8OEM
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![BU of 8oem by Molmil](/molmil-images/mine/8oem) | Crystal structure of FutA bound to Fe(II) | 分子名称: | FE (II) ION, Putative iron ABC transporter, substrate binding protein | 著者 | Bolton, R, Tews, I. | 登録日 | 2023-03-10 | 公開日 | 2023-08-30 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A redox switch allows binding of Fe(II) and Fe(III) ions in the cyanobacterial iron-binding protein FutA from Prochlorococcus. Proc.Natl.Acad.Sci.USA, 121, 2024
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8OGG
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![BU of 8ogg by Molmil](/molmil-images/mine/8ogg) | Crystal structure of FutA after an accumulated dose of 5 kGy | 分子名称: | FE (III) ION, Putative iron ABC transporter, substrate binding protein | 著者 | Bolton, R, Tews, I. | 登録日 | 2023-03-20 | 公開日 | 2023-08-30 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | A redox switch allows binding of Fe(II) and Fe(III) ions in the cyanobacterial iron-binding protein FutA from Prochlorococcus. Proc.Natl.Acad.Sci.USA, 121, 2024
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8RK1
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3ZXH
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5KJ2
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![BU of 5kj2 by Molmil](/molmil-images/mine/5kj2) | The novel p300/CBP inhibitor A-485 uncovers a unique mechanism of action to target AR in castrate resistant prostate cancer | 分子名称: | Histone acetyltransferase p300, N-[(4-fluorophenyl)methyl]-2-{(1R)-5-[(methylcarbamoyl)amino]-2',4'-dioxo-2,3-dihydro-3'H-spiro[indene-1,5'-[1,3]oxazolidin]-3'-yl}-N-[(2S)-1,1,1-trifluoropropan-2-yl]acetamide, SODIUM ION | 著者 | Jakob, C.G, Qiu, W, Edalji, R.P, Sun, C. | 登録日 | 2016-06-17 | 公開日 | 2017-09-27 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours. Nature, 550, 2017
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6UUZ
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6CV7
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6GSS
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1ZIS
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![BU of 1zis by Molmil](/molmil-images/mine/1zis) | Recombinant Lumazine synthase (hexagonal form) | 分子名称: | 5-NITRO-6-RIBITYL-AMINO-2,4(1H,3H)-PYRIMIDINEDIONE, 6,7-dimethyl-8-ribityllumazine synthase, PHOSPHATE ION | 著者 | Lopez-Jaramillo, F.J. | 登録日 | 2005-04-27 | 公開日 | 2006-10-03 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Crystal structure of recombinant Lumazine synthase (hexagonal form) To be Published
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4KVO
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4KVM
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4KVX
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5YJE
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![BU of 5yje by Molmil](/molmil-images/mine/5yje) | Crystal structure of HIRA(644-1017) | 分子名称: | Protein HIRA, SULFATE ION | 著者 | Sato, Y, Senda, M, Senda, T. | 登録日 | 2017-10-10 | 公開日 | 2018-06-20 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Functional activity of the H3.3 histone chaperone complex HIRA requires trimerization of the HIRA subunit Nat Commun, 9, 2018
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1GNE
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![BU of 1gne by Molmil](/molmil-images/mine/1gne) | THE THREE-DIMENSIONAL STRUCTURE OF GLUTATHIONE S-TRANSFERASE OF SCHISTOSOMA JAPONICUM FUSED WITH A CONSERVED NEUTRALIZING EPITOPE ON GP41 OF HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | 分子名称: | GLUTATHIONE, GLUTATHIONE S-TRANSFERASE | 著者 | Lim, K, Ho, J.X, Keeling, K, Gilliland, G.L, Ji, X, Ruker, F, Carter, D.C. | 登録日 | 1994-06-16 | 公開日 | 1994-11-30 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Three-dimensional structure of Schistosoma japonicum glutathione S-transferase fused with a six-amino acid conserved neutralizing epitope of gp41 from HIV. Protein Sci., 3, 1994
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4OGS
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7LJE
