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7API
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BU of 7api by Molmil
THE S VARIANT OF HUMAN ALPHA1-ANTITRYPSIN, STRUCTURE AND IMPLICATIONS FOR FUNCTION AND METABOLISM
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ALPHA 1-ANTITRYPSIN, ...
Authors:Loebermann, H, Tokuoka, R, Deisenhofer, J, Huber, R.
Deposit date:1988-09-08
Release date:1990-10-15
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (3 Å)
Cite:The S variant of human alpha 1-antitrypsin, structure and implications for function and metabolism.
Protein Eng., 2, 1989
8API
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THE S VARIANT OF HUMAN ALPHA1-ANTITRYPSIN, STRUCTURE AND IMPLICATIONS FOR FUNCTION AND METABOLISM
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ALPHA-1 ANTITRYPSIN (CHAIN A), ...
Authors:Loebermann, H, Tokuoka, R, Deisenhofer, J, Huber, R.
Deposit date:1988-09-08
Release date:1990-10-15
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (3.1 Å)
Cite:The S variant of human alpha 1-antitrypsin, structure and implications for function and metabolism.
Protein Eng., 2, 1989
9API
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BU of 9api by Molmil
THE S VARIANT OF HUMAN ALPHA1-ANTITRYPSIN, STRUCTURE AND IMPLICATIONS FOR FUNCTION AND METABOLISM
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ALPHA 1-ANTITRYPSIN, ...
Authors:Loebermann, H, Tokuoka, R, Deisenhofer, J, Huber, R.
Deposit date:1988-09-08
Release date:1990-10-15
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (3 Å)
Cite:The S variant of human alpha 1-antitrypsin, structure and implications for function and metabolism.
Protein Eng., 2, 1989
1OVA
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BU of 1ova by Molmil
CRYSTAL STRUCTURE OF UNCLEAVED OVALBUMIN AT 1.95 ANGSTROMS RESOLUTION
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, OVALBUMIN
Authors:Stein, P.E, Leslie, A.G.W.
Deposit date:1990-11-26
Release date:1992-04-15
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Crystal structure of uncleaved ovalbumin at 1.95 A resolution.
J.Mol.Biol., 221, 1991
1HLE
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BU of 1hle by Molmil
CRYSTAL STRUCTURE OF CLEAVED EQUINE LEUCOCYTE ELASTASE INHIBITOR DETERMINED AT 1.95 ANGSTROMS RESOLUTION
Descriptor: CALCIUM ION, HORSE LEUKOCYTE ELASTASE INHIBITOR
Authors:Baumann, U, Bode, W, Huber, R, Travis, J, Potempa, J.
Deposit date:1992-04-13
Release date:1994-01-31
Last modified:2017-11-29
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Crystal structure of cleaved equine leucocyte elastase inhibitor determined at 1.95 A resolution.
J.Mol.Biol., 226, 1992
1ATT
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BU of 1att by Molmil
CRYSTAL STRUCTURE OF CLEAVED BOVINE ANTITHROMBIN III AT 3.2 ANGSTROMS RESOLUTION
Descriptor: ANTITHROMBIN III
Authors:Mourey, L, Samama, J.P, Delarue, M, Moras, D.
Deposit date:1993-03-29
Release date:1994-07-31
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:Crystal structure of cleaved bovine antithrombin III at 3.2 A resolution.
J.Mol.Biol., 232, 1993
2ACH
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BU of 2ach by Molmil
CRYSTAL STRUCTURE OF CLEAVED HUMAN ALPHA1-ANTICHYMOTRYPSIN AT 2.7 ANGSTROMS RESOLUTION AND ITS COMPARISON WITH OTHER SERPINS
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ALPHA 1-ANTICHYMOTRYPSIN, PHOSPHATE ION, ...
Authors:Baumann, U, Huber, R, Bode, W, Grosse, D, Lesjak, M, Laurell, C.B.
Deposit date:1993-04-26
Release date:1993-07-15
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Crystal structure of cleaved human alpha 1-antichymotrypsin at 2.7 A resolution and its comparison with other serpins.
J.Mol.Biol., 218, 1991
1ATH
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BU of 1ath by Molmil
THE INTACT AND CLEAVED HUMAN ANTITHROMBIN III COMPLEX AS A MODEL FOR SERPIN-PROTEINASE INTERACTIONS
Descriptor: ANTITHROMBIN III
Authors:Schreuder, H.A, Hol, W.G.J.
Deposit date:1993-12-14
Release date:1995-02-07
Last modified:2017-11-29
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:The intact and cleaved human antithrombin III complex as a model for serpin-proteinase interactions.
