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8XW1
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BU of 8xw1 by Molmil
Cryo-EM structure of OSCA1.2-V335W-DDM state
分子名称: Calcium permeable stress-gated cation channel 1
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (4.49 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XW2
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BU of 8xw2 by Molmil
Cryo-EM structure of OSCA1.2-DOPC-1:50-contracted state
分子名称: Calcium permeable stress-gated cation channel 1
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.59 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XS5
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BU of 8xs5 by Molmil
Cryo-EM structure of OSCA1.2-DOPC-1:20-contracted2 state
分子名称: Calcium permeable stress-gated cation channel 1
著者Zhang, Y, Han, Y.
登録日2024-01-08
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.33 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XW0
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BU of 8xw0 by Molmil
Cryo-EM structure of OSCA3.1-GDN state
分子名称: CSC1-like protein ERD4, O-[(R)-{[(2R)-2,3-bis(octadecanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-L-serine
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.11 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XW3
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BU of 8xw3 by Molmil
Cryo-EM structure of OSCA1.2-DOPC-1:50-expanded state
分子名称: Calcium permeable stress-gated cation channel 1
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.63 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XVY
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BU of 8xvy by Molmil
Cryo-EM structure of OSCA3.1-2E(R611E-R619E)-closed/open state
分子名称: CSC1-like protein ERD4
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.71 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XVZ
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BU of 8xvz by Molmil
Cryo-EM structure of OSCA3.1-2E(R611E-R619E)-closed/'desensitized' state
分子名称: CSC1-like protein ERD4
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.78 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XW4
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BU of 8xw4 by Molmil
Cryo-EM structure of TMEM63B-Digitonin state
分子名称: CSC1-like protein 2
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.84 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XAJ
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BU of 8xaj by Molmil
Cryo-EM structure of OSCA1.2-liposome-inside-in open state
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Calcium permeable stress-gated cation channel 1
著者Zhang, Y, Han, Y.
登録日2023-12-04
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.29 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XS0
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BU of 8xs0 by Molmil
Cryo-EM structure of OSCA3.1-1.1ver(Y367N-G454S-Y458I)-open/'desensitized' state
分子名称: CSC1-like protein ERD4
著者Zhang, Y, Han, Y.
登録日2024-01-08
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.89 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
8XVX
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BU of 8xvx by Molmil
Cryo-EM structure of OSCA1.2-DOPC-1:20-expanded state
分子名称: Calcium permeable stress-gated cation channel 1
著者Zhang, Y, Han, Y.
登録日2024-01-15
公開日2024-04-10
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.32 Å)
主引用文献Mechanical activation opens a lipid-lined pore in OSCA ion channels.
Nature, 628, 2024
2N78
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BU of 2n78 by Molmil
NMR structure of IF1 from Pseudomonas aeruginosa
分子名称: Translation initiation factor IF-1
著者Zhang, Y.
登録日2015-09-04
公開日2016-09-07
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献(1)H, (13)C and (15)N resonance assignments and secondary structure analysis of translation initiation factor 1 from Pseudomonas aeruginosa.
Biomol.Nmr Assign., 10, 2016
3PCU
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BU of 3pcu by Molmil
Crystal structure of human retinoic X receptor alpha ligand-binding domain complexed with LX0278 and SRC1 peptide
分子名称: 2-[(2S)-6-(2-methylbut-3-en-2-yl)-7-oxo-2,3-dihydro-7H-furo[3,2-g]chromen-2-yl]propan-2-yl acetate, Nuclear receptor coactivator 2, Retinoic acid receptor RXR-alpha
著者Zhang, H, Zhang, Y, Shen, H, Chen, J, Li, C, Chen, L, Hu, L, Jiang, H, Shen, X.
登録日2010-10-22
公開日2011-11-16
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献(+)-Rutamarin as a Dual Inducer of Both GLUT4 Translocation and Expression Efficiently Ameliorates Glucose Homeostasis in Insulin-Resistant Mice.
Plos One, 7, 2012
8AEY
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BU of 8aey by Molmil
3 A CRYO-EM STRUCTURE OF MYCOBACTERIUM TUBERCULOSIS FERRITIN FROM TIMEPIX3 detector
分子名称: Ferritin BfrB
著者Zhang, Y, van Schayck, J.P, Knoops, K, Peters, P.J, Ravelli, R.B.G.
登録日2022-07-14
公開日2023-01-18
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Integration of an Event-driven Timepix3 Hybrid Pixel Detector into a Cryo-EM Workflow
Microsc Microanal, 2023
4MQ9
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BU of 4mq9 by Molmil
Crystal structure of Thermus thermophilus RNA polymerase holoenzyme in complex with GE23077
分子名称: (2Z)-2-methylbut-2-enoic acid, DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ...
著者Ho, M.X, Arnold, E, Ebright, R.H, Zhang, Y, Tuske, S.
登録日2013-09-16
公開日2014-05-07
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.35 Å)
主引用文献GE23077 binds to the RNA polymerase 'i' and 'i+1' sites and prevents the binding of initiating nucleotides.
Elife, 3, 2014
5Y4O
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BU of 5y4o by Molmil
Cryo-EM structure of MscS channel, YnaI
分子名称: Low conductance mechanosensitive channel YnaI
著者Zhang, Y, Yu, J.
