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1QKU

WILD TYPE ESTROGEN NUCLEAR RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH ESTRADIOL

Summary for 1QKU
Entry DOI10.2210/pdb1qku/pdb
Related1A52 1AKF 1ERE 1ERR 1HCP 1HCQ 1QKM 1QKN 1QKU 3ERD 3ERT
DescriptorESTRADIOL RECEPTOR, ESTRADIOL (3 entities in total)
Functional Keywordsnuclear receptor, agonism, antagonism, estradiol receptor, steroid, structural proteomics in europe, spine, structural genomics
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationIsoform 1: Nucleus . Isoform 3: Nucleus. Nucleus: P03372
Total number of polymer chains3
Total formula weight86676.33
Authors
Ruff, M.,Gangloff, M.,Eiler, S.,Duclaud, S.,Wurtz, J.M.,Moras, D. (deposition date: 1999-08-05, release date: 2000-08-18, Last modification date: 2018-02-28)
Primary citationGangloff, M.,Ruff, M.,Eiler, S.,Duclaud, S.,Wurtz, J.M.,Moras, D.
Crystal structure of a mutant hERalpha ligand-binding domain reveals key structural features for the mechanism of partial agonism.
J. Biol. Chem., 276:15059-15065, 2001
Cited by
PubMed: 11278577
DOI: 10.1074/jbc.M009870200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3.2 Å)
Structure validation

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