2ZZU
Human Factor VIIA-Tissue Factor Complexed with ethylsulfonamide-D-5-(3-carboxybenzyloxy)-Trp-Gln-p-aminobenzamidine
Summary for 2ZZU
Entry DOI | 10.2210/pdb2zzu/pdb |
Related | 1WQV 1WSS 1WTG 1WUN 1WV7 2ZWL |
Descriptor | Factor VII light chain, Factor VII heavy chain, Tissue factor, ... (8 entities in total) |
Functional Keywords | serine protease, blood coagulation, cleavage on pair of basic residues, disease mutation, egf-like domain, gamma-carboxyglutamic acid, glycoprotein, hydrolase, hydroxylation, protease, zymogen, lipoprotein, membrane, palmitate, transmembrane, hydrolase-blood clotting complex, secreted, hydrolase/blood clotting |
Biological source | Homo sapiens (Human) More |
Cellular location | Secreted: P08709 P08709 Isoform 1: Membrane; Single-pass type I membrane protein. Isoform 2: Secreted: P13726 |
Total number of polymer chains | 3 |
Total formula weight | 71698.53 |
Authors | Kadono, S.,Sakamoto, A.,Kikuchi, Y.,Oh-Eda, M.,Yabuta, N.,Koga, T.,Hattori, K.,Shiraishi, T.,Haramura, M.,Sato, H.,Ohta, M.,Kozono, T. (deposition date: 2009-02-25, release date: 2009-03-24, Last modification date: 2023-11-15) |
Primary citation | Shiraishi, T.,Kadono, S.,Haramura, M.,Kodama, H.,Ono, Y.,Iikura, H.,Esaki, T.,Koga, T.,Hattori, K.,Watanabe, Y.,Sakamoto, A.,Yoshihashi, K.,Kitazawa, T.,Esaki, K.,Ohta, M.,Sato, H.,Kozono, T. Design and synthesis of peptidomimetic factor VIIa inhibitors Chem.Pharm.Bull., 58:38-44, 2010 Cited by PubMed: 20045964DOI: 10.1248/cpb.58.38 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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