6T6F

Crystal structure of human calmodulin-dependent protein kinase 1D (CAMK1D) bound to compound 8 (CS275)

Summary for 6T6F

• Entry DOI: 10.2210/pdb6t6f/pdb
• Related: 6T28 6T29
• Descriptor: Calcium/calmodulin-dependent protein kinase type 1D, 2-[(3~{S})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide (3 entities in total)
• Functional Keywords: inhibitor, complex, kinase, structural genomics, structural genomics consortium, sgc, transferase
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 2
• Total formula weight: 74158.70

Authors

Sorrell, F.,Kraemer, A.,Butterworth, S.,Edwards, A.M.,Arrowsmith, C.H.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2019-10-18, release date: 2020-01-15, Last modification date: 2024-01-24)

• Primary citation: Sorrell, F.,Kraemer, A.,Butterworth, S.,Edwards, A.M.,Arrowsmith, C.H.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC); CAMK1D bound to CS275; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.97 Å)