登録日2017-08-04
公開日2019-03-20
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献A binding-block ion selective mechanism revealed by a Na/K selective channel.
Protein Cell, 9, 2018
1R0V
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BU of 1r0v by Molmil
Structure Determination of the Dimeric Endonuclease in a Pseudo-face-centerd P21212 space group
分子名称: tRNA-intron endonuclease
著者Li, H, Zhang, Y.
登録日2003-09-23
公開日2004-03-09
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure determination of a truncated dimeric splicing endonuclease in pseudo-face-centered space group P2(1)2(1)2.
Acta Crystallogr.,Sect.D, 60, 2004
1R11
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BU of 1r11 by Molmil
Structure Determination of the Dimeric Endonuclease in a Pseudo-face-centerd P21 space group
分子名称: tRNA-intron endonuclease
著者Li, H, Zhang, Y.
登録日2003-09-23
公開日2004-03-09
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure determination of a truncated dimeric splicing endonuclease in pseudo-face-centered space group P2(1)2(1)2.
Acta Crystallogr.,Sect.D, 60, 2004
5HMC
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BU of 5hmc by Molmil
Crystal structure of S. sahachiroi AziG complexed with 5-methyl naphthoic acid
分子名称: 5-methylnaphthalene-1-carboxylic acid, Azi13, SULFATE ION
著者Zhang, Y, Erb, M.S, Ealick, S.E.
登録日2016-01-15
公開日2016-02-03
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Polyketide Ring Expansion Mediated by a Thioesterase, Chain Elongation and Cyclization Domain, in Azinomycin Biosynthesis: Characterization of AziB and AziG.
Biochemistry, 55, 2016
2I0I
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BU of 2i0i by Molmil
X-ray crystal structure of Sap97 PDZ3 bound to the C-terminal peptide of HPV18 E6
分子名称: Disks large homolog 1, peptide E6
著者Chen, X.S, Zhang, Y, Dasgupta, J, Banks, L, Thomas, M.
登録日2006-08-10
公開日2007-02-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structures of a Human Papillomavirus (HPV) E6 Polypeptide Bound to MAGUK Proteins: Mechanisms of Targeting Tumor Suppressors by a High-Risk HPV Oncoprotein.
J.Virol., 81, 2007
2I0L
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BU of 2i0l by Molmil
X-ray crystal structure of Sap97 PDZ2 bound to the C-terminal peptide of HPV18 E6.
分子名称: Disks large homolog 1, peptide E6
著者Chen, X.S, Zhang, Y, Dasgupta, J, Banks, L, Thomas, M.
登録日2006-08-10
公開日2007-02-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.31 Å)
主引用文献Structures of a Human Papillomavirus (HPV) E6 Polypeptide Bound to MAGUK Proteins: Mechanisms of Targeting Tumor Suppressors by a High-Risk HPV Oncoprotein.
J.Virol., 81, 2007
2I04
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BU of 2i04 by Molmil
X-ray crystal structure of MAGI-1 PDZ1 bound to the C-terminal peptide of HPV18 E6
分子名称: Membrane-associated guanylate kinase, WW and PDZ domain-containing protein 1, SULFATE ION, ...
著者Chen, X.S, Zhang, Y, Dasgupta, J, Banks, L, Thomas, M.
登録日2006-08-09
公開日2007-02-20
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structures of a Human Papillomavirus (HPV) E6 Polypeptide Bound to MAGUK Proteins: Mechanisms of Targeting Tumor Suppressors by a High-Risk HPV Oncoprotein.
J.Virol., 81, 2007
3LZD
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BU of 3lzd by Molmil
Crystal structure of Dph2 from Pyrococcus horikoshii with 4Fe-4S cluster
分子名称: Dph2, IRON/SULFUR CLUSTER, SULFATE ION
著者Torelli, A.T, Zhang, Y, Zhu, X, Lee, M, Dzikovski, B, Koralewski, R.M, Wang, E, Freed, J, Krebs, C, Lin, H, Ealick, S.E.
登録日2010-03-01
公開日2010-07-14
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Diphthamide biosynthesis requires an organic radical generated by an iron-sulphur enzyme.
Nature, 465, 2010
2ITK
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BU of 2itk by Molmil
human Pin1 bound to D-PEPTIDE
分子名称: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, D-Peptide, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1
著者Noel, J.P, Zhang, Y.
登録日2006-10-19
公開日2007-05-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Structural basis for high-affinity peptide inhibition of human Pin1.
Acs Chem.Biol., 2, 2007
7KHK
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BU of 7khk by Molmil
Crystal structure of KIT kinase domain with a small molecule inhibitor, PLX9486 (bezuclastinib) in the DFG-in state
分子名称: 4,5-dimethyl-N-(2-phenyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-1H-pyrazole-3-carboxamide, Mast/stem cell growth factor receptor Kit
著者Zhang, Y.
登録日2020-10-21
公開日2021-07-07
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.34 Å)
主引用文献Association of Combination of Conformation-Specific KIT Inhibitors With Clinical Benefit in Patients With Refractory Gastrointestinal Stromal Tumors: A Phase 1b/2a Nonrandomized Clinical Trial.
Jama Oncol, 7, 2021

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件を2024-10-02に公開中

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