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3ADU

Human PPARgamma ligand-binding domain in complex with 5-methoxy-indole acetate

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE MYI A 1
ChainResidue
AMYI2
ACYS285
AARG288
ASER289
AILE326
ALEU330
ALEU333

site_idAC2
Number of Residues9
DetailsBINDING SITE FOR RESIDUE MYI A 2
ChainResidue
ASER289
AHIS323
AILE326
ATYR327
AMET364
AHIS449
ATYR473
AMYI1
APHE282

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MYI B 3
ChainResidue
BMYI4
BARG288
BILE326
BLEU333
BSER342
BHOH1017

site_idAC4
Number of Residues9
DetailsBINDING SITE FOR RESIDUE MYI B 4
ChainResidue
BMYI3
BILE281
BGLY284
BCYS285
BLEU330
BVAL339
BSER342
BMET348
BMET364

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MYI B 5
ChainResidue
BGLN286
BSER289
BHIS323
BTYR327
BHIS449

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
ChainResidueDetails
AGLN286
AHIS323
AHIS449
ATYR473
BGLN286
BHIS323
BHIS449
BTYR473

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224
BLYS224

218196

PDB entries from 2024-04-10

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