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1B2Y
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BU of 1b2y by Molmil
STRUCTURE OF HUMAN PANCREATIC ALPHA-AMYLASE IN COMPLEX WITH THE CARBOHYDRATE INHIBITOR ACARBOSE
分子名称: CALCIUM ION, CHLORIDE ION, Pancreatic alpha-amylase, ...
著者Nahoum, V, Payan, F.
登録日1998-12-03
公開日2000-02-16
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Crystal structures of human pancreatic alpha-amylase in complex with carbohydrate and proteinaceous inhibitors.
Biochem.J., 346 Pt 1, 2000
7EK6
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BU of 7ek6 by Molmil
Structure of viral peptides IPB19/N52
分子名称: Spike protein S2
著者Yu, D, Qin, B, Cui, S, He, Y.
登録日2021-04-04
公開日2021-06-09
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.243 Å)
主引用文献Structure-based design and characterization of novel fusion-inhibitory lipopeptides against SARS-CoV-2 and emerging variants.
Emerg Microbes Infect, 10, 2021
3AA3
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BU of 3aa3 by Molmil
A52L E. coli RNase HI
分子名称: Ribonuclease HI
著者Takano, K.
登録日2009-11-11
公開日2010-10-06
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Protein core adaptability: crystal structures of the cavity-filling variants of Escherichia coli RNase HI
Protein Pept.Lett., 17, 2010
3AA2
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A52I E. coli RNase HI
分子名称: Ribonuclease HI
著者Takano, K.
登録日2009-11-11
公開日2010-10-06
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Protein core adaptability: crystal structures of the cavity-filling variants of Escherichia coli RNase HI
Protein Pept.Lett., 17, 2010
3AA5
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BU of 3aa5 by Molmil
A52F E.coli RNase HI
分子名称: Ribonuclease HI
著者Takano, K.
登録日2009-11-11
公開日2010-10-06
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Protein core adaptability: crystal structures of the cavity-filling variants of Escherichia coli RNase HI
Protein Pept.Lett., 17, 2010
4KQQ
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BU of 4kqq by Molmil
CRYSTAL STRUCTURE OF PENICILLIN-BINDING PROTEIN 3 FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH (5S)-Penicilloic Acid
分子名称: (2S,4S)-2-[(R)-carboxy{[(2R)-2-{[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]amino}-2-phenylacetyl]amino}methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, CHLORIDE ION, GLYCEROL, ...
著者Nettleship, J.E, Stuart, D.I, Owens, R.J, Ren, J.
登録日2013-05-15
公開日2013-11-06
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Binding of (5S)-Penicilloic Acid to Penicillin Binding Protein 3.
Acs Chem.Biol., 8, 2013
8PEO
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BU of 8peo by Molmil
H3K36me2 nucleosome-LEDGF/p75 PWWP domain complex
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-14
公開日2023-08-16
最終更新日2024-09-11
実験手法ELECTRON MICROSCOPY (2.69 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
8PC5
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BU of 8pc5 by Molmil
H3K36me3 nucleosome-LEDGF/p75 PWWP domain complex
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-09
公開日2023-08-16
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (3.02 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
8PC6
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BU of 8pc6 by Molmil
H3K36me3 nucleosome-LEDGF/p75 PWWP domain complex - pose 2
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-09
公開日2023-08-16
最終更新日2024-10-16
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
1KIR
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BU of 1kir by Molmil
FV MUTANT Y(A 50)S (VL DOMAIN) OF MOUSE MONOCLONAL ANTIBODY D1.3 COMPLEXED WITH HEN EGG WHITE LYSOZYME
分子名称: LYSOZYME, MONOCLONAL ANTIBODY D1.3
著者Fields, B.A, Poljak, R.J, Mariuzza, R.A.
登録日1996-10-23
公開日1996-12-23
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Hydrogen bonding and solvent structure in an antigen-antibody interface. Crystal structures and thermodynamic characterization of three Fv mutants complexed with lysozyme.
Biochemistry, 35, 1996
1YC4
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BU of 1yc4 by Molmil
Crystal structure of human HSP90alpha complexed with dihydroxyphenylpyrazoles
分子名称: 4-(1H-IMIDAZOL-4-YL)-3-(5-ETHYL-2,4-DIHYDROXY-PHENYL)-1H-PYRAZOLE, Heat shock protein HSP 90-alpha
著者Kreusch, A, Han, S, Brinker, A, Zhou, V, Choi, H, He, Y, Lesley, S.A, Caldwell, J, Gu, X.