Nat.Struct.Biol., 1, 1994
1ANT
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BU of 1ant by Molmil
BIOLOGICAL IMPLICATIONS OF A 3 ANGSTROMS STRUCTURE OF DIMERIC ANTITHROMBIN
Descriptor: ANTITHROMBIN
Authors:Carrell, R.W, Stein, P.E, Fermi, G, Wardell, M.R.
Deposit date:1994-02-28
Release date:1995-01-26
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (3 Å)
Cite:Biological implications of a 3 A structure of dimeric antithrombin.
Structure, 2, 1994
1PSI
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BU of 1psi by Molmil
Intact recombined alpha1-antitrypsin mutant PHE 51 to LEU
Descriptor: ALPHA=1=-ANTITRYPSIN
Authors:Abrahams, J.P, Elliott, P.R, Lomas, D.A, Carrell, R.W.
Deposit date:1996-06-11
Release date:1996-12-07
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.92 Å)
Cite:Inhibitory conformation of the reactive loop of alpha 1-antitrypsin.
Nat.Struct.Biol., 3, 1996
1KCT
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BU of 1kct by Molmil
ALPHA1-ANTITRYPSIN
Descriptor: ALPHA1-ANTITRYPSIN
Authors:Song, H.K, Suh, S.W.
Deposit date:1996-08-06
Release date:1997-01-11
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (3.46 Å)
Cite:Crystal structure of an uncleaved alpha 1-antitrypsin reveals the conformation of its inhibitory reactive loop.
FEBS Lett., 377, 1995
2ANT
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BU of 2ant by Molmil
THE 2.6 A STRUCTURE OF ANTITHROMBIN INDICATES A CONFORMATIONAL CHANGE AT THE HEPARIN BINDING SITE
Descriptor: 2-acetamido-2-deoxy-beta-D-allopyranose, ANTITHROMBIN
Authors:Skinner, R, Abrahams, J.-P, Whisstock, J.C, Lesk, A.M, Carrell, R.W, Wardell, M.R.
Deposit date:1997-01-28
Release date:1997-06-16
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:The 2.6 A structure of antithrombin indicates a conformational change at the heparin binding site.
J.Mol.Biol., 266, 1997
1ATU
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BU of 1atu by Molmil
UNCLEAVED ALPHA-1-ANTITRYPSIN
Descriptor: ALPHA-1-ANTITRYPSIN
Authors:Ryu, S.-E, Choi, H.-J.
Deposit date:1997-05-11
Release date:1997-08-20
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:The native strains in the hydrophobic core and flexible reactive loop of a serine protease inhibitor: crystal structure of an uncleaved alpha1-antitrypsin at 2.7 A.
Structure, 4, 1996
1AS4
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BU of 1as4 by Molmil
CLEAVED ANTICHYMOTRYPSIN A349R
Descriptor: ACETATE ION, ANTICHYMOTRYPSIN
Authors:Lukacs, C.M, Christianson, D.W.
Deposit date:1997-08-12
Release date:1998-02-25
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction.
Biochemistry, 37, 1998
4CAA
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BU of 4caa by Molmil
CLEAVED ANTICHYMOTRYPSIN T345R
Descriptor: ANTICHYMOTRYPSIN
Authors:Lukacs, C.M, Christianson, D.W.
Deposit date:1997-08-14
Release date:1998-02-25
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction.
Biochemistry, 37, 1998
3CAA
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BU of 3caa by Molmil
CLEAVED ANTICHYMOTRYPSIN A347R
Descriptor: ANTICHYMOTRYPSIN
Authors:Lukacs, C.M, Christianson, D.W.
Deposit date:1997-08-18
Release date:1998-02-25
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction.
Biochemistry, 37, 1998
1AZX
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BU of 1azx by Molmil
ANTITHROMBIN/PENTASACCHARIDE COMPLEX
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,4-di-O-methyl-2,6-di-O-sulfo-alpha-D-glucopyranose-(1-4)-2,3-di-O-methyl-beta-D-glucopyranuronic acid-(1-4)-2,3,6-tri-O-sulfo-alpha-D-glucopyranose-(1-4)-3-O-methyl-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-methyl 2,3,6-tri-O-sulfo-alpha-D-glucopyranoside, ANTITHROMBIN
Authors:Jin, L, Abrahams, J.P, Skinner, R, Petitou, M, Pike, R.N, Carrell, R.W.
Deposit date:1997-11-23
Release date:1999-01-13
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:The anticoagulant activation of antithrombin by heparin.
