3HUB
Human p38 MAP Kinase in Complex with Scios-469
3HUB の概要
エントリーDOI | 10.2210/pdb3hub/pdb |
関連するPDBエントリー | 3GCP 3GCQ 3GCS 3GCU 3GCV 3HUC |
分子名称 | Mitogen-activated protein kinase 14, octyl beta-D-glucopyranoside, 2-(6-chloro-5-{[(2R,5S)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide, ... (4 entities in total) |
機能のキーワード | dfg-in, glycine-rich loop, scios-469, alternative splicing, atp-binding, cytoplasm, kinase, nucleotide-binding, nucleus, phosphoprotein, polymorphism, serine/threonine-protein kinase, transferase |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 42040.35 |
構造登録者 | |
主引用文献 | Simard, J.R.,Getlik, M.,Grutter, C.,Schneider, R.,Wulfert, S.,Rauh, D. Fluorophore labeling of the glycine-rich loop as a method of identifying inhibitors that bind to active and inactive kinase conformations. J.Am.Chem.Soc., 132:4152-4160, 2010 Cited by PubMed: 20201574DOI: 10.1021/ja908083e 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.25 Å) |
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