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5MWG

Crystal structure of the human BRPF1 bromodomain in complex with BZ091

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue WGX A 801
ChainResidue
AILE652
APHE714
AHOH912
AHOH917
BLYS639
APHE653
AVAL657
APRO658
AGLU661
AVAL662
ACYS704
ATYR707
AASN708

site_idAC2
Number of Residues5
Detailsbinding site for residue NO3 A 802
ChainResidue
ALEU630
ATHR631
ALEU634
AILE635
AARG638

site_idAC3
Number of Residues13
Detailsbinding site for residue WGX B 801
ChainResidue
ALYS639
AHOH927
BILE652
BPHE653
BVAL657
BPRO658
BGLU661
BCYS704
BTYR707
BASN708
BILE713
BPHE714
BHOH935

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

250835

PDB entries from 2026-03-18

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