登録日2004-12-21
公開日2005-02-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Crystal structures of human HSP90alpha-complexed with dihydroxyphenylpyrazoles.
Bioorg.Med.Chem.Lett., 15, 2005
8PEP
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BU of 8pep by Molmil
H3K36me2 nucleosome-LEDGF/p75 PWWP domain complex - pose 2
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-14
公開日2023-08-16
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (3.33 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
1KIP
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BU of 1kip by Molmil
FV MUTANT Y(B 32)A (VH DOMAIN) OF MOUSE MONOCLONAL ANTIBODY D1.3 COMPLEXED WITH HEN EGG WHITE LYSOZYME
分子名称: LYSOZYME, MONOCLONAL ANTIBODY D1.3
著者Fields, B.A, Poljak, R.J, Mariuzza, R.A.
登録日1996-10-23
公開日1996-12-23
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Hydrogen bonding and solvent structure in an antigen-antibody interface. Crystal structures and thermodynamic characterization of three Fv mutants complexed with lysozyme.
Biochemistry, 35, 1996
1KIQ
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BU of 1kiq by Molmil
FV MUTANT Y(B 101)F (VH DOMAIN) OF MOUSE MONOCLONAL ANTIBODY D1.3 COMPLEXED WITH HEN EGG WHITE LYSOZYME
分子名称: LYSOZYME, MONOCLONAL ANTIBODY D1.3
著者Fields, B.A, Poljak, R.J, Mariuzza, R.A.
登録日1996-10-23
公開日1996-12-23
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Hydrogen bonding and solvent structure in an antigen-antibody interface. Crystal structures and thermodynamic characterization of three Fv mutants complexed with lysozyme.
Biochemistry, 35, 1996
1YC1
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BU of 1yc1 by Molmil
Crystal Structures of human HSP90alpha complexed with dihydroxyphenylpyrazoles
分子名称: 4-(1,3-BENZODIOXOL-5-YL)-5-(5-ETHYL-2,4-DIHYDROXYPHENYL)-2H-PYRAZOLE-3-CARBOXYLIC ACID, Heat shock protein HSP 90-alpha
著者Kreusch, A, Han, S, Brinker, A, Zhou, V, Choi, H, He, Y, Lesley, S.A, Caldwell, J, Gu, X.
登録日2004-12-21
公開日2005-02-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of human HSP90alpha-complexed with dihydroxyphenylpyrazoles.
Bioorg.Med.Chem.Lett., 15, 2005
1YC3
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BU of 1yc3 by Molmil
Crystal Structure of human HSP90alpha complexed with dihydroxyphenylpyrazoles
分子名称: 4-(1,3-BENZODIOXOL-5-YL)-5-(5-ETHYL-2,4-DIHYDROXYPHENYL)-2H-PYRAZOLE-3-CARBOXYLIC ACID, Heat shock protein HSP 90-alpha
著者Kreusch, A, Han, S, Brinker, A, Zhou, V, Choi, H, He, Y, Lesley, S.A, Caldwell, J, Gu, X.
登録日2004-12-21
公開日2005-02-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Crystal structures of human HSP90alpha-complexed with dihydroxyphenylpyrazoles.
Bioorg.Med.Chem.Lett., 15, 2005
1A7N
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BU of 1a7n by Molmil
FV FRAGMENT OF MOUSE MONOCLONAL ANTIBODY D1.3 (BALB/C, IGG1, K) VARIANT FOR CHAIN L GLU81->ASP AND CHAIN H LEU312->VAL
分子名称: IGG1-KAPPA D1.3 FV (HEAVY CHAIN), IGG1-KAPPA D1.3 FV (LIGHT CHAIN)
著者Marks, C, Henrick, K, Winter, G.
登録日1998-03-16
公開日1998-04-29
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献X-Ray Structures of D1.3 Fv Mutants
To be Published
1A7Q
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BU of 1a7q by Molmil
FV FRAGMENT OF MOUSE MONOCLONAL ANTIBODY D1.3 (BALB/C, IGG1, K) HIGH AFFINITY EXPRESSED VARIANT CONTAINING SER26L->GLY, ILE29L->THR, GLU81L->ASP, THR97L->SER, PRO240H->LEU, ASP258H->ALA, LYS281H->GLU, ASN283H->ASP AND LEU312H->VAL
分子名称: IGG1-KAPPA D1.3 FV (HEAVY CHAIN), IGG1-KAPPA D1.3 FV (LIGHT CHAIN)
著者Marks, C, Henrick, K, Winter, G.
