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4JYG

Crystal structure of RARbeta LBD in complex with agonist BMS411 [4-{[(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)carbonyl]amino}benzoic acid]

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0048384biological_processretinoic acid receptor signaling pathway
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
B0048384biological_processretinoic acid receptor signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 1NY A 501
ChainResidue
APHE221
AGLY384
AHOH716
AALA225
ALEU262
AILE266
AARG269
APHE279
ASER280
APHE295
AVAL302

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PE4 B 501
ChainResidue
AGLU273
BARG212
BLEU213
BLEU215
BHOH645
BHOH648

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 1NY B 502
ChainResidue
BPHE192
BTRP218
BPHE221
BALA225
BCYS228
BLEU262
BILE266
BARG269
BPHE279
BSER280
BVAL302
BLEU391
BHOH629

site_idAC4
Number of Residues10
DetailsBINDING SITE FOR RESIDUE FLC G 701
ChainResidue
AGLU337
APRO338
ATHR339
GHIS630
GLYS631
GILE632
GARG635
GHOH804
GHOH807
GHOH808

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
FSER641
GSER641

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PDB entries from 2025-06-18

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