1W8B
Factor7 - 413 complex
Summary for 1W8B
Entry DOI | 10.2210/pdb1w8b/pdb |
Related | 1BF9 1CVW 1DAN 1DVA 1F7E 1F7M 1FAK 1FF7 1FFM 1J9C 1JBU 1KLI 1KLJ 1NL8 1QFK 1W0Y 1W2K 1W7X |
Descriptor | BLOOD COAGULATION FACTOR VIIA, CALCIUM ION, (S)-[(R)-2-(4-BENZYLOXY-3-METHOXY-PHENYL)-2-(4-CARBAMIMIDOYL-PHENYLAMINO)-ACETYLAMINO]-PHENYL-ACETIC ACID, ... (5 entities in total) |
Functional Keywords | serine protease, coagulation, enzyme complex, hydrolase |
Biological source | HOMO SAPIENS (HUMAN) More |
Cellular location | Secreted: P08709 P08709 |
Total number of polymer chains | 2 |
Total formula weight | 34954.04 |
Authors | Ackermann, J.,Alig, L.,Banner, D.W.,Boehm, H.-J.,Groebke-Zbinden, K.,Hilpert, K.,Lave, T.,Kuehne, H.,Obst-Sander, U.,Riederer, M.A.,Stahl, M.,Tschopp, T.B.,Weber, L.,Wessel, H.P. (deposition date: 2004-09-17, release date: 2005-10-25, Last modification date: 2023-12-13) |
Primary citation | Groebke-Zbinden, K.,Obst-Sander, U.,Hilpert, K.,Kuehne, H.,Banner, D.W.,Boehm, H.-J.,Stahl, M.,Ackermann, J.,Alig, L.,Weber, L.,Wessel, H.P.,Riederer, M.A.,Tschopp, T.B.,Lave, T. Selective and Orally Bioavailable Phenylglycine Tissue Factor/Factor Viia Inhibitors Bioorg.Med.Chem.Lett., 15:5344-, 2005 Cited by PubMed: 16213138DOI: 10.1016/J.BMCL.2005.04.079 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3 Å) |
Structure validation
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