3TLM
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![BU of 3tlm by Molmil](/molmil-images/mine/3tlm) | Crystal Structure of Endoplasmic Reticulum Ca2+-ATPase (SERCA) From Bovine Muscle | Descriptor: | CALCIUM ION, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... | Authors: | Sacchetto, R, Bertipaglia, I, Giannetti, S, Cendron, L, Mascarello, F, Damiani, E, Carafoli, E, Zanotti, G. | Deposit date: | 2011-08-30 | Release date: | 2012-03-21 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.95 Å) | Cite: | Crystal structure of sarcoplasmic reticulum Ca(2+)-ATPase (SERCA) from bovine muscle. J.Struct.Biol., 178, 2012
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3HPE
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5M98
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5LL1
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8OI2
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![BU of 8oi2 by Molmil](/molmil-images/mine/8oi2) | Crystal structure of Alb1 megabody in complex with human serum albumin | Descriptor: | Alb1 Megabody, Albumin | Authors: | De Felice, S, Zoia, G, Romanyuk, Z, Pardon, E, Steyaert, J, Angelini, A, Cendron, L. | Deposit date: | 2023-03-22 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (3.3 Å) | Cite: | Crystal structure of human serum albumin in complex with megabody reveals unique human and murine cross-reactive binding site. Protein Sci., 33, 2024
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7ZRR
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![BU of 7zrr by Molmil](/molmil-images/mine/7zrr) | Crystal structure of human Urokinase-type plasminogen activator in complex with bicycle peptide inhibitor UK965 | Descriptor: | 1,2-ETHANEDIOL, 1,3,5-tris(bromomethyl)benzene, AMINO GROUP, ... | Authors: | Caregnato, A, Angela, P, Mazzoccato, Y, Frasson, N, Angelini, A, Cendron, L. | Deposit date: | 2022-05-05 | Release date: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.64 Å) | Cite: | Crystal structure of human Urokinase-type plasminogen activator in complex with bicycle peptide inhibitor UK965 To Be Published
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7ZRT
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![BU of 7zrt by Molmil](/molmil-images/mine/7zrt) | Crystal structure of human Urokinase-type plasminogen activator in complex with bicycle peptide inhibitor UK970 | Descriptor: | 1,2-ETHANEDIOL, 1,3,5-tris(bromomethyl)benzene, DI(HYDROXYETHYL)ETHER, ... | Authors: | Caregnato, A, Angela, P, Mazzoccato, Y, Frasson, N, Angelini, A, Cendron, L. | Deposit date: | 2022-05-05 | Release date: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Crystal structure of human Urokinase-type plasminogen activator in complex with bicycle peptide inhibitor UK970 To Be Published
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3ISL
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![BU of 3isl by Molmil](/molmil-images/mine/3isl) | Crystal structure of ureidoglycine-glyoxylate aminotransferase (pucG) from Bacillus subtilis | Descriptor: | PYRIDOXAL-5'-PHOSPHATE, Purine catabolism protein pucG | Authors: | Costa, R, Cendron, L, Ramazzina, I, Berni, R, Peracchi, A, Percudani, R, Zanotti, G. | Deposit date: | 2009-08-26 | Release date: | 2010-09-15 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.06 Å) | Cite: | Amino acids from purines in GUT bacteria To be Published
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3IBX
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![BU of 3ibx by Molmil](/molmil-images/mine/3ibx) | Crystal structure of F47Y variant of TenA (HP1287) from Helicobacter pylori | Descriptor: | Putative thiaminase II | Authors: | Barison, N, Cendron, L, Trento, A, Angelini, A, Zanotti, G. | Deposit date: | 2009-07-17 | Release date: | 2009-11-17 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Structural and mutational analysis of TenA protein (HP1287) from the Helicobacter pylori thiamin salvage pathway - evidence of a different substrate specificity. Febs J., 276, 2009
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7BN7
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![BU of 7bn7 by Molmil](/molmil-images/mine/7bn7) | Crystal structure of ene-reductase OYE2 from S. cerevisiae | Descriptor: | FLAVIN MONONUCLEOTIDE, GLYCEROL, OYE2 isoform 1 | Authors: | Robescu, M.S, Bergantino, E, Hall, M, Cendron, L. | Deposit date: | 2021-01-21 | Release date: | 2022-07-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.45 Å) | Cite: | Asymmetric Proton Transfer Catalysis by Stereocomplementary Old Yellow Enzymes for C=C Bond Isomerization Reaction Acs Catalysis, 12, 2022
