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5HJS

Identification of LXRbeta selective agonists for the treatment of Alzheimer's Disease

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006629biological_processlipid metabolic process
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 668 A 301
ChainResidue
APHE93
ALEU152
ALEU167
APHE171
AHIS257
AGLN260
ALEU264
ALEU271
ATRP279
ATHR94
ALEU96
AALA97
AGLU103
AMET134
ATHR138
AARG141
APHE151

site_idAC2
Number of Residues16
Detailsbinding site for residue 668 B 301
ChainResidue
BPHE90
BTHR94
BLEU96
BGLU103
BILE131
BMET134
BTHR138
BARG141
BPHE151
BLEU152
BLEU167
BHIS257
BGLN260
BLEU264
BLEU271
BTRP279

site_idAC3
Number of Residues8
Detailsbinding site for residue SO4 C 101
ChainResidue
AARG119
AARG119
CHIS6
CHIS6
CGLN10
CGLN10
CHOH202
CHOH202

site_idAC4
Number of Residues8
Detailsbinding site for residue SO4 D 101
ChainResidue
BARG119
BARG119
DHIS6
DHIS6
DGLN10
DGLN10
DHOH201
DHOH201

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
CSER13
DSER13

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PDB entries from 2024-07-24

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