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3MJR

Human dCK complex with Acyclic Nucleoside

Functional Information from GO Data
ChainGOidnamespacecontents
A0000166molecular_functionnucleotide binding
A0004136molecular_functiondeoxyadenosine kinase activity
A0004137molecular_functiondeoxycytidine kinase activity
A0004138molecular_functiondeoxyguanosine kinase activity
A0005524molecular_functionATP binding
A0005634cellular_componentnucleus
A0005654cellular_componentnucleoplasm
A0005737cellular_componentcytoplasm
A0005739cellular_componentmitochondrion
A0005829cellular_componentcytosol
A0006139biological_processnucleobase-containing compound metabolic process
A0006220biological_processpyrimidine nucleotide metabolic process
A0008144molecular_functionobsolete drug binding
A0009224biological_processCMP biosynthetic process
A0016301molecular_functionkinase activity
A0016310biological_processphosphorylation
A0016740molecular_functiontransferase activity
A0019136molecular_functiondeoxynucleoside kinase activity
A0042803molecular_functionprotein homodimerization activity
A0043771molecular_functioncytidine kinase activity
A0106383biological_processdAMP salvage
A1901135biological_processcarbohydrate derivative metabolic process
A1901293biological_processnucleoside phosphate biosynthetic process
B0000166molecular_functionnucleotide binding
B0004136molecular_functiondeoxyadenosine kinase activity
B0004137molecular_functiondeoxycytidine kinase activity
B0004138molecular_functiondeoxyguanosine kinase activity
B0005524molecular_functionATP binding
B0005634cellular_componentnucleus
B0005654cellular_componentnucleoplasm
B0005737cellular_componentcytoplasm
B0005739cellular_componentmitochondrion
B0005829cellular_componentcytosol
B0006139biological_processnucleobase-containing compound metabolic process
B0006220biological_processpyrimidine nucleotide metabolic process
B0008144molecular_functionobsolete drug binding
B0009224biological_processCMP biosynthetic process
B0016301molecular_functionkinase activity
B0016310biological_processphosphorylation
B0016740molecular_functiontransferase activity
B0019136molecular_functiondeoxynucleoside kinase activity
B0042803molecular_functionprotein homodimerization activity
B0043771molecular_functioncytidine kinase activity
B0106383biological_processdAMP salvage
B1901135biological_processcarbohydrate derivative metabolic process
B1901293biological_processnucleoside phosphate biosynthetic process
C0000166molecular_functionnucleotide binding
C0004136molecular_functiondeoxyadenosine kinase activity
C0004137molecular_functiondeoxycytidine kinase activity
C0004138molecular_functiondeoxyguanosine kinase activity
C0005524molecular_functionATP binding
C0005634cellular_componentnucleus
C0005654cellular_componentnucleoplasm
C0005737cellular_componentcytoplasm
C0005739cellular_componentmitochondrion
C0005829cellular_componentcytosol
C0006139biological_processnucleobase-containing compound metabolic process
C0006220biological_processpyrimidine nucleotide metabolic process
C0008144molecular_functionobsolete drug binding
C0009224biological_processCMP biosynthetic process
C0016301molecular_functionkinase activity
C0016310biological_processphosphorylation
C0016740molecular_functiontransferase activity
C0019136molecular_functiondeoxynucleoside kinase activity
C0042803molecular_functionprotein homodimerization activity
C0043771molecular_functioncytidine kinase activity
C0106383biological_processdAMP salvage
C1901135biological_processcarbohydrate derivative metabolic process
C1901293biological_processnucleoside phosphate biosynthetic process
D0000166molecular_functionnucleotide binding
D0004136molecular_functiondeoxyadenosine kinase activity
D0004137molecular_functiondeoxycytidine kinase activity
D0004138molecular_functiondeoxyguanosine kinase activity
D0005524molecular_functionATP binding
D0005634cellular_componentnucleus
D0005654cellular_componentnucleoplasm
D0005737cellular_componentcytoplasm
D0005739cellular_componentmitochondrion
D0005829cellular_componentcytosol
D0006139biological_processnucleobase-containing compound metabolic process
D0006220biological_processpyrimidine nucleotide metabolic process
D0008144molecular_functionobsolete drug binding
D0009224biological_processCMP biosynthetic process
D0016301molecular_functionkinase activity
D0016310biological_processphosphorylation
D0016740molecular_functiontransferase activity
D0019136molecular_functiondeoxynucleoside kinase activity
D0042803molecular_functionprotein homodimerization activity
D0043771molecular_functioncytidine kinase activity
D0106383biological_processdAMP salvage
D1901135biological_processcarbohydrate derivative metabolic process
D1901293biological_processnucleoside phosphate biosynthetic process
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE AC2 A 301
ChainResidue
AILE30
AGLU53
APHE96
AGLN97
AARG128
AASP133
APHE137
ATYR204

