4E7R
Thrombin in complex with 3-amidinophenylalanine inhibitor
Summary for 4E7R
Entry DOI | 10.2210/pdb4e7r/pdb |
Related | 3F68 3QWC 3QX5 |
Descriptor | Thrombin light chain, Thrombin heavy chain, Hirudin variant-2, ... (9 entities in total) |
Functional Keywords | hydrolase-hydrolase inhibitor complex, serine protease, kringle, hydrolase, blood coagulation, blood clotting, convertion of fibrinogen to fibrin, blood clotting inhibitor, thrombin inhibitor, glycosylation, blood, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 6 |
Total formula weight | 72942.31 |
Authors | Ruehmann, E.,Heine, A.,Klebe, G. (deposition date: 2012-03-19, release date: 2012-06-20, Last modification date: 2023-12-06) |
Primary citation | Hammami, M.,Ruehmann, E.,Mauerer, M.,Heine, A.,Guetschow, M.,Klebe, G.,Steinmetzer, T. New 3-amidinophenylalanine-derived inhibitors of matriptase MEDCHEMCOMM, 3:807-813, 2012 Cited by DOI: 10.1039/C2MD20074KPDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.25 Å) |
Structure validation
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