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4F1Q

Human Artd8 (Parp14, Bal2) - catalytic domain in complex with A16(E)

Summary for 4F1Q
Entry DOI10.2210/pdb4f1q/pdb
Related3GOY 3SE2 3SMI 3SMJ 4F1L
DescriptorPoly [ADP-ribose] polymerase 14, (2E)-4-[(3-carbamoylphenyl)amino]-4-oxobut-2-enoic acid, NITRATE ION (3 entities in total)
Functional Keywordsnad, adp-ribose, parp14, bal2, artd8, artd transferase domain, adp-ribose transferase, adp-ribosylation, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Cellular locationNucleus: Q460N5
Total number of polymer chains2
Total formula weight44767.60
Authors
Karlberg, T.,Andersson, C.D.,Lindgren, A.,Spjut, S.,Thorsell, A.G.,Ekblad, T.,Weigelt, J.,Elofsson, M.,Linusson, A.,Schuler, H. (deposition date: 2012-05-07, release date: 2012-09-05, Last modification date: 2023-09-13)
Primary citationAndersson, C.D.,Karlberg, T.,Ekblad, T.,Lindgren, A.E.,Thorsell, A.G.,Spjut, S.,Uciechowska, U.,Niemiec, M.S.,Wittung-Stafshede, P.,Weigelt, J.,Elofsson, M.,Schuler, H.,Linusson, A.
Discovery of Ligands for ADP-Ribosyltransferases via Docking-Based Virtual Screening.
J.Med.Chem., 55:7706-7718, 2012
Cited by
PubMed: 22823910
DOI: 10.1021/jm300746d
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.8 Å)
Structure validation

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