Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
3K9V
DownloadVisualize
BU of 3k9v by Molmil
Crystal structure of rat mitochondrial P450 24A1 S57D in complex with CHAPS
分子名称: 1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial, 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, ...
著者Annalora, A.J, Goodin, D.B, Hong, W, Zhang, Q, Johnson, E.F, Stout, C.D.
登録日2009-10-16
公開日2009-12-15
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of CYP24A1, a mitochondrial cytochrome P450 involved in vitamin D metabolism.
J.Mol.Biol., 396, 2010
3K9Y
DownloadVisualize
BU of 3k9y by Molmil
Crystal structure of rat mitochondrial P450 24A1 S57D in complex with CYMAL-5
分子名称: 1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial, 5-CYCLOHEXYL-1-PENTYL-BETA-D-MALTOSIDE, ...
著者Annalora, A.J, Goodin, D.B, Hong, W, Zhang, Q, Johnson, E.F, Stout, C.D.
登録日2009-10-16
公開日2009-12-15
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of CYP24A1, a mitochondrial cytochrome P450 involved in vitamin D metabolism.
J.Mol.Biol., 396, 2010
5XJD
DownloadVisualize
BU of 5xjd by Molmil
TEAD in complex with fragment
分子名称: (2S)-2-phenyl-2-pyrrol-1-yl-ethanoic acid, Transcriptional enhancer factor TEF-3
著者Kaan, H.Y.K, Sim, A.Y.L, Tan, S.K.J, Verma, C, Song, H.
登録日2017-05-01
公開日2018-01-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献Targeting YAP/TAZ-TEAD protein-protein interactions using fragment-based and computational modeling approaches.
PLoS ONE, 12, 2017
3L15
DownloadVisualize
BU of 3l15 by Molmil
Human Tead2 transcriptional factor
分子名称: GLYCEROL, Transcriptional enhancer factor TEF-4
著者Tomchick, D.R, Luo, X, Tian, W.
登録日2009-12-10
公開日2010-04-07
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and functional analysis of the YAP-binding domain of human TEAD2.
Proc.Natl.Acad.Sci.USA, 107, 2010
3JUA
DownloadVisualize
BU of 3jua by Molmil
Structural basis of YAP recognition by TEAD4 in the Hippo pathway
分子名称: 65 kDa Yes-associated protein, Transcriptional enhancer factor TEF-3
著者Chen, L, Song, H.
登録日2009-09-15
公開日2010-02-23
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis of YAP recognition by TEAD4 in the hippo pathway.
Genes Dev., 24, 2010
5GN0
DownloadVisualize
BU of 5gn0 by Molmil
Structure of TAZ-TEAD complex
分子名称: CITRIC ACID, PALMITIC ACID, Transcriptional enhancer factor TEF-3, ...
著者Kaan, H.Y.K, Song, H.
登録日2016-07-18
公開日2017-05-31
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of TAZ-TEAD complex reveals a distinct interaction mode from that of YAP-TEAD complex
Sci Rep, 7, 2017
5DQE
DownloadVisualize
BU of 5dqe by Molmil
Crystal structure of human transcription factor TEAD2 in complex with bromo-fenamic acid
分子名称: 2-[(3-bromophenyl)amino]benzoic acid, Transcriptional enhancer factor TEF-4
著者Han, X, Luo, X.
登録日2015-09-14
公開日2015-11-25
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.183 Å)
主引用文献Targeting the Central Pocket in Human Transcription Factor TEAD as a Potential Cancer Therapeutic Strategy.
Structure, 23, 2015
6HAW
DownloadVisualize
BU of 6haw by Molmil
Crystal structure of bovine cytochrome bc1 in complex with 2-pyrazolyl quinolone inhibitor WDH2G7
分子名称: 1,2-DIHEXANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIPALMITOYL-SN-GLYCERO-3-PHOSPHATE, ...
著者Amporndanai, K, Hong, W.D, O'Neill, P.M, Hasnain, S.S, Antonyuk, S.V.
登録日2018-08-08
公開日2019-01-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Potent Antimalarial 2-Pyrazolyl Quinolonebc1(Qi) Inhibitors with Improved Drug-like Properties.
ACS Med Chem Lett, 9, 2018
5DQ8
DownloadVisualize
BU of 5dq8 by Molmil
Crystal structure of human transcription factor TEAD2 in complex with flufenamic acid
分子名称: 2-[[3-(TRIFLUOROMETHYL)PHENYL]AMINO] BENZOIC ACID, Transcriptional enhancer factor TEF-4
著者Han, X, Luo, X.
登録日2015-09-14
公開日2015-11-25
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.305 Å)
主引用文献Targeting the Central Pocket in Human Transcription Factor TEAD as a Potential Cancer Therapeutic Strategy.
