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7L9A

Crystal structure of BRDT bromodomain 2 in complex with CDD-1102

Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue XWP A 401
ChainResidue
AVAL298
AASN351
APRO352
AHIS355
AHOH512
BTRP292
BTYR295
BASN296
ALEU303
ALEU305
AHIS306
ATYR308
AVAL311
AASN346
ACYS347
ATYR350

site_idAC2
Number of Residues5
Detailsbinding site for residue BME A 402
ChainResidue
AVAL312
ALYS313
AASN314
AASN346
ALYS349

site_idAC3
Number of Residues21
Detailsbinding site for residue XWP B 401
ChainResidue
ATYR348
ALYS349
AARG362
AGLN365
BLYS285
BTRP292
BPRO293
BVAL298
BLEU303
BLEU305
BHIS306
BTYR308
BVAL311
BASN346
BCYS347
BTYR350
BASN351
BPRO352
BHIS355
BHOH504
BHOH516

site_idAC4
Number of Residues6
Detailsbinding site for residue BME B 402
ChainResidue
BTRP292
BPRO293
BTYR295
BASN296
BPRO297
BASP299

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFynpvDvnalglhNYYdvVknpMdlgtIkekmdnqe..Ykdaykfaadvrl.MfmNCykY
ChainResidueDetails
AALA291-TYR350

219869

PDB entries from 2024-05-15

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