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE UDP A 261
ChainResidue
AALA32
AGLY33
ALYS34
ASER35
ATHR36
AGLU127
AARG188
AARG192
AASP241
APHE242
ALYS243
AALA31

site_idAC3
Number of Residues9
DetailsBINDING SITE FOR RESIDUE AC2 B 401
ChainResidue
BGLU53
BVAL55
BPHE96
BGLN97
BARG104
BARG128
BASP133
BPHE137
BHOH275

site_idAC4
Number of Residues11
DetailsBINDING SITE FOR RESIDUE UDP B 261
ChainResidue
BALA31
BALA32
BGLY33
BLYS34
BSER35
BTHR36
BARG188
BLEU191
BARG192
BASP241
BPHE242

site_idAC5
Number of Residues12
DetailsBINDING SITE FOR RESIDUE UDP C 501
ChainResidue
CALA31
CGLY33
CLYS34
CSER35
CTHR36
CGLU127
CARG188
CLEU191
CARG192
CASP241
CPHE242
CLYS243

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE AC2 D 601
ChainResidue
DGLU53
DTYR86
DGLN97
DARG104
DARG128
DASP133
DPHE137

site_idAC7
Number of Residues11
DetailsBINDING SITE FOR RESIDUE UDP D 261
ChainResidue
DALA31
DALA32
DGLY33
DLYS34
DSER35
DTHR36
DARG188
DLEU191
DARG192
DASP241
DPHE242

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsACT_SITE: Proton acceptor => ECO:0000255
ChainResidueDetails
AGLU127
BGLU127
CGLU127
DGLU127

site_idSWS_FT_FI2
Number of Residues36
DetailsBINDING:
ChainResidueDetails
AGLY28
BGLY28
BGLU53
BTYR86
BGLN97
BARG128
BASP133
BARG188
BGLU197
BGLU240
CGLY28
AGLU53
CGLU53
CTYR86
CGLN97
CARG128
CASP133
CARG188
CGLU197
CGLU240
DGLY28
DGLU53
ATYR86
DTYR86
DGLN97
DARG128
DASP133
DARG188
DGLU197
DGLU240
AGLN97
AARG128
AASP133
AARG188
AGLU197
AGLU240

site_idSWS_FT_FI3
Number of Residues8
DetailsMOD_RES: Phosphoserine; by CK1 => ECO:0000305|PubMed:20637175
ChainResidueDetails
ASER11
ASER15
BSER11
BSER15
CSER11
CSER15
DSER11
DSER15

site_idSWS_FT_FI4
Number of Residues4
DetailsMOD_RES: Phosphothreonine; by CK1 => ECO:0000305|PubMed:20637175
ChainResidueDetails
ATHR72
BTHR72
CTHR72
DTHR72

site_idSWS_FT_FI5
Number of Residues4
DetailsMOD_RES: Phosphoserine => ECO:0000269|PubMed:20637175, ECO:0007744|PubMed:18669648, ECO:0007744|PubMed:20068231, ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER74
BSER74
CSER74
DSER74

218853

PDB entries from 2024-04-24

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