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5I2R

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C2(=NN(c1cccc(c1)OC(F)(F)F)C=CC2=O)c3ccnn3c4ccccc4, micromolar IC50=0.019462

Resources
File formatFile name (file size)
PDBx/mmCIF5i2r.cif.gz Display(273.22 KB)
5i2r.cif
PDBx/mmJSONall5i2r.json.gz Display (Tree)(168.64 KB)
5i2r.json
no-atom5i2r-noatom.json.gz Display (Header)(19.82 KB)
5i2r-noatom.json
add only5i2r-plus.json.gz Display(1.18 KB)
5i2r-plus.json
PDBMLall5i2r.xml.gz Display(370.83 KB)
5i2r.xml
no-atom5i2r-noatom.xml.gz Display(52.38 KB)
5i2r-noatom.xml
ext-atom5i2r-extatom.xml.gz Display(242.23 KB)
5i2r-extatom.xml
pdb_nextgenallpdb_00005i2r_xyz-enrich.cif.gz Display(299.87 KB)
pdb_00005i2r_xyz-enrich.cif
no-atompdb_00005i2r_xyz-no-atom-enrich.xml.gz Display(67.36 KB)
pdb_00005i2r_xyz-no-atom-enrich.xml
ng-only5i2r-plus.json.gz Display(3.52 KB)
5i2r-plus.json
PDBpdb5i2r.ent.gz Display(221.46 KB)
pdb5i2r.ent
RDF5i2r.rdf.gz Visualize(143.21 KB)
5i2r.rdf
Structure factorsr5i2rsf.ent.gz Display(2.26 MB)
r5i2rsf.ent
Biological unit (mmCIF format)5i2r-assembly1.cif.gz Display(71.22 KB)
5i2r-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5i2r-assembly2.cif.gz Display(72.09 KB)
5i2r-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5i2r-assembly3.cif.gz Display(71.97 KB)
5i2r-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5i2r-assembly4.cif.gz Display(69.03 KB)
5i2r-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5i2r.pdb1.gz Display(56.88 KB)
5i2r.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5i2r.pdb2.gz Display(57.75 KB)
5i2r.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5i2r.pdb3.gz Display(57.55 KB)
5i2r.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5i2r.pdb4.gz Display(55.46 KB)
5i2r.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5i2r_validation.pdf.gz Display(1.61 MB)
5i2r_validation.pdf
PDF-full5i2r_full_validation.pdf.gz Display(1.62 MB)
5i2r_full_validation.pdf
mmCIF5i2r_validation.cif.gz Display(77.31 KB)
5i2r_validation.cif
XML5i2r_validation.xml.gz Display(59.40 KB)
5i2r_validation.xml
PNG5i2r_multipercentile_validation.png.gz Display(169.26 KB)
5i2r_multipercentile_validation.png
SVG5i2r_multipercentile_validation.svg.gz Display(960.00 B)
5i2r_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5i2r_validation_2fo-fc_map_coef.cif.gz Display(834.08 KB)
5i2r_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5i2r_validation_fo-fc_map_coef.cif.gz Display(836.63 KB)
5i2r_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5i2r_validation_2fo-fc_map_coef.mtz Visualize(1.28 MB)
fo-fc (MTZ)5i2r_validation_fo-fc_map_coef.mtz Visualize(1.28 MB)

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PDB entries from 2026-01-14

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