Structure, 23, 2015
2OGD
DownloadVisualize
BU of 2ogd by Molmil
T. Brucei Farnesyl Diphosphate Synthase Complexed with Bisphosphonate BPH-527
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, ACETATE ION, BETA-MERCAPTOETHANOL, ...
著者Cao, R, Gao, Y, Robinson, H, Goddard, A, Oldfield, E.
登録日2007-01-05
公開日2007-10-02
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Bisphosphonates: Teaching Old Drugs with New Tricks
TO BE PUBLISHED
2OPN
DownloadVisualize
BU of 2opn by Molmil
Human Farnesyl Diphosphate Synthase Complexed with Bisphosphonate BPH-527
分子名称: Farnesyl pyrophosphate synthetase (FPP synthetase) (FPS) (Farnesyl diphosphate synthetase) [Includes: Dimethylallyltranstransferase (EC 2.5.1.1); Geranyltranstransferase (EC 2.5.1.10)], MAGNESIUM ION, PHOSPHATE ION, ...
著者Cao, R, Gao, Y.G, Robinson, H, Goddard, A, Oldfield, E.
登録日2007-01-29
公開日2007-10-02
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Bisphosphonates: Teaching Old Drugs with New Tricks
To be Published
5Y16
DownloadVisualize
BU of 5y16 by Molmil
Crystal structure of human DUSP28(Y102H)
分子名称: CHLORIDE ION, Dual specificity phosphatase 28, PHOSPHATE ION
著者Ku, B, Kim, M, Kim, S.J, Ryu, S.E.
登録日2017-07-19
公開日2017-11-22
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.399 Å)
主引用文献Structural and biochemical analysis of atypically low dephosphorylating activity of human dual-specificity phosphatase 28
PLoS ONE, 12, 2017
5Z2Q
DownloadVisualize
BU of 5z2q by Molmil
Vgll1-TEAD4 core complex
分子名称: PHOSPHATE ION, Transcription cofactor vestigial-like protein 1, Transcriptional enhancer factor TEF-3
著者Pobbati, A.V, Song, H.
登録日2018-01-03
公開日2018-01-31
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.74 Å)
主引用文献Structural and functional similarity between the Vgll1-TEAD and the YAP-TEAD complexes.
Structure, 20, 2012
7V7M
DownloadVisualize
BU of 7v7m by Molmil
crystal structure of SARS-CoV-2 3CL protease
分子名称: 3C-like proteinase
著者Yi, Y, Zhang, M, Ye, M.
登録日2021-08-21
公開日2022-06-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Schaftoside inhibits 3CL pro and PL pro of SARS-CoV-2 virus and regulates immune response and inflammation of host cells for the treatment of COVID-19.
Acta Pharm Sin B, 12, 2022
7YAC
DownloadVisualize
BU of 7yac by Molmil
Paltusotine-bound SSTR2-Gi complex
分子名称: Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(i) subunit alpha-1, ...
著者Zhao, J, Shao, Z.
登録日2022-06-27
公開日2023-04-19
最終更新日2023-09-27
実験手法ELECTRON MICROSCOPY (3.24 Å)
主引用文献Prospect of acromegaly therapy: molecular mechanism of clinical drugs octreotide and paltusotine.
Nat Commun, 14, 2023
7YAE
DownloadVisualize
BU of 7yae by Molmil
Octreotide-bound SSTR2-Gi complex
分子名称: CHOLESTEROL, DPN-CYS-PHE-DTR-LYS-THR-CYS-THO, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ...
著者Zhao, J, Shao, Z.
登録日2022-06-28
公開日2023-04-19
実験手法ELECTRON MICROSCOPY (3.37 Å)
主引用文献Prospect of acromegaly therapy: molecular mechanism of clinical drugs octreotide and paltusotine.
Nat Commun, 14, 2023
7XQ3
DownloadVisualize
BU of 7xq3 by Molmil
Crystal structure of the tetramer of thioredoxin domain containing-protein of Oncomelania hupensis(OhTRP14)
分子名称: Thioredoxin domain-containing protein 17
著者Wang, S.Q, Huang, S.Q.
登録日2022-05-06
公開日2022-10-12
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Structural insights into the redox regulation of Oncomelania hupensis TRP14 and its potential role in the snail host response to parasite invasion.
Fish Shellfish Immunol., 128, 2022
7XPW
DownloadVisualize
BU of 7xpw by Molmil
Structure of OhTRP14
分子名称: Thioredoxin domain-containing protein 17
著者Wang, S.Q, Huang, S.Q.
登録日2022-05-05
公開日2022-10-12
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Structural insights into the redox regulation of Oncomelania hupensis TRP14 and its potential role in the snail host response to parasite invasion.
Fish Shellfish Immunol., 128, 2022
<12

 

221051

件を2024-06-12に公開中

PDB statisticsPDBj update infoContact PDBjnumon