4JYG
Crystal structure of RARbeta LBD in complex with agonist BMS411 [4-{[(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)carbonyl]amino}benzoic acid]
Summary for 4JYG
Entry DOI | 10.2210/pdb4jyg/pdb |
Related | 1XAP 4DM6 4DM8 4JYH 4JYI |
Descriptor | Retinoic acid receptor beta, Steroid Receptor Coactivator 1, 4-{[(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)carbonyl]amino}benzoic acid, ... (6 entities in total) |
Functional Keywords | ligand binding domain, nuclear hormone receptor, transcription-agonist complex, transcription/agonist |
Biological source | Homo sapiens (human) More |
Cellular location | Isoform Beta-1: Nucleus. Isoform Beta-2: Nucleus. Isoform Beta-4: Cytoplasm: P10826 Nucleus : Q15788 |
Total number of polymer chains | 4 |
Total formula weight | 64916.23 |
Authors | Nadendla, E.K.,Teyssier, C.,Germain, P.,Delfosse, V.,Bourguet, W. (deposition date: 2013-03-29, release date: 2014-03-19, Last modification date: 2024-02-28) |
Primary citation | Nadendla, E.,Teyssier, C.,Delfosse, V.,Vivat, V.,Krishnasamy, G.,Gronemeyer, H.,Bourguet, W.,Germain, P. An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor beta (RAR beta , NR1B2) Selective Agonist. Plos One, 10:e0123195-e0123195, 2015 Cited by PubMed: 25933005DOI: 10.1371/journal.pone.0123195 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.35 Å) |
Structure validation
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