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5JBT

Mesotrypsin in complex with cleaved amyloid precursor like protein 2 inhibitor (APLP2)

Summary for 5JBT
Entry DOI10.2210/pdb5jbt/pdb
DescriptorPRSS3 protein, Amyloid-like protein 2, CALCIUM ION, ... (6 entities in total)
Functional Keywordsinhibitor protease serine, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains3
Total formula weight30299.41
Authors
Kayode, O.,Wang, R.,Pendlebury, D.,Soares, A.,Radisky, E.S. (deposition date: 2016-04-13, release date: 2016-11-09, Last modification date: 2023-09-27)
Primary citationKayode, O.,Wang, R.,Pendlebury, D.F.,Cohen, I.,Henin, R.D.,Hockla, A.,Soares, A.S.,Papo, N.,Caulfield, T.R.,Radisky, E.S.
An Acrobatic Substrate Metamorphosis Reveals a Requirement for Substrate Conformational Dynamics in Trypsin Proteolysis.
J. Biol. Chem., 291:26304-26319, 2016
Cited by
PubMed: 27810896
DOI: 10.1074/jbc.M116.758417
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.4 Å)
Structure validation

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