-02-15 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.137 Å) | 主引用文献 | Structural mechanism of a dual-functional enzyme DgpA/B/C as both a C -glycoside cleaving enzyme and an O - to C -glycoside isomerase. Acta Pharm Sin B, 13, 2023
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7XR9
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![BU of 7xr9 by Molmil](/molmil-images/mine/7xr9) | Crystal structure of DgpA with glucose | 分子名称: | DgpA, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, beta-D-glucopyranose | 著者 | Ma, W, He, P. | 登録日 | 2022-05-09 | 公開日 | 2023-04-05 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.42 Å) | 主引用文献 | Structural mechanism of a dual-functional enzyme DgpA/B/C as both a C -glycoside cleaving enzyme and an O - to C -glycoside isomerase. Acta Pharm Sin B, 13, 2023
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2FGV
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![BU of 2fgv by Molmil](/molmil-images/mine/2fgv) | X-ray crystal structure of HIV-1 Protease T80N variant in complex with the inhibitor saquinavir used to explore the role of invariant Thr80 in HIV-1 protease structure, function, and viral infectivity. | 分子名称: | (2S)-2-amino-3-phenylpropane-1,1-diol, 2-METHYL-DECAHYDRO-ISOQUINOLINE-3-CARBOXYLIC ACID, ASPARAGINE, ... | 著者 | Foulkes, J.E, Prabu-Jeyabalan, M, Cooper, D, Schiffer, C.A. | 登録日 | 2005-12-22 | 公開日 | 2006-11-07 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Role of invariant Thr80 in human immunodeficiency virus type 1 protease structure, function, and viral infectivity. J.Virol., 80, 2006
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2FGU
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![BU of 2fgu by Molmil](/molmil-images/mine/2fgu) | X-ray crystal structure of HIV-1 Protease T80S variant in complex with the inhibitor saquinavir used to explore the role of invariant Thr80 in HIV-1 protease structure, function, and viral infectivity. | 分子名称: | (2S)-2-amino-3-phenylpropane-1,1-diol, 2-METHYL-DECAHYDRO-ISOQUINOLINE-3-CARBOXYLIC ACID, ASPARAGINE, ... | 著者 | Foulkes, J.E, Prabu-Jeyabalan, M, Cooper, D, Schiffer, C.A. | 登録日 | 2005-12-22 | 公開日 | 2006-11-07 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Role of invariant Thr80 in human immunodeficiency virus type 1 protease structure, function, and viral infectivity. J.Virol., 80, 2006
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5VQF
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![BU of 5vqf by Molmil](/molmil-images/mine/5vqf) | Crystal Structure of pro-TGF-beta 1 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Transforming growth factor beta-1, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose | 著者 | Zhao, B, Xu, S, Dong, X, Lu, C, Springer, T.A. | 登録日 | 2017-05-08 | 公開日 | 2017-11-15 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Prodomain-growth factor swapping in the structure of pro-TGF-beta 1. J. Biol. Chem., 293, 2018
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5GSK
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![BU of 5gsk by Molmil](/molmil-images/mine/5gsk) | Crystal structure of duplex DNA3 in complex with Hg(II) and Sr(II) | 分子名称: | DNA (5'-D(*GP*GP*TP*CP*GP*TP*CP*C)-3'), MERCURY (II) ION, STRONTIUM ION | 著者 | Liu, H.H, Wang, R, Yao, Q.Q, Cheng, Y.Q, Yang, C, Luo, Q, Wu, B.X, Li, J.X, Ma, J.B, Sheng, J, Gan, J.H. | 登録日 | 2016-08-16 | 公開日 | 2017-02-08 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Flexibility and stabilization of HgII-mediated C:T and T:T base pairs in DNA duplex Nucleic Acids Res., 45, 2017
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3P5O
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![BU of 3p5o by Molmil](/molmil-images/mine/3p5o) | Crystal Structure of the First Bromodomain of Human Brd4 in complex with IBET inhibitor | 分子名称: | 1,2-ETHANEDIOL, 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide, Bromodomain-containing protein 4 | 著者 | Chung, C. | 登録日 | 2010-10-09 | 公開日 | 2010-11-17 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Suppression of inflammation by a synthetic histone mimic Nature, 468, 2010
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7X2M
