7UMB
NanoBRET tracer Tram-bo bound to a KSR2-MEK1 complex
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | B | Kinase suppressor of Ras 2 | polymer | 342 | 39748.7 | 1 | UniProt (Q6VAB6) Pfam (PF07714) In PDB | Homo sapiens (human) | hKSR2 |
2 | C | Dual specificity mitogen-activated protein kinase kinase 1 | polymer | 384 | 43119.4 | 1 | UniProt (Q02750) Pfam (PF00069) In PDB | Homo sapiens (human) | |
3 | B, C | PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER | non-polymer | 506.2 | 2 | Chemie (ANP) | |||
4 | C | {3-[(1M,2M)-2-{[(1S,2P)-1H,1'H-[2,2'-bipyrrol]-5-yl-kappaN~1~]methylidene}-2H-pyrrol-5-yl-kappaN]-N-(2-{2-[3-({(3M)-3-[(4aM)-3-cyclopropyl-5-(2-fluoro-4-iodoanilino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7-tetrahydropyrido[4,3-d]pyrimidin-1(2H)-yl]phenyl}amino)-3-oxopropoxy]ethoxy}ethyl)propanamidato}(difluorido)boron | non-polymer | 1043.6 | 1 | Chemie (U9F) |
Sequence modifications
B: 634 - 950 (UniProt: Q6VAB6)
C: 35 - 393 (UniProt: Q02750)
PDB | External Database | Details |
---|---|---|
Met 609 | - | initiating methionine |
Ser 610 | - | expression tag |
Tyr 611 | - | expression tag |
Tyr 612 | - | expression tag |
His 613 | - | expression tag |
His 614 | - | expression tag |
His 615 | - | expression tag |
His 616 | - | expression tag |
His 617 | - | expression tag |
His 618 | - | expression tag |
Asp 619 | - | expression tag |
Tyr 620 | - | expression tag |
Asp 621 | - | expression tag |
Ile 622 | - | expression tag |
Pro 623 | - | expression tag |
Thr 624 | - | expression tag |
Thr 625 | - | expression tag |
Glu 626 | - | expression tag |
Asn 627 | - | expression tag |
Leu 628 | - | expression tag |
Tyr 629 | - | expression tag |
Phe 630 | - | expression tag |
Gln 631 | - | expression tag |
Gly 632 | - | expression tag |
Ala 633 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Met 10 | - | initiating methionine |
Ser 11 | - | expression tag |
Tyr 12 | - | expression tag |
Tyr 13 | - | expression tag |
His 14 | - | expression tag |
His 15 | - | expression tag |
His 16 | - | expression tag |
His 17 | - | expression tag |
His 18 | - | expression tag |
His 19 | - | expression tag |
Asp 20 | - | expression tag |
Tyr 21 | - | expression tag |
Asp 22 | - | expression tag |
Ile 23 | - | expression tag |
Pro 24 | - | expression tag |
Thr 25 | - | expression tag |
Thr 26 | - | expression tag |
Glu 27 | - | expression tag |
Asn 28 | - | expression tag |
Leu 29 | - | expression tag |
Tyr 30 | - | expression tag |
Phe 31 | - | expression tag |
Gln 32 | - | expression tag |
Gly 33 | - | expression tag |
Ala 34 | - | expression tag |
Ala 328 | Gly 328 | conflict |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 82868.1 | |
Non-Polymers* | Number of molecules | 3 |
Total formula weight | 2056.0 | |
All* | Total formula weight | 84924.1 |