6P3A
Crystal Structure Analysis of TAF1 Bromodomain
Summary for 6P3A
Entry DOI | 10.2210/pdb6p3a/pdb |
Descriptor | Transcription initiation factor TFIID subunit 1, 4-{[(3R)-1-(but-3-en-1-yl)-3-methyl-4-(oxan-4-yl)-2-oxo-1,2,3,4-tetrahydropyrido[2,3-b]pyrazin-6-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide (3 entities in total) |
Functional Keywords | kinase, bromodomain, inhibitor, transcription, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 32891.03 |
Authors | Seo, H.-S.,Dhe-Paganon, S. (deposition date: 2019-05-23, release date: 2020-05-27, Last modification date: 2023-10-11) |
Primary citation | Seo, H.-S.,Dhe-Paganon, S. Crystal Structure Analysis of TAF1 Bromodomain To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.99 Å) |
Structure validation
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