登録日1998-03-16
公開日1998-04-29
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献X-Ray Structures of D1.3 Fv Mutants
To be Published
1A7O
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BU of 1a7o by Molmil
FV FRAGMENT OF MOUSE MONOCLONAL ANTIBODY D1.3 (BALB/C, IGG1, K) R96L DELETION MUTANT ON VARIANT FOR CHAIN L GLU81->ASP AND CHAIN H LEU312->VAL
分子名称: IGG1-KAPPA D1.3 FV (HEAVY CHAIN), IGG1-KAPPA D1.3 FV (LIGHT CHAIN)
著者Marks, C, Henrick, K, Winter, G.
登録日1998-03-16
公開日1998-04-29
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献X-Ray Structures of D1.3 Fv Mutants
To be Published
3KAS
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BU of 3kas by Molmil
Machupo virus GP1 bound to human transferrin receptor 1
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Glycoprotein, ...
著者Abraham, J, Corbett, K.D, Harrison, S.C.
登録日2009-10-19
公開日2010-03-09
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis for receptor recognition by New World hemorrhagic fever arenaviruses.
Nat.Struct.Mol.Biol., 17, 2010
1GFZ
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BU of 1gfz by Molmil
FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE
分子名称: CAFFEINE, GLYCOGEN PHOSPHORYLASE, INOSINIC ACID, ...
著者Oikonomakos, N.G, Zographos, S.E, Skamnaki, V.T, Tsitsanou, K.E, Johnson, L.N.
登録日2000-06-29
公開日2000-07-26
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor site.
J.Biol.Chem., 275, 2000
1A7R
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BU of 1a7r by Molmil
FV FRAGMENT OF MOUSE MONOCLONAL ANTIBODY D1.3 (BALB/C, IGG1, K) VARIANT CHAIN L GLU81->ASP
分子名称: IGG1-KAPPA D1.3 FV (HEAVY CHAIN), IGG1-KAPPA D1.3 FV (LIGHT CHAIN)
著者Marks, C, Henrick, K, Winter, G.
登録日1998-03-16
公開日1998-04-29
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献X-Ray Structures of D1.3 Fv Mutants
To be Published
1A7P
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BU of 1a7p by Molmil
FV FRAGMENT OF MOUSE MONOCLONAL ANTIBODY D1.3 (BALB/C, IGG1, K) ENGINEERED MUTANT PRO95L->SER ON VARIANT CHAIN L GLU81->ASP AND CHAIN H LEU312->VAL
分子名称: ACETIC ACID, IGG1-KAPPA D1.3 FV (HEAVY CHAIN), IGG1-KAPPA D1.3 FV (LIGHT CHAIN)
著者Marks, C, Henrick, K, Winter, G.
登録日1998-03-16
公開日1998-04-29
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献X-Ray Structures of D1.3 Fv Mutants
To be Published
2GV0
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BU of 2gv0 by Molmil
The structure of the orthorhombic form of soft-shelled turtle lysozyme at 1.9 angstroms resolution
分子名称: Lysozyme C, SULFATE ION
著者Siritapetawee, J, Thammasirirak, S, Yuvaniyama, J, Robinson, R.C.
登録日2006-05-02
公開日2007-05-08
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystallization and the 1.9 angstroms of the egg-white lysozyme from a taiwanese soft-shelled turtle (trionyx sinensis wiegmann)
to be published
8STG
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BU of 8stg by Molmil
Discovery and clinical validation of RLY-4008, the first highly selective FGFR2 inhibitor with activity across FGFR2 alterations and resistance mutations
分子名称: Fibroblast growth factor receptor 2, N-{4-[(5P)-4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}-2-methylpropanamide
著者Valverde, R, Foster, L.
登録日2023-05-10
公開日2023-06-07
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.79 Å)
主引用文献RLY-4008, the First Highly Selective FGFR2 Inhibitor with Activity across FGFR2 Alterations and Resistance Mutations.
Cancer Discov, 13, 2023

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