Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5FZB

Crystal structure of the catalytic domain of human JARID1B in complex with Maybridge fragment 4-Pyridylthiourea (N06275b) (ligand modelled based on PANDDA event map, SGC - Diamond I04-1 fragment screening)

5FZB の概要
エントリーDOI10.2210/pdb5fzb/pdb
関連するPDBエントリー5FYB 5FYC 5FYH 5FYI 5FYM 5FYS 5FYT 5FYU 5FYV 5FYY 5FYZ 5FZ0 5FZ1 5FZ3 5FZ4 5FZ6 5FZ7 5FZ8 5FZ9 5FZA 5FZC 5FZD 5FZE 5FZF 5FZG 5FZH 5FZI 5FZK 5FZL 5FZM 5FZO
分子名称LYSINE-SPECIFIC DEMETHYLASE 5B, ZINC ION, DIMETHYL SULFOXIDE, ... (10 entities in total)
機能のキーワードoxidoreductase, jarid1b, plu1, fragment screening, structural genomics consortium, sgc, diamond i04-1, pandda
由来する生物種HOMO SAPIENS (HUMAN)
細胞内の位置Nucleus : Q9UGL1
タンパク質・核酸の鎖数1
化学式量合計56683.80
構造登録者
主引用文献Nowak, R.,Krojer, T.,Johansson, C.,Kupinska, K.,Szykowska, A.,Pearce, N.,Talon, R.,Collins, P.,Gileadi, C.,Strain-Damerell, C.,Burgess-Brown, N.A.,Arrowsmith, C.H.,Bountra, C.,Edwards, A.M.,von Delft, F.,Brennan, P.E.,Oppermann, U.
Crystal Structure of the Catalytic Domain of Human Jarid1B in Complex with Maybridge Fragment 4-Pyridylthiourea (N06275B) (Ligand Modelled Based on Pandda Event Map, Sgc -Diamond I04-1 Fragment Screening)
To be Published,
実験手法
X-RAY DIFFRACTION (2.18 Å)
構造検証レポート
Validation report summary of 5fzb
検証レポート(詳細版)ダウンロードをダウンロード

217705

件を2024-03-27に公開中

PDB statisticsPDBj update infoContact PDBjnumon