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5BNM

E. coli FabH with Small Molecule Inhibitor 1

Summary for 5BNM
Entry DOI10.2210/pdb5bnm/pdb
Related5BNR 5BNS 5BQS
Descriptor3-oxoacyl-[acyl-carrier-protein] synthase 3, SULFATE ION, N-{[3'-(hydroxymethyl)biphenyl-4-yl]methyl}benzenesulfonamide, ... (5 entities in total)
Functional Keywordsfabh, fatty acid synthesis, bacterial enzyme, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceEscherichia coli
Cellular locationCytoplasm : P0A6R0
Total number of polymer chains2
Total formula weight67737.78
Authors
Kazmirski, S.L.,McKinney, D.C. (deposition date: 2015-05-26, release date: 2016-05-18, Last modification date: 2024-03-06)
Primary citationMcKinney, D.C.,Eyermann, C.J.,Gu, R.F.,Hu, J.,Kazmirski, S.L.,Lahiri, S.D.,McKenzie, A.R.,Shapiro, A.B.,Breault, G.
Antibacterial FabH Inhibitors with Mode of Action Validated in Haemophilus influenzae by in Vitro Resistance Mutation Mapping.
Acs Infect Dis., 2:456-464, 2016
Cited by
PubMed: 27626097
DOI: 10.1021/acsinfecdis.6b00053
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

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