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7BO0
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![BU of 7bo0 by Molmil](/molmil-images/mine/7bo0) | Crystal structure of ene-reductase GsOYE from Galdieria sulphuraria in complex with alpha-angelica lactone | Descriptor: | 5-methyl-3~{H}-furan-2-one, FLAVIN MONONUCLEOTIDE, NADPH2 dehydrogenase-like protein | Authors: | Robescu, M.S, Bergantino, E, Hall, M, Cendron, L. | Deposit date: | 2021-01-23 | Release date: | 2022-07-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.63 Å) | Cite: | Asymmetric Proton Transfer Catalysis by Stereocomplementary Old Yellow Enzymes for C=C Bond Isomerization Reaction Acs Catalysis, 12, 2022
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7BN6
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![BU of 7bn6 by Molmil](/molmil-images/mine/7bn6) | Crystal structure of G. sulphuraria ene-reductase GsOYE in complex with b-angelica lactone | Descriptor: | (2~{R})-2-methyl-2~{H}-furan-5-one, FLAVIN MONONUCLEOTIDE, NADPH2 dehydrogenase-like protein | Authors: | Robescu, M.S, Bergantino, E, Hall, M, Cendron, L. | Deposit date: | 2021-01-21 | Release date: | 2022-07-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.5 Å) | Cite: | Asymmetric Proton Transfer Catalysis by Stereocomplementary Old Yellow Enzymes for C=C Bond Isomerization Reaction Acs Catalysis, 12, 2022
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7BLF
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![BU of 7blf by Molmil](/molmil-images/mine/7blf) | Crystal structure of ene-reductase OYE4 from Botryotinia fuckeliana (BfOYE4) | Descriptor: | FLAVIN MONONUCLEOTIDE, FORMIC ACID, Oxidored_FMN domain-containing protein | Authors: | Robescu, M.S, Bergantino, E, Hall, M, Cendron, L. | Deposit date: | 2021-01-18 | Release date: | 2022-07-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.15 Å) | Cite: | Asymmetric Proton Transfer Catalysis by Stereocomplementary Old Yellow Enzymes for C=C Bond Isomerization Reaction Acs Catalysis, 12, 2022
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5LL7
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![BU of 5ll7 by Molmil](/molmil-images/mine/5ll7) | Crystal structure of KPC-2 carbapenemase in complex with a phenyl boronic inhibitor. | Descriptor: | (~{E})-3-[2-(dihydroxyboranyl)phenyl]prop-2-enoic acid, 1,2-ETHANEDIOL, Beta-lactamase | Authors: | Vicario, M, Celenza, G, Bellio, P, Perilli, M.G, Tondi, D, Cendron, L. | Deposit date: | 2016-07-26 | Release date: | 2018-02-21 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance. Chemmedchem, 13, 2018
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5MGI
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![BU of 5mgi by Molmil](/molmil-images/mine/5mgi) | Crystal structure of KPC-2 carbapenemase in complex with a phenyl boronic inhibitor. | Descriptor: | (~{E})-3-[2-(dihydroxyboranyl)phenyl]prop-2-enoic acid, Carbapenem-hydrolyzing beta-lactamase KPC | Authors: | Vicario, M, Celenza, G, Bellio, P, Perilli, M.G, Tondi, D, Cendron, L. | Deposit date: | 2016-11-21 | Release date: | 2018-03-14 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.5 Å) | Cite: | Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance. Chemmedchem, 13, 2018
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6TGD
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![BU of 6tgd by Molmil](/molmil-images/mine/6tgd) | Crystal structure of NDM-1 in complex with triazole-based inhibitor OP31 | Descriptor: | 4-[[(2~{S})-oxolan-2-yl]methyl]-3-pyridin-3-yl-1~{H}-1,2,4-triazole-5-thione, CALCIUM ION, Metallo-beta-lactamase NDM-1, ... | Authors: | Maso, L, Spirakis, F, Santucci, M, Simon, C, Docquier, J.D, Cruciani, G, Costi, M.P, Tondi, D, Cendron, L. | Deposit date: | 2019-11-15 | Release date: | 2020-08-26 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.33 Å) | Cite: | Virtual screening identifies broad-spectrum beta-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases. Sci Rep, 10, 2020
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6TGI
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![BU of 6tgi by Molmil](/molmil-images/mine/6tgi) | Crystal structure of VIM-2 in complex with triazole-based inhibitor OP24 | Descriptor: | 5-(4-chloranyl-1,5-dimethyl-pyrazol-3-yl)-4-ethyl-1,2,4-triazole-3-thiol, FORMIC ACID, Vim-1, ... | Authors: | Maso, L, Spirakis, F, Santucci, M, Simon, C, Docquier, J.D, Cruciani, G, Costi, M.P, Tondi, D, Cendron, L. | Deposit date: | 2019-11-15 | Release date: | 2020-10-14 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Virtual screening identifies broad-spectrum beta-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases. Sci Rep, 10, 2020