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![BU of 7x2m by Molmil](/molmil-images/mine/7x2m) | Crystal structure of nanobody 1-2C7 with SARS-CoV-2 RBD | 分子名称: | 1-2C7, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-D-mannopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Spike protein S1 | 著者 | Wang, X.Q, Zhang, L.Q, Ren, Y.F, Li, M.X. | 登録日 | 2022-02-25 | 公開日 | 2022-12-14 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Broadly neutralizing and protective nanobodies against SARS-CoV-2 Omicron subvariants BA.1, BA.2, and BA.4/5 and diverse sarbecoviruses. Nat Commun, 13, 2022
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7X2J
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![BU of 7x2j by Molmil](/molmil-images/mine/7x2j) | Crystal structure of nanobody Nb70 with SARS-CoV RBD | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Nb70, Spike protein S1 | 著者 | Wang, X.Q, Zhang, L.Q, Ren, Y.F, Li, M.X. | 登録日 | 2022-02-25 | 公開日 | 2022-12-21 | 最終更新日 | 2023-06-28 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Broadly neutralizing and protective nanobodies against SARS-CoV-2 Omicron subvariants BA.1, BA.2, and BA.4/5 and diverse sarbecoviruses. Nat Commun, 13, 2022
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7X2K
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![BU of 7x2k by Molmil](/molmil-images/mine/7x2k) | Crystal structure of nanobody Nb70 with antibody 1F11 fab and SARS-CoV-2 RBD | 分子名称: | 1F11-H, 1F11-L, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Wang, X.Q, Zhang, L.Q, Ren, Y.F, Li, M.X. | 登録日 | 2022-02-25 | 公開日 | 2022-12-21 | 最終更新日 | 2023-06-28 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Broadly neutralizing and protective nanobodies against SARS-CoV-2 Omicron subvariants BA.1, BA.2, and BA.4/5 and diverse sarbecoviruses. Nat Commun, 13, 2022
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7X2L
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![BU of 7x2l by Molmil](/molmil-images/mine/7x2l) | Crystal structure of nanobody 3-2A2-4 with SARS-CoV-2 RBD | 分子名称: | Nanobody 3-2A2-4, Spike protein S1, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose | 著者 | Wang, X.Q, Zhang, L.Q, Ren, Y.F, Li, M.X. | 登録日 | 2022-02-25 | 公開日 | 2022-12-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Broadly neutralizing and protective nanobodies against SARS-CoV-2 Omicron subvariants BA.1, BA.2, and BA.4/5 and diverse sarbecoviruses. Nat Commun, 13, 2022
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7WAA
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2JUU
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![BU of 2juu by Molmil](/molmil-images/mine/2juu) | allo-ThrA3 DKP-insulin | 分子名称: | Insulin A chain, Insulin B chain | 著者 | Huang, K, Chan, S, Hua, Q, Chu, Y, Wang, R, Klaproth, B, Jia, W, Whittaker, J, De Meyts, P, Nakagawa, S.H, Steiner, D.F, Katsoyannis, P.G, Weiss, M.A. | 登録日 | 2007-09-03 | 公開日 | 2007-10-16 | 最終更新日 | 2021-10-20 | 実験手法 | SOLUTION NMR | 主引用文献 | The A-chain of Insulin Contacts the Insert Domain of the Insulin Receptor: PHOTO-CROSS-LINKING AND MUTAGENESIS OF A DIABETES-RELATED CREVICE. J.Biol.Chem., 282, 2007
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2JUM
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![BU of 2jum by Molmil](/molmil-images/mine/2jum) | ThrA3-DKP-insulin | 分子名称: | Insulin A chain, Insulin B chain | 著者 | Huang, K, Chan, S, Hua, Q, Chu, Y, Wang, R, Klaproth, B, Jia, W, Whittaker, J, De Meyts, P, Nakagawa, S.H, Steiner, D.F, Katsoyannis, P.G, Weiss, M.A. | 登録日 | 2007-08-31 | 公開日 | 2007-10-16 | 最終更新日 | 2021-10-20 | 実験手法 | SOLUTION NMR | 主引用文献 | The A-chain of Insulin Contacts the Insert Domain of the Insulin Receptor: PHOTO-CROSS-LINKING AND MUTAGENESIS OF A DIABETES-RELATED CREVICE. J.Biol.Chem., 282, 2007
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2JUV
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![BU of 2juv by Molmil](/molmil-images/mine/2juv) | AbaA3-DKP-insulin | 分子名称: | Insulin A chain, Insulin B chain | 著者 | Huang, K, Chan, S, Hua, Q, Chu, Y, Wang, R, Klaproth, B, Jia, W, Whittaker, J, De Meyts, P, Nakagawa, S.H, Steiner, D.F, Katsoyannis, P.G, Weiss, M.A. | 登録日 | 2007-09-05 | 公開日 | 2007-10-16 | 最終更新日 | 2021-10-20 | 実験手法 | SOLUTION NMR | 主引用文献 | The A-chain of Insulin Contacts the Insert Domain of the Insulin Receptor: PHOTO-CROSS-LINKING AND MUTAGENESIS OF A DIABETES-RELATED CREVICE. J.Biol.Chem., 282, 2007
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