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![BU of 7lje by Molmil](/molmil-images/mine/7lje) | Discovery of Spirohydantoins as Selective, Orally Bioavailable Inhibitors of p300/CBP Histone Acetyltransferases | 分子名称: | 2-[4-[(3'R,4S)-3'-fluoro-1-[2-[(4-fluorophenyl)methyl-[(1S)-2,2,2-trifluoro-1-methyl-ethyl]amino]-2-oxo-ethyl]-2,5-dioxo-spiro[imidazolidine-4,1'-indane]-5'-yl]pyrazol-1-yl]-N-methyl-acetamide, Histone acetyltransferase p300 | 著者 | Jakob, C.G. | 登録日 | 2021-01-29 | 公開日 | 2021-03-17 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.607 Å) | 主引用文献 | Discovery of spirohydantoins as selective, orally bioavailable inhibitors of p300/CBP histone acetyltransferases. Bioorg.Med.Chem.Lett., 39, 2021
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5GSS
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3PUP
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![BU of 3pup by Molmil](/molmil-images/mine/3pup) | Structure of Glycogen Synthase Kinase 3 beta (GSK3B) in complex with a ruthenium octasporine ligand (OS1) | 分子名称: | Glycogen synthase kinase-3 beta, Ruthenium octasporine | 著者 | Filippakopoulos, P, Kraling, K, Essen, L.O, Meggers, E, Knapp, S. | 登録日 | 2010-12-06 | 公開日 | 2010-12-22 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.99 Å) | 主引用文献 | Structurally sophisticated octahedral metal complexes as highly selective protein kinase inhibitors. J.Am.Chem.Soc., 133, 2011
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5IJN
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![BU of 5ijn by Molmil](/molmil-images/mine/5ijn) | Composite structure of the inner ring of the human nuclear pore complex (32 copies of Nup205) | 分子名称: | NUCLEAR PORE COMPLEX PROTEIN NUP155, NUCLEAR PORE COMPLEX PROTEIN NUP205, NUCLEAR PORE COMPLEX PROTEIN NUP54, ... | 著者 | Kosinski, J, Mosalaganti, S, von Appen, A, Beck, M. | 登録日 | 2016-03-02 | 公開日 | 2016-04-27 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (21.4 Å) | 主引用文献 | Molecular architecture of the inner ring scaffold of the human nuclear pore complex. Science, 352, 2016
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5CMB
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5CMC
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1GDC
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![BU of 1gdc by Molmil](/molmil-images/mine/1gdc) | REFINED SOLUTION STRUCTURE OF THE GLUCOCORTICOID RECEPTOR DNA-BINDING DOMAIN | 分子名称: | GLUCOCORTICOID RECEPTOR, ZINC ION | 著者 | Baumann, H, Paulsen, K, Kovacs, H, Berglund, H, Wright, A.P.H, Gustafsson, J.-A, Hard, T. | 登録日 | 1994-03-15 | 公開日 | 1994-06-22 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Refined solution structure of the glucocorticoid receptor DNA-binding domain. Biochemistry, 32, 1993
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7RGF
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![BU of 7rgf by Molmil](/molmil-images/mine/7rgf) | Protocadherin gammaC4 EC1-4 crystal structure disrupted trans interface | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ... | 著者 | Goodman, K.M, Mannepalli, S, Honig, B, Shapiro, L. | 登録日 | 2021-07-15 | 公開日 | 2022-03-16 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | How clustered protocadherin binding specificity is tuned for neuronal self-/nonself-recognition. Elife, 11, 2022
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4HWU
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![BU of 4hwu by Molmil](/molmil-images/mine/4hwu) | Crystal structure of the Ig-C2 type 1 domain from mouse Fibroblast growth factor receptor 2 (FGFR2) [NYSGRC-005912] | 分子名称: | Fibroblast growth factor receptor 2 | 著者 | Kumar, P.R, Ahmed, M, Banu, R, Bhosle, R, Calarese, D, Celikigil, A, Chamala, S, Chan, M.K, Chowdhury, S, Fiser, A, Garforth, S, Glenn, A.S, Hillerich, B, Khafizov, K, Love, J, Patel, H, Rubinstein, R, Seidel, R, Stead, M, Toro, R, Nathenson, S.G, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC), Atoms-to-Animals: The Immune Function Network (IFN) | 登録日 | 2012-11-08 | 公開日 | 2012-11-21 | 実験手法 | X-RAY DIFFRACTION (2.903 Å) | 主引用文献 | Crystal structure of the Ig-C2 type 1 domain from mouse FGFR2 [NYSGRC-005912] to be published
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5DZW
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![BU of 5dzw by Molmil](/molmil-images/mine/5dzw) | Protocadherin alpha 4 extracellular cadherin domains 1-4 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Protocadherin alpha-4, ... | 著者 | Goodman, K.M, Bahna, F, Mannepalli, S, Honig, B, Shapiro, L. | 登録日 | 2015-09-26 | 公開日 | 2016-05-04 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | Structural Basis of Diverse Homophilic Recognition by Clustered alpha- and beta-Protocadherins. Neuron, 90, 2016
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