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3ADU

Human PPARgamma ligand-binding domain in complex with 5-methoxy-indole acetate

Summary for 3ADU
Entry DOI10.2210/pdb3adu/pdb
Related3ADS 3ADT 3ADV 3ADW 3ADX
DescriptorPeroxisome proliferator-activated receptor gamma, (5-methoxy-1H-indol-3-yl)acetic acid (3 entities in total)
Functional Keywordsnuclear receptor, ligand-dependent transcription factor, ligand-binding domain, activator, diabetes mellitus, disease mutation, dna-binding, metal-binding, nucleus, obesity, phosphoprotein, receptor, transcription, transcription regulation, zinc-finger
Biological sourceHomo sapiens (human)
Cellular locationNucleus: P37231
Total number of polymer chains2
Total formula weight66413.70
Authors
Waku, T.,Shiraki, T.,Oyama, T.,Morikawa, K. (deposition date: 2010-01-29, release date: 2010-12-22, Last modification date: 2023-11-01)
Primary citationWaku, T.,Shiraki, T.,Oyama, T.,Maebara, K.,Nakamori, R.,Morikawa, K.
The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites
Embo J., 29:3395-3407, 2010
Cited by
PubMed: 20717101
DOI: 10.1038/emboj.2010.197
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.77 Å)
Structure validation

217705

건을2024-03-27부터공개중

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