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8V9C

HIV-1 Integrase F185H Complexed with Allosteric Inhibitor GSK1264

Replaces:  5HOT
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues82
DetailsZN_FING: Integrase-type => ECO:0000255|PROSITE-ProRule:PRU00450
ChainResidueDetails
AASP3-GLN44
BASP3-GLN44

site_idSWS_FT_FI2
Number of Residues94
DetailsDNA_BIND: Integrase-type => ECO:0000255|PROSITE-ProRule:PRU00506
ChainResidueDetails
APHE223-ASP270
BPHE223-ASP270

site_idSWS_FT_FI3
Number of Residues8
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00450
ChainResidueDetails
AHIS12
AHIS16
ACYS40
ACYS43
BHIS12
BHIS16
BCYS40
BCYS43

site_idSWS_FT_FI4
Number of Residues4
DetailsBINDING:
ChainResidueDetails
AASP64
AASP116
BASP64
BASP116

site_idSWS_FT_FI5
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152
BGLU152

237735

PDB entries from 2025-06-18

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