3G4K
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![BU of 3g4k by Molmil](/molmil-images/mine/3g4k) | Crystal structure of human phosphodiesterase 4d with rolipram | Descriptor: | 1,2-ETHANEDIOL, MAGNESIUM ION, ROLIPRAM, ... | Authors: | Staker, B.L. | Deposit date: | 2009-02-03 | Release date: | 2010-01-19 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Design of phosphodiesterase 4D (PDE4D) allosteric modulators for enhancing cognition with improved safety. Nat.Biotechnol., 28, 2010
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3FUK
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![BU of 3fuk by Molmil](/molmil-images/mine/3fuk) | |
3FTZ
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![BU of 3ftz by Molmil](/molmil-images/mine/3ftz) | Leukotriene A4 hydrolase in complex with fragment 2-(pyridin-3-ylmethoxy)aniline | Descriptor: | 2-(pyridin-3-ylmethoxy)aniline, ACETATE ION, IMIDAZOLE, ... | Authors: | Davies, D.R. | Deposit date: | 2009-01-13 | Release date: | 2010-01-05 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Discovery of 4-[(2S)-2-{[4-(4-chlorophenoxy)phenoxy]methyl}-1-pyrrolidinyl]butanoic acid (DG-051) as a novel leukotriene A4 hydrolase inhibitor of leukotriene B4 biosynthesis. J.Med.Chem., 53, 2010
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3FU0
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![BU of 3fu0 by Molmil](/molmil-images/mine/3fu0) | |
3FUH
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![BU of 3fuh by Molmil](/molmil-images/mine/3fuh) | |
3FTX
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![BU of 3ftx by Molmil](/molmil-images/mine/3ftx) | Leukotriene A4 hydrolase in complex with dihydroresveratrol and bestatin | Descriptor: | 2-(3-AMINO-2-HYDROXY-4-PHENYL-BUTYRYLAMINO)-4-METHYL-PENTANOIC ACID, 5-[2-(4-hydroxyphenyl)ethyl]benzene-1,3-diol, ACETATE ION, ... | Authors: | Davies, D.R. | Deposit date: | 2009-01-13 | Release date: | 2009-07-28 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.96 Å) | Cite: | Discovery of leukotriene A4 hydrolase inhibitors using metabolomics biased fragment crystallography. J.Med.Chem., 52, 2009
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3FUI
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![BU of 3fui by Molmil](/molmil-images/mine/3fui) | |
3FU5
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![BU of 3fu5 by Molmil](/molmil-images/mine/3fu5) | |
3FUJ
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![BU of 3fuj by Molmil](/molmil-images/mine/3fuj) | |
3FTV
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![BU of 3ftv by Molmil](/molmil-images/mine/3ftv) | |
3FUM
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![BU of 3fum by Molmil](/molmil-images/mine/3fum) | |
3G45
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![BU of 3g45 by Molmil](/molmil-images/mine/3g45) | |
3G4G
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![BU of 3g4g by Molmil](/molmil-images/mine/3g4g) | |
3IAD
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![BU of 3iad by Molmil](/molmil-images/mine/3iad) | |
3FH5
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![BU of 3fh5 by Molmil](/molmil-images/mine/3fh5) | |
3FHE
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![BU of 3fhe by Molmil](/molmil-images/mine/3fhe) | |