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5LLS

Porcine dipeptidyl peptidase IV in complex with 8-(3-aminopiperidin-1-yl)-7-[(2-bromophenyl)methyl]-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione

Summary for 5LLS
Entry DOI10.2210/pdb5lls/pdb
DescriptorDipeptidyl peptidase 4, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total)
Functional Keywordspeptidase, inhibitor, complex, hydrolase
Biological sourceSus scrofa (Pig)
Total number of polymer chains4
Total formula weight364428.55
Authors
Nar, H.,Blaesse, M. (deposition date: 2016-07-28, release date: 2016-09-14, Last modification date: 2024-01-10)
Primary citationSchnapp, G.,Klein, T.,Hoevels, Y.,Bakker, R.A.,Nar, H.
Comparative Analysis of Binding Kinetics and Thermodynamics of Dipeptidyl Peptidase-4 Inhibitors and Their Relationship to Structure.
J.Med.Chem., 59:7466-7477, 2016
Cited by
PubMed: 27438064
DOI: 10.1021/acs.jmedchem.6b00475
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.41 Å)
Structure validation

217705

PDB entries from 2024-03-27

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