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7KDZ

Crystal structure of the bromodomain (BD) of human Bromodomain and PHD finger-containing Transcription Factor (BPTF) bound to TP-238

Functional Information from GO Data
ChainGOidnamespacecontents
A0006357biological_processregulation of transcription by RNA polymerase II
A0016589cellular_componentNURF complex
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue EDO A 3101
ChainResidue
ATYR2965
AHOH3201
AHOH3217

site_idAC2
Number of Residues14
Detailsbinding site for residue WCS A 3102
ChainResidue
ACYS3003
ATYR3006
AASN3007
APRO3012
APHE3013
APHE3013
AHOH3203
AHOH3274
ATRP2950
APRO2951
APHE2952
AVAL2956
AASP2957
AASP2960

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFlepvDpndap..DYYgvIkepMdlatMeervqrry..Yekltefvadmtk.IfdNCryY
ChainResidueDetails
AALA2949-TYR3006

223532

PDB entries from 2024-08-07

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