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5VNY
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BU of 5vny by Molmil
Crystal structure of DM14-3 domain of Lgd
分子名称: Lethal (2) giant discs 1, isoform B
著者McMillan, B.J, Blacklow, S.C.
登録日2017-05-01
公開日2017-06-14
実験手法X-RAY DIFFRACTION (1.101 Å)
主引用文献Structural Basis for Regulation of ESCRT-III Complexes by Lgd.
Cell Rep, 19, 2017
5VO5
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BU of 5vo5 by Molmil
Crystal structure of Lgd-Shrub complex, single chain fusion
分子名称: Coiled-coil and C2 domain-containing protein 1-like,GH13992p
著者McMillan, B.J, Seegar, T.C.M, Blacklow, S.C.
登録日2017-05-02
公開日2017-06-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.004 Å)
主引用文献Structural Basis for Regulation of ESCRT-III Complexes by Lgd.
Cell Rep, 19, 2017
1AXW
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BU of 1axw by Molmil
E. COLI THYMIDYLATE SYNTHASE IN COMPLEX WITH METHOTREXATE (MTX) AND 2'-DEOXYURIDINE 5'-MONOPHOSPHATE (DUMP)
分子名称: 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, METHOTREXATE, THYMIDYLATE SYNTHASE
著者Stout, T.J, Sage, C.R, Stroud, R.M.
登録日1997-10-23
公開日1998-10-28
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Discovery of Thymidylate Synthase Inhibitors Using Flexible Docking and an Empirically Tuned Scoring Function
To be Published
1IAG
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BU of 1iag by Molmil
FIRST STRUCTURE OF A SNAKE VENOM METALLOPROTEINASE: A PROTOTYPE FOR MATRIX METALLOPROTEINASES(SLASH)COLLAGENASES
分子名称: ADAMALYSIN II, CALCIUM ION, SULFATE ION, ...
著者Gomis-Rueth, F.-X, Bode, W.
登録日1994-05-09
公開日1994-08-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献First structure of a snake venom metalloproteinase: a prototype for matrix metalloproteinases/collagenases.
EMBO J., 12, 1993
1RJU
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BU of 1rju by Molmil
Crystal structure of a truncated form of yeast copper thionein
分子名称: COPPER (I) ION, Metallothionein
著者Calderone, V, Dolderer, B, Hartmann, H.J, Echner, H, Luchinat, C, Del Bianco, C, Mangani, S, Weser, U.
登録日2003-11-20
公開日2004-12-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献The Crystal Structure of Yeast Copper Thionein: the solution of a long lasting Enigma.
Proc.Natl.Acad.Sci.USA, 102, 2005
1ZVX
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BU of 1zvx by Molmil
Crystal structure of the complex between MMP-8 and a phosphonate inhibitor (R-enantiomer)
分子名称: (1R)-1-{[(4'-METHOXY-1,1'-BIPHENYL-4-YL)SULFONYL]AMINO}-2-METHYLPROPYLPHOSPHONIC ACID, CALCIUM ION, Neutrophil collagenase, ...
著者Pochetti, G, Gavuzzo, E, Campestre, C, Agamennone, M, Tortorella, P, Consalvi, V, Gallina, C, Hiller, O, Tschesche, H, Tucker, P.A, Mazza, F.
登録日2005-06-03
公開日2006-05-16
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates.
J.Med.Chem., 49, 2006
1ZS0
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BU of 1zs0 by Molmil
Crystal structure of the complex between MMP-8 and a phosphonate inhibitor (S-enantiomer)
分子名称: (1S)-1-{[(4'-METHOXY-1,1'-BIPHENYL-4-YL)SULFONYL]AMINO}-2-METHYLPROPYLPHOSPHONIC ACID, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
著者Pochetti, G, Gavuzzo, E, Campestre, C, Agamennone, M, Tortorella, P, Consalvi, V, Gallina, C, Hiller, O, Tschesche, H, Tucker, P.A, Mazza, F.
登録日2005-05-23
公開日2006-05-02
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates.
J.Med.Chem., 49, 2006
1I73
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BU of 1i73 by Molmil
COMPLEX OF PRO-LEU-L-TRP PHOSPHONATE WITH THE CATALITIC DOMAIN OF MATRIX METALLO PROTEINASE-8 (MET80 FORM)
分子名称: CALCIUM ION, NEUTROPHIL COLLAGENASE, THREE RESIDUE PEPTIDE INHIBITOR, ...
著者Gavuzzo, E, Pochetti, G, Mazza, F, Gallina, C, Gorini, B, D'Alessio, S, Pieper, M, Tschesche, H, Tucker, P.A.
登録日2001-03-07
公開日2001-03-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Two crystal structures of human neutrophil collagenase, one complexed with a primed- and the other with an unprimed-side inhibitor: implications for drug design.
J.Med.Chem., 43, 2000
1I76
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COMPLEX OF 2-(BIPHENYL-4-SULFONYL)-1,2,3,4-TETRAHYDRO-ISOQUINOLINE-3-CARBOXYLIC ACID (D-TIC DERIVATIVE) WITH T CATALITIC DOMAIN OF MATRIX METALLO PROTEINASE-8 (MET80 FORM)
分子名称: 2-(BIPHENYL-4-SULFONYL)-1,2,3,4-TETRAHYDRO-ISOQUINOLINE-3-CARBOXYLIC ACID, CALCIUM ION, NEUTROPHIL COLLAGENASE, ...
著者Gavuzzo, E, Pochetti, G, Mazza, F, Gallina, C, Gorini, B, D'Alessio, S, Pieper, M, Tschesche, H, Tucker, P.A.
登録日2001-03-08
公開日2001-03-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Two crystal structures of human neutrophil collagenase, one complexed with a primed- and the other with an unprimed-side inhibitor: implications for drug design.
J.Med.Chem., 43, 2000
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