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8OE4
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BU of 8oe4 by Molmil
Cryo-EM structure of a pre-dimerized human IL-23 complete extracellular signaling complex.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-12 receptor subunit beta-1,Death-associated protein kinase 1, ...
著者Bloch, Y, Felix, J, Savvides, S.N.
登録日2023-03-10
公開日2024-02-07
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structures of complete extracellular receptor assemblies mediated by IL-12 and IL-23.
Nat.Struct.Mol.Biol., 31, 2024
8ODX
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BU of 8odx by Molmil
Interleukin 12 receptor subunit beta-1 Fn domains in complex with antagonistic FAb4 fragment and VHH.
分子名称: FAb4 Heavy chain, FAb4 Light chain, Interleukin-12 receptor subunit beta-1, ...
著者Bloch, Y, Savvides, S.N.
登録日2023-03-09
公開日2024-02-07
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (4.4 Å)
主引用文献Structures of complete extracellular receptor assemblies mediated by IL-12 and IL-23.
Nat.Struct.Mol.Biol., 31, 2024
8OE0
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BU of 8oe0 by Molmil
Cryo-EM structure of a pre-dimerized murine IL-12 complete extracellular signaling complex (Class 2).
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-12 receptor subunit beta-1,Death-associated protein kinase 1, ...
著者Felix, J, Bloch, Y, Savvides, S.N.
登録日2023-03-10
公開日2024-02-07
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (4.6 Å)
主引用文献Structures of complete extracellular receptor assemblies mediated by IL-12 and IL-23.
Nat.Struct.Mol.Biol., 31, 2024
8PPM
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BU of 8ppm by Molmil
IL-12Rb1 neutralizing Fab4, crystal kappa variant
分子名称: Fab4 Light chain, crystal kappa variant, Fab4 heavy chain, ...
著者Bloch, Y, Savvides, S.N.
登録日2023-07-07
公開日2024-02-07
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Structures of complete extracellular receptor assemblies mediated by IL-12 and IL-23.
Nat.Struct.Mol.Biol., 31, 2024
8PB1
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BU of 8pb1 by Molmil
Cryo-EM structure of a pre-dimerized murine IL-12 complete extracellular signaling complex (Class 1), obtained after local refinement.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-12 receptor subunit beta-1,Death-associated protein kinase 1, Interleukin-12 receptor subunit beta-2,Calmodulin-1, ...
著者Felix, J, Bloch, Y, Savvides, S.N.
登録日2023-06-08
公開日2024-02-07
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structures of complete extracellular receptor assemblies mediated by IL-12 and IL-23.
Nat.Struct.Mol.Biol., 31, 2024
6QI5
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BU of 6qi5 by Molmil
Near Atomic Structure of an Atadenovirus Shows a possible gene duplication event and Intergenera Variations in Cementing Proteins
分子名称: Hexon protein, PIIIa, Penton protein, ...
著者Condezo, G.N, Marabini, R, Gomez-Blanco, J, SanMartin, C.
登録日2019-01-17
公開日2020-08-05
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Near-atomic structure of an atadenovirus reveals a conserved capsid-binding motif and intergenera variations in cementing proteins.
Sci Adv, 7, 2021
7P0H
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BU of 7p0h by Molmil
Crystal structure of Helicobacter pylori ComF fused to an artificial alphaREP crystallization helper(named B2)
分子名称: 1-O-pyrophosphono-5-O-phosphono-alpha-D-ribofuranose, GLYCEROL, Helicobacter pylori ComF fused to an artificial alphaREP crystallization helper (named B2), ...
著者Celma, L, Walbott, H, Legrand, P, Quevillon-Cheruel, S.
登録日2021-06-29
公開日2022-04-06
最終更新日2022-04-27
実験手法X-RAY DIFFRACTION (2.499 Å)
主引用文献ComFC mediates transport and handling of single-stranded DNA during natural transformation.
Nat Commun, 13, 2022
6TN3
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BU of 6tn3 by Molmil
Crystal Structure of Aspergillus fumigatus UDP-N-acetylglucosamine pyrophosphorylase in complex with GlcNAc-1P
分子名称: 2-acetamido-2-deoxy-1-O-phosphono-alpha-D-glucopyranose, PHOSPHATE ION, UDP-N-acetylglucosamine pyrophosphorylase
著者Raimi, O.G, Guerrero, R.H.
登録日2019-12-05
公開日2020-04-01
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.282 Å)
主引用文献A mechanism-inspired UDP- N -acetylglucosamine pyrophosphorylase inhibitor.
Rsc Chem Biol, 1, 2020
8BI2
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BU of 8bi2 by Molmil
Syk kinase domain in complex with macrocyclic inhibitor 20a
分子名称: 10,13,23-trimethyl-16-oxa-2,4,8,9,13,19,23,30-octazapentacyclo[19.5.2.1^{3,7}.1^{8,11}.0^{24,28}]triaconta-1(27),3,5,7(30),9,11(29),21,24(28),25-nonaen-20-one, Tyrosine-protein kinase SYK
著者Read, J.A, Patel, J.
登録日2022-11-01
公開日2023-06-14
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.508 Å)
主引用文献Optimization of a series of novel, potent and selective Macrocyclic SYK inhibitors.
Bioorg.Med.Chem.Lett., 91, 2023
8CIQ
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BU of 8ciq by Molmil
JzTx-34 toxin peptide
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-10
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJP
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BU of 8cjp by Molmil
JzTx-34 toxin peptide H18A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJS
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BU of 8cjs by Molmil
JzTx-34 toxin peptide W31A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJQ
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BU of 8cjq by Molmil
JzTx-34 toxin peptide E20A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJR
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BU of 8cjr by Molmil
JzTx-34 toxin peptide W25A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJT
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BU of 8cjt by Molmil
JzTx-34 toxin peptide W33A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CBQ
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BU of 8cbq by Molmil
structure of LEDGF/p75 PWWP domain bound to the H3K36 trimethylated dinucleosome
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Novacek, J, Veverka, V.
登録日2023-01-25
公開日2023-09-06
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
8CBN
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BU of 8cbn by Molmil
structure of LEDGF/p75 PWWP domain bound to the H3K36 trimethylated dinucleosome
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Novacek, J, Veverka, V.
登録日2023-01-25
公開日2023-12-27
実験手法ELECTRON MICROSCOPY (3.34 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
7AYY
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BU of 7ayy by Molmil
Structure of the human 8-oxoguanine DNA Glycosylase hOGG1 in complex with activator TH10785
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, N-glycosylase/DNA lyase, ...
著者Masuyer, G, Davies, J.R, Stenmark, P.
登録日2020-11-13
公開日2022-06-01
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Small-molecule activation of OGG1 increases oxidative DNA damage repair by gaining a new function.
Science, 376, 2022
7AYZ
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BU of 7ayz by Molmil
Structure of the mouse 8-oxoguanine DNA Glycosylase mOGG1 in complex with activator TH10785
分子名称: N-glycosylase/DNA lyase, NICKEL (II) ION, ~{N}-cyclohexyl-2-cyclopropyl-quinazolin-4-amine
著者Masuyer, G, Davies, J.R, Stenmark, P.
登録日2020-11-13
公開日2022-06-01
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Small-molecule activation of OGG1 increases oxidative DNA damage repair by gaining a new function.
Science, 376, 2022
7AZ0
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BU of 7az0 by Molmil
Structure of the mouse 8-oxoguanine DNA Glycosylase mOGG1 in complex with TH12161
分子名称: 2-cyclopropyl-~{N}-(4-iodophenyl)quinazolin-4-amine, N-glycosylase/DNA lyase, NICKEL (II) ION
著者Davies, J.R, Masuyer, G, Stenmark, P.
登録日2020-11-13
公開日2022-06-01
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Small-molecule activation of OGG1 increases oxidative DNA damage repair by gaining a new function.
Science, 376, 2022
8PEP
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BU of 8pep by Molmil
H3K36me2 nucleosome-LEDGF/p75 PWWP domain complex - pose 2
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-14
公開日2023-08-16
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (3.33 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
8PC5
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BU of 8pc5 by Molmil
H3K36me3 nucleosome-LEDGF/p75 PWWP domain complex
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-09
公開日2023-08-16
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (3.02 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
8PEO
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BU of 8peo by Molmil
H3K36me2 nucleosome-LEDGF/p75 PWWP domain complex
分子名称: (2R)-2-amino-3-(2-dimethylaminoethylsulfanyl)propanoic acid, Histone H2A, Histone H2B 1.1, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-14
公開日2023-08-16
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (2.69 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
8PC6
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BU of 8pc6 by Molmil
H3K36me3 nucleosome-LEDGF/p75 PWWP domain complex - pose 2
分子名称: Histone H2A, Histone H2B 1.1, Histone H3, ...
著者Koutna, E, Kouba, T, Veverka, V.
登録日2023-06-09
公開日2023-08-16
最終更新日2023-11-15
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Multivalency of nucleosome recognition by LEDGF.
Nucleic Acids Res., 51, 2023
6SPF
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BU of 6spf by Molmil
Pseudomonas aeruginosa 70s ribosome from an aminoglycoside resistant clinical isolate
分子名称: 16S rRNA, 30S ribosomal protein S10, 30S ribosomal protein S11, ...
著者Halfon, Y, Jimenez-Fernande, A, La Ros, R, Espinos, R, Krogh Johansen, H, Matzov, D, Eyal, Z, Bashan, A, Zimmerman, E, Belousoff, M, Molin, S, Yonath, A.
登録日2019-09-01
公開日2019-10-23
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (2.89 Å)
主引用文献Structure ofPseudomonas aeruginosaribosomes from an aminoglycoside-resistant clinical isolate.
Proc.Natl.Acad.Sci.USA, 116, 2019

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