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6DBC

Second bromodomain of Human BRD2 with a Tetrahydroquinoline analogue

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue EDO A 501
ChainResidue
ALEU350
AHOH604
AHOH611
AHOH687

site_idAC2
Number of Residues7
Detailsbinding site for residue EDO A 502
ChainResidue
ALYS427
AASP455
AILE389
AILE390
ALYS391
AHIS392
AASN424

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 503
ChainResidue
ATYR368
ALYS402
AASP407
AGLU413
AMET438
ALYS441
AHOH672

site_idAC4
Number of Residues7
Detailsbinding site for residue EDO A 504
ChainResidue
ATYR426
AARG440
AGLN443
AGLN443
AASP444
APHE448
AHOH629

site_idAC5
Number of Residues3
Detailsbinding site for residue EDO A 505
ChainResidue
AHIS433
AASP434
AG3J508

site_idAC6
Number of Residues6
Detailsbinding site for residue EDO A 506
ChainResidue
ALEU361
ATYR373
AHOH650
AHOH653
AHOH668
AHOH689

site_idAC7
Number of Residues3
Detailsbinding site for residue EDO A 507
ChainResidue
ALEU381
AG3J508
AHOH655

site_idAC8
Number of Residues10
Detailsbinding site for residue G3J A 508
ChainResidue
ATRP370
APRO371
ALEU383
AASN429
AHIS433
AVAL435
AEDO505
AEDO507
AHOH609
AHOH655

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

218500

PDB entries from 2024-04-17

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