5YL4
CRYSTAL STRUCTURE OF T2R-TTL-8WR COMPLEX
Summary for 5YL4
Entry DOI | 10.2210/pdb5yl4/pdb |
Related | 5XHC 5XI5 5XI7 |
Descriptor | Tubulin alpha chain, (3Z,6Z)-3-[(4-tert-butyl-1H-imidazol-5-yl)methylidene]-6-[[3-(phenylcarbonyl)phenyl]methylidene]piperazine-2,5-dione, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... (12 entities in total) |
Functional Keywords | tubulin, microtubule, colchicine, diketopiperazine, structural protein |
Biological source | Rattus norvegicus (Rat) More |
Cellular location | Cytoplasm, cytoskeleton : A0A0R4I993 A0A0R4I995 Golgi apparatus : P63043 |
Total number of polymer chains | 6 |
Total formula weight | 264871.35 |
Authors | |
Primary citation | Fu, Z.Y.,Li, W.B. Design, synthesis and biological activity evaluation of plinabulin derivatives based on co-crystal structure To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.64 Å) |
Structure validation
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