Proc.Natl.Acad.Sci.USA, 94, 1997
1SEK
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BU of 1sek by Molmil
THE STRUCTURE OF ACTIVE SERPIN K FROM MANDUCA SEXTA AND A MODEL FOR SERPIN-PROTEASE COMPLEX FORMATION
Descriptor: SERPIN K
Authors:Li, J, Wang, Z, Canagarajah, B, Jiang, H, Kanost, M, Goldsmith, E.J.
Deposit date:1998-03-06
Release date:1999-03-23
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:The structure of active serpin 1K from Manduca sexta.
Structure Fold.Des., 7, 1999
1A7C
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BU of 1a7c by Molmil
HUMAN PLASMINOGEN ACTIVATOR INHIBITOR TYPE-1 IN COMPLEX WITH A PENTAPEPTIDE
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-D-ribopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, PENTAPEPTIDE, ...
Authors:Xue, Y, Inghardt, T, Sjolin, L, Deinum, J.
Deposit date:1998-03-12
Release date:1999-03-23
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Interfering with the inhibitory mechanism of serpins: crystal structure of a complex formed between cleaved plasminogen activator inhibitor type 1 and a reactive-centre loop peptide
Structure, 6, 1998
1BR8
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BU of 1br8 by Molmil
IMPLICATIONS FOR FUNCTION AND THERAPY OF A 2.9A STRUCTURE OF BINARY-COMPLEXED ANTITHROMBIN
Descriptor: PROTEIN (ANTITHROMBIN-III), PROTEIN (PEPTIDE)
Authors:Skinner, R, Chang, W.S.W, Jin, L, Pei, X.Y, Huntington, J.A, Abrahams, J.P, Carrell, R.W, Lomas, D.A.
Deposit date:1998-08-26
Release date:1998-09-02
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Implications for function and therapy of a 2.9 A structure of binary-complexed antithrombin.
J.Mol.Biol., 283, 1998
1BY7
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BU of 1by7 by Molmil
HUMAN PLASMINOGEN ACTIVATOR INHIBITOR-2. LOOP (66-98) DELETION MUTANT
Descriptor: PROTEIN (PLASMINOGEN ACTIVATOR INHIBITOR-2)
Authors:Harrop, S.J, King, G.C, Mabbutt, B.C, Curmi, P.M.G.
Deposit date:1998-10-27
Release date:1999-10-24
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2 Å)
Cite:The crystal structure of plasminogen activator inhibitor 2 at 2.0 A resolution: implications for serpin function.
Structure Fold.Des., 7, 1999
1B3K
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Plasminogen activator inhibitor-1
Descriptor: PLASMINOGEN ACTIVATOR INHIBITOR-1
Authors:Sharp, A.M, Stein, P.E, Pannu, N.S, Read, R.J.
Deposit date:1998-12-11
Release date:1999-12-11
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.99 Å)
Cite:The active conformation of plasminogen activator inhibitor 1, a target for drugs to control fibrinolysis and cell adhesion.
Structure Fold.Des., 7, 1999
9PAI
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BU of 9pai by Molmil
CLEAVED SUBSTRATE VARIANT OF PLASMINOGEN ACTIVATOR INHIBITOR-1
Descriptor: PROTEIN (PLASMINOGEN ACTIVATOR INHIBITOR-1) residues 19-364, PROTEIN (PLASMINOGEN ACTIVATOR INHIBITOR-1) residues 365-397
Authors:Aertgeerts, K, De Bondt, H.L, De Ranter, C.J, Declerck, P.J.
Deposit date:1999-03-11
Release date:1999-03-19
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Mechanisms contributing to the conformational and functional flexibility of plasminogen activator inhibitor-1.
Nat.Struct.Biol., 2, 1995
1QLP
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2.0 ANGSTROM STRUCTURE OF INTACT ALPHA-1-ANTITRYPSIN: A CANONICAL TEMPLATE FOR ACTIVE SERPINS
Descriptor: ALPHA-1-ANTITRYPSIN
Authors:Elliott, P.R, Pei, X.Y, Dafforn, T, Read, R.J, Carrell, R.W, Lomas, D.A.
Deposit date:1999-09-10
Release date:1999-09-27
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2 Å)
Cite:Topography of a 2.0 A structure of alpha1-antitrypsin reveals targets for rational drug design to prevent conformational disease.
Protein Sci., 9, 2000
1QMB
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Cleaved alpha-1-antitrypsin polymer
Descriptor: ALPHA-1-ANTITRYPSIN
Authors:Huntington, J.A, Pannu, N.S, Hazes, B, Read, R.J, Lomas, D.A, Carrell, R.W.
Deposit date:1999-09-24
Release date:2000-02-06
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:A 2.6A Structure of a Serpin Polymer and Implications for Conformational Disease
J.Mol.Biol., 293, 1999

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