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4KZS
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![BU of 4kzs by Molmil](/molmil-images/mine/4kzs) | Crystal structure of the secreted protein HP1454 from the human pathogen Helicobacter pylori | Descriptor: | LPP20 lipofamily protein, PENTAETHYLENE GLYCOL | Authors: | Quarantini, S, Cendron, L, Fischer, W, Zanotti, G. | Deposit date: | 2013-05-30 | Release date: | 2014-06-04 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Crystal structure of the secreted protein HP1454 from the human pathogen Helicobacter pylori. Proteins, 82, 2014
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4LS3
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![BU of 4ls3 by Molmil](/molmil-images/mine/4ls3) | THE crystal STRUCTURE OF HELICOBACTER PYLORI CEUE(HP1561)/NI-HIS COMPL | Descriptor: | HISTIDINE, NICKEL (II) ION, Nickel (III) ABC transporter, ... | Authors: | Salamina, M, Shaik, M.M, Cendron, L, Zanotti, G. | Deposit date: | 2013-07-22 | Release date: | 2014-01-22 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Helicobacter pylori periplasmic receptor CeuE (HP1561) modulates its nickel affinity via organic metallophores. Mol.Microbiol., 91, 2014
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4INP
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![BU of 4inp by Molmil](/molmil-images/mine/4inp) | The crystal structure of Helicobacter pylori Ceue (HP1561) with Ni(II) bound | Descriptor: | ACETATE ION, Iron (III) ABC transporter, periplasmic iron-binding protein, ... | Authors: | Shaik, M.M, Cendron, L, Zanotti, G. | Deposit date: | 2013-01-05 | Release date: | 2014-01-08 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Helicobacter pylori periplasmic receptor CeuE (HP1561) modulates its nickel affinity via organic metallophores. Mol.Microbiol., 91, 2014
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4INO
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4INN
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![BU of 4inn by Molmil](/molmil-images/mine/4inn) | Protein HP1028 from the human pathogen Helicobacter pylori belongs to the lipocalin family | Descriptor: | 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, HP1028 | Authors: | Barison, N, Cendron, L, Loconte, V, Zanotti, G. | Deposit date: | 2013-01-05 | Release date: | 2013-07-31 | Last modified: | 2014-02-05 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Protein HP1028 from the human pathogen Helicobacter pylori belongs to the lipocalin family. Acta Crystallogr.,Sect.D, 69, 2013
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3BT0
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![BU of 3bt0 by Molmil](/molmil-images/mine/3bt0) | Crystal structure of transthyretin variant V20S | Descriptor: | Transthyretin | Authors: | Zanotti, G, Folli, C, Cendron, L, Gliubich, F, Negro, A, Berni, R. | Deposit date: | 2007-12-27 | Release date: | 2008-11-11 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (1.59 Å) | Cite: | Structural and mutational analyses of protein-protein interactions between transthyretin and retinol-binding protein. Febs J., 275, 2008
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2H6U
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![BU of 2h6u by Molmil](/molmil-images/mine/2h6u) | Crystal structure of 5-hydroxyisourate hydrolase (formerly known as TRP, transthyretin related protein) | Descriptor: | 5-HYDROXYISOURATE HYDROLASE (FORMERLY KNOWN AS TRP, TRANSTHYRETIN RELATED PROTEIN) | Authors: | Zanotti, G, Cendron, L, Folli, C, Ramazzina, I, Percudani, R, Berni, R. | Deposit date: | 2006-06-01 | Release date: | 2006-10-31 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Structure of Zebra fish HIUase: Insights into Evolution of an Enzyme to a Hormone Transporter. J.Mol.Biol., 363, 2006
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2H1X
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![BU of 2h1x by Molmil](/molmil-images/mine/2h1x) | Crystal structure of 5-hydroxyisourate Hydrolase (formerly known as TRP, Transthyretin Related Protein) | Descriptor: | 5-hydroxyisourate Hydrolase (formerly known as TRP, Transthyretin Related Protein) | Authors: | Zanotti, G, Cendron, L, Folli, C, Ramazzina, I, Percudani, R, Berni, R. | Deposit date: | 2006-05-17 | Release date: | 2006-10-31 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (1.98 Å) | Cite: | Structure of Zebra fish HIUase: Insights into Evolution of an Enzyme to a Hormone Transporter. J.Mol.Biol., 363, 2006
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