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6ZC8

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

Functional Information from GO Data
ChainGOidnamespacecontents
A0016055biological_processWnt signaling pathway
B0016055biological_processWnt signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue QEK A 401
ChainResidue
APHE259
ALEU260
AGLY261
AILE262
AILE262
AMET282
AARG320
AVAL323
AHIS324

site_idAC2
Number of Residues12
Detailsbinding site for residue QEK B 401
ChainResidue
BPHE259
BLEU260
BGLY261
BILE262
BSER263
BILE264
BMET282
BLEU319
BARG320
BVAL323
BHIS324
BHOH505

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsModified residue: {"description":"Symmetric dimethylarginine; by PRMT7; alternate","evidences":[{"source":"PubMed","id":"23150776","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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