2M3Z
NMR solution structure of HIV-1 nucleocapsid protein in complex with an inhibitor displaying a 2 inhibitors:1 NC stoichiometry
Summary for 2M3Z
Entry DOI | 10.2210/pdb2m3z/pdb |
Related | 1A1T 1F6U |
NMR Information | BMRB: 18980 |
Descriptor | NUCLEOCAPSID PROTEIN P7, ZINC ION, (3E)-3-{(2Z)-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-1,3-thiazolidin-2-ylidene]hydrazinylidene}-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid (3 entities in total) |
Functional Keywords | hiv-1 nc, viral protein |
Biological source | Human immunodeficiency virus type 1 (HIV-1) |
Cellular location | Matrix protein p17: Virion (Potential). Capsid protein p24: Virion (Potential). Nucleocapsid protein p7: Virion (Potential). Reverse transcriptase/ribonuclease H: Virion (Potential). Integrase: Virion (Potential): P12497 |
Total number of polymer chains | 1 |
Total formula weight | 7336.08 |
Authors | Goudreau, N.,Hucke, O. (deposition date: 2013-01-28, release date: 2013-02-27, Last modification date: 2024-05-15) |
Primary citation | Goudreau, N.,Hucke, O.,Faucher, A.M.,Grand-Maitre, C.,Lepage, O.,Bonneau, P.R.,Mason, S.W.,Titolo, S. Discovery and Structural Characterization of a New Inhibitor Series of HIV-1 Nucleocapsid Function: NMR Solution Structure Determination of a Ternary Complex Involving a 2:1 Inhibitor/NC Stoichiometry. J.Mol.Biol., 425:1982-1998, 2013 Cited by PubMed: 23485336DOI: 10.1016/j.jmb.2013.02.022 PDB entries with the same primary citation |
Experimental method | SOLUTION NMR |
Structure validation
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