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1QKU

WILD TYPE ESTROGEN NUCLEAR RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH ESTRADIOL

Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE EST A 600
ChainResidue
AGLU353
ALEU525
ALEU387
AMET388
AARG394
APHE404
AMET421
AILE424
AGLY521
AHIS524

site_idAC2
Number of Residues11
DetailsBINDING SITE FOR RESIDUE EST B 600
ChainResidue
BGLU353
BLEU387
BMET388
BLEU391
BARG394
BPHE404
BMET421
BILE424
BGLY521
BHIS524
BLEU525

site_idAC3
Number of Residues11
DetailsBINDING SITE FOR RESIDUE EST C 600
ChainResidue
CGLU353
CLEU387
CMET388
CLEU391
CARG394
CPHE404
CMET421
CILE424
CGLY521
CHIS524
CLEU525

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537
BTYR537
CTYR537

site_idSWS_FT_FI2
Number of Residues3
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447
CCYS447

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PDB entries from 2024-04-24

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