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4E2J

X-Ray Crystal Structure of the Ancestral Glucocorticoid Receptor 2 ligand binding domain in complex with mometasone furoate and TIF-2 coactivator fragment

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 301
ChainResidue
AGLY37
AARG38
APRO219
AGLU220
AMET221
AHOH424
ETYR747

site_idAC2
Number of Residues13
DetailsBINDING SITE FOR RESIDUE MOF A 302
ChainResidue
AGLY36
AGLN39
AARG80
APHE92
AMET108
AGLN111
AMET115
APHE204
ACYS205
ATHR208
APHE218
ALEU32
AASN33

site_idAC3
Number of Residues12
DetailsBINDING SITE FOR RESIDUE MOF B 301
ChainResidue
BMET29
BLEU32
BASN33
BGLY36
BGLN39
BARG80
BPHE92
BMET108
BMET115
BPHE204
BCYS205
BTHR208

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE FMT B 302
ChainResidue
BTYR67
BSER68
BTRP69
BMET70
BSER71
BLEU202

site_idAC5
Number of Residues1
DetailsBINDING SITE FOR RESIDUE GOL B 303
ChainResidue
AARG54

221716

PDB entries from